Issue 8, 2012
From the journal:

RSC Advances

Synthesis of 2-amino-imidazoles, purines, and benzoxazolamines through DIB oxidation†

Jean-Christophe Andrez*a  

* Corresponding authors

a Cardiome Pharma Corp, 6190 Agronomy Rd., 6th Floor, Vancouver, British Columbia, Canada
E-mail: jandrez@cardiome.com
Tel: 604-677-6905 (ext112)

Abstract

A wide range of fused 2-amino-imidazoles and 2-amino-benzoxazoles can be prepared in one-pot under very mild conditions from 1,2-diamino-arenes or 2-amino-phenols and Vilsmeier reagents. The oxidation proceeds using diacetoxy-iodobenzene (DIB) and is tolerant to different functionalities.

Graphical abstract: Synthesis of 2-amino-imidazoles, purines, and benzoxazolamines through DIB oxidation

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Article information

DOI
https://doi.org/10.1039/C2RA20101A
Article type
Communication
Submitted
17 Jan 2012
Accepted
22 Feb 2012
First published
24 Feb 2012

RSC Adv., 2012,2, 3261-3264

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Synthesis of 2-amino-imidazoles, purines, and benzoxazolamines through DIB oxidation

J. Andrez, RSC Adv., 2012, 2, 3261 DOI: 10.1039/C2RA20101A

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