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Issue 37, 2013
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Pd(0)-catalyzed benzylic arylation–oxidation of 4-methylquinazolines via sp3 C–H activation under air conditions

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Abstract

An efficient and selective Pd(0)-catalyzed sp3 C–H bond arylation–oxidation of 4-methylquinazolines is reported. The method enables the introduction of arylketone at the benzylic position of 4-methylquinazolines without the use of an additional directing group, and atmospheric oxygen is used as the sole oxidant.

Graphical abstract: Pd(0)-catalyzed benzylic arylation–oxidation of 4-methylquinazolines via sp3 C–H activation under air conditions

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Supplementary files

Article information


Submitted
19 Jul 2013
Accepted
01 Aug 2013
First published
02 Aug 2013

Org. Biomol. Chem., 2013,11, 6246-6249
Article type
Communication

Pd(0)-catalyzed benzylic arylation–oxidation of 4-methylquinazolines via sp3 C–H activation under air conditions

D. Zhao, M. Zhu, Y. Wang, Q. Shen and J. Li, Org. Biomol. Chem., 2013, 11, 6246
DOI: 10.1039/C3OB41488D

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