Issue 3, 2003
From the journal:

Organic & Biomolecular Chemistry

First synthesis of 2′,3′-epimino-carbocyclic nucleosides

Minoru Ishikura,*a   Atsushi Murakamia  and  Nobuya Katagiria  

* Corresponding authors

a Faculty of Pharmaceutical Sciences, Health Sciences University of Hokkaido, Ishikari-Tobetsu, Hokkaido 061-0293, Japan
E-mail: ishikura@hoku-iryo-u.ac.jp
Fax: (+81)-(0)1332-3-1245

Abstract

The preparation of 2′,3′-epimino-carbocyclic analogues of adenosine is reported. The reaction of p-tosyl azide with N-substituted 2-azabicyclo[2.2.1]hept-5-en-3-one (ABH) (1a) provided aziridine-fused ABH (2), which was converted to 2′,3′-epimino-carbocyclic nucleosides (11).

Graphical abstract: First synthesis of 2′,3′-epimino-carbocyclic nucleosides

About
Cited by
Related
Download options Please wait...

Article information

DOI
https://doi.org/10.1039/B210963H
Article type
Communication
Submitted
07 Nov 2002
Accepted
16 Dec 2002
First published
07 Jan 2003

Org. Biomol. Chem., 2003,1, 452-453

Permissions

Request permissions

First synthesis of 2′,3′-epimino-carbocyclic nucleosides

M. Ishikura, A. Murakami and N. Katagiri, Org. Biomol. Chem., 2003, 1, 452 DOI: 10.1039/B210963H

To request permission to reproduce material from this article, please go to the Copyright Clearance Center request page.

If you are an author contributing to an RSC publication, you do not need to request permission provided correct acknowledgement is given.

If you are the author of this article, you do not need to request permission to reproduce figures and diagrams provided correct acknowledgement is given. If you want to reproduce the whole article in a third-party publication (excluding your thesis/dissertation for which permission is not required) please go to the Copyright Clearance Center request page.

Read more about how to correctly acknowledge RSC content.

Social activity

Spotlight

Advertisements