DOI: 10.1039/A800452H
(Paper)
Reference Section for: J. Chem. Res. (S), 1998, 430-431
Convenient Synthesis of 2,6-di-tert-Butyl-4-[5-(3-pyridyl)-4-oxapentyl]phenols and their thia-Analogues
(Note: The full text of this document is currently only available in the PDF Version )
Osvalds Pugovičs, Valerjans Kauss, Ivars Kalvinsh, Markus R. Gold and Günther Quack
Abstract
A convenient large scale procedure for the synthesis of Nicanartine {2,6-di-tert-butyl-4-[5-(3-pyridyl)-4-oxapentyl]phenol}, an antiatherosclerotic compound has been developed, the synthetic route towards the thia-analogue as well as various branched-chain oxa- and thia-derivatives of the parent compound has also been investigated.
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