Issue 5, 2014
From the journal:

Organic & Biomolecular Chemistry

Synthesis of substituted indenones and indanones by a Suzuki–Miyaura coupling/acid-promoted cyclisation sequence†

Alexey N. Butkevich,a   Beatrice Ranieri,a   Lieven Meerpoel,b   Ian Stansfield,c   Patrick Angibaud,c   Andrei Corbua  and  Janine Cossy*a  

* Corresponding authors

a Laboratoire de Chimie Organique, ESPCI ParisTech, CNRS, 10 rue Vauquelin, 75231 Paris Cedex 05, France
E-mail: Janine.cossy@espci.fr

b Janssen Research & Development, Division of Janssen Pharmaceutica NV, Turnhoutsweg 30, 2340 Beerse, Belgium

c Janssen Research & Development, Division of Janssen-Cilag, Oncology and Medicinal Chemistry, Campus de Maigremont, 27106 Val de Reuil, Cedex, France

Abstract

A one-pot Suzuki–Miyaura cross-coupling/acid-catalyzed cyclisation leading to indenones and indanones in modest to good yields is reported.

Graphical abstract: Synthesis of substituted indenones and indanones by a Suzuki–Miyaura coupling/acid-promoted cyclisation sequence

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Article information

DOI
https://doi.org/10.1039/C3OB41974F
Article type
Communication
Submitted
30 Sep 2013
Accepted
18 Nov 2013
First published
19 Nov 2013

Org. Biomol. Chem., 2014,12, 728-731

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Synthesis of substituted indenones and indanones by a Suzuki–Miyaura coupling/acid-promoted cyclisation sequence

A. N. Butkevich, B. Ranieri, L. Meerpoel, I. Stansfield, P. Angibaud, A. Corbu and J. Cossy, Org. Biomol. Chem., 2014, 12, 728 DOI: 10.1039/C3OB41974F

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