The preparation of 1,3-amino alcohols by the reduction of azetidin-2-ones with diborane is described. New methods for the cyclisation of the aminopropanols to the corresponding azetidines are reported; these methods centre on the use of a modified Mitsunobu reaction.
P. G. Sammes and S. Smith, J. Chem. Soc., Perkin Trans. 1, 1984, 2415 DOI: 10.1039/P19840002415
To request permission to reproduce material from this article, please go to the Copyright Clearance Center request page.
If you are an author contributing to an RSC publication, you do not need to request permission provided correct acknowledgement is given.
If you are the author of this article, you do not need to request permission to reproduce figures and diagrams provided correct acknowledgement is given. If you want to reproduce the whole article in a third-party publication (excluding your thesis/dissertation for which permission is not required) please go to the Copyright Clearance Center request page.
Read more about how to correctly acknowledge RSC content.
Please wait while we load your content...