This website uses cookies to give you the best user experience. If you continue without changing your settings we'll assume you are happy to receive all RSC cookies. You can change your cookie settings by navigating to our Privacy and Cookies page and following the instructions. These instructions are also obtainable from the privacy link at the bottom of any RSC page.
Lite Version|Standard version
Home > Organic & Biomolecular ... >
To gain access to this content please
Log in via your home Institution.
Log in with your member or subscriber username and password.
Download


Buy PDF Add PDF to Basket (£42.50*)
*Exclusive of taxes
This article contains 5 page(s)
Abstract | Cited by

A simple and efficient transition-metal-free oxidative halogenation (Cl, Br) of the C5 C–H bond of 8-aminoquinoline amides has been developed. This method employed low-cost and innoxious sodium halides as halogenation reagents and oxone as an oxidant. The reactions demonstrated air and moisture tolerance, and good functional group compatibility, giving highly selective C5-halogenated products in good to excellent yields.

Graphical abstract: Transition-metal-free oxidative C5 C–H-halogenation of 8-aminoquinoline amides using sodium halides

Page: ^ Top


Enter Keywords, author, title,reference, or DOI
Log in | Register