Cycloaddition Reaction: Synthesis of 5-Substituted 1,3,4-Thiadiazolo[3,2-a]pyrimidin-6-one

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B. C. Dutta, K. K. Das and B. N. Goswami


Abstract

1,3,4-Thiadiazolo[3,2-a]pyrimidin-6-ones are synthesised by a (4+2) cycloaddition reaction of arylidineamino-1,3,4-thiadiazole and aryl ketenes formed in situ.


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