Kazuyuki Miyashita, Hiroshi Iwaki, Kuninori Tai, Hidenobu Murafuji and Takeshi Imanishi
Chem. Commun., 1998, 1987-1988
DOI:
10.1039/A805596C,
Paper
Stereoselective and N-terminal selective α-alkylation of peptides is achieved using a pyridoxal model compound as an N-terminal activator which also functions as a chiral auxiliary.