Issue 39, 2014

NIS-mediated regioselective amidation of indole with quinazolinone and pyrimidone

Abstract

A mild, metal-free condition was developed for the direct regioselective C2 amidation of indoles and pyrroles with quinazolinone and pyrimidone derivatives in intermolecular fashion, which led to novel indolyl/pyrrolyl quinazolinone and pyrimidone derivatives in moderate to good yields.

Graphical abstract: NIS-mediated regioselective amidation of indole with quinazolinone and pyrimidone

Supplementary files

Article information

Article type
Paper
Submitted
31 Jan 2014
Accepted
03 Apr 2014
First published
04 Apr 2014

RSC Adv., 2014,4, 20136-20144

Author version available

NIS-mediated regioselective amidation of indole with quinazolinone and pyrimidone

S. K. Ghosh and R. Nagarajan, RSC Adv., 2014, 4, 20136 DOI: 10.1039/C4RA02417F

To request permission to reproduce material from this article, please go to the Copyright Clearance Center request page.

If you are an author contributing to an RSC publication, you do not need to request permission provided correct acknowledgement is given.

If you are the author of this article, you do not need to request permission to reproduce figures and diagrams provided correct acknowledgement is given. If you want to reproduce the whole article in a third-party publication (excluding your thesis/dissertation for which permission is not required) please go to the Copyright Clearance Center request page.

Read more about how to correctly acknowledge RSC content.

Social activity

Spotlight

Advertisements