Maxim Frizler, Ilia V. Yampolsky, Mikhail S. Baranov, Marit Stirnberg and Michael Gütschow
Org. Biomol. Chem., 2013,11, 5913-5921
DOI:
10.1039/C3OB41341A,
Paper
An activity-based probe, containing an irreversibly locked GFP-like fluorophore, was synthesized and evaluated as an inhibitor of human cathepsins and, as exemplified with cathepsin K, it proved to be suitable for ex vivo imaging and quantification of cysteine cathepsins by SDS-PAGE.
