The title compound 4, prepared by lead tetraacetate oxidation of 5, is stable at room temperature and aziridinates alkenes in better yield and higher diastereoselectivity than, e.g. the 2-ethyl compound 1; hydrazinolysis of the quinazolinone ring in 20 gives the corresponding N-aminoaziridine 21 in 64% yield.
R. S. Atkinson, M. P. Coogan and C. L. Cornell, J. Chem. Soc., Chem. Commun., 1993, 1215 DOI: 10.1039/C39930001215
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