DOI: 10.1039/A801030G
(Paper)
Reference Section for: Chem. Commun., 1998, 1171-1172
Binding of D-serine-terminating cell-wall analogues to glycopeptide antibiotics
(Note: The full text of this document is currently only available in the PDF Version )
André M. A. van Wageningen, Thomas Staroske and Dudley H. Williams
Abstract
Binding studies of –L-Lys-D-Ala-D-Ser-terminating ligands, used as model systems for cell-wall precursors found in VanC resistant bacteria, with vancomycin, chloroeremomycin and teicoplanin show that they bind to these glycopeptides in a similar manner as –L-Lys-D-Ala-D-Ala-terminating ligands, but that the binding constants are one to two orders of magnitude lower.
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