Issue 38, 2014
From the journal:

Organic & Biomolecular Chemistry

Palladium-catalyzed ortho-acylation of 2-benzyl-1,2,3-triazoles with aldehydes†

Qingshan Tian,a   Ping Hea  and  Chunxiang Kuang*ab  

* Corresponding authors

a Department of Chemistry, Tongji University, Siping Road 1239, Shanghai 200092, P. R. China

b Key Laboratory of Yangtze River Water Environment, Ministry of Education, Siping Road 1239, Shanghai 200092, P. R. China
E-mail: kuangcx@tongji.edu.cn

Abstract

A palladium-catalyzed ortho-acylation of 2-benzyl-1,2,3-triazoles with aldehydes as an acyl source was developed. A wide variety of ketones containing 1,2,3-triazoles were obtained in good to excellent yields. This methodology provides a convenient access to the acylation of 2-substituted-1,2,3-triazoles.

Graphical abstract: Palladium-catalyzed ortho-acylation of 2-benzyl-1,2,3-triazoles with aldehydes

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Article information

DOI
https://doi.org/10.1039/C4OB01406E
Article type
Communication
Submitted
07 Jul 2014
Accepted
12 Aug 2014
First published
13 Aug 2014

Org. Biomol. Chem., 2014,12, 7474-7477

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Palladium-catalyzed ortho-acylation of 2-benzyl-1,2,3-triazoles with aldehydes

Q. Tian, P. He and C. Kuang, Org. Biomol. Chem., 2014, 12, 7474 DOI: 10.1039/C4OB01406E

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