Issue 25, 2016

Palladium-catalyzed decarboxylative ortho-aroylation of N-acetyl-1,2,3,4-tetrahydroquinolines with α-oxoarylacetic acids

Abstract

A mild, practical and efficient palladium-catalyzed decarboxylative ortho-aroylation of N-acetyl-1,2,3,4-tetrahydroquinolines with α-oxoarylacetic acids via C–H bond activation is described. This protocol provides efficient access to a series of C8-aroyl terahydroquinolines.

Graphical abstract: Palladium-catalyzed decarboxylative ortho-aroylation of N-acetyl-1,2,3,4-tetrahydroquinolines with α-oxoarylacetic acids

Supplementary files

Article information

Article type
Paper
Submitted
04 Jan 2016
Accepted
05 Feb 2016
First published
08 Feb 2016

RSC Adv., 2016,6, 20637-20643

Author version available

Palladium-catalyzed decarboxylative ortho-aroylation of N-acetyl-1,2,3,4-tetrahydroquinolines with α-oxoarylacetic acids

L. Han, Y. Wang, H. Song, H. Han, L. Wang, W. Chu and Z. Sun, RSC Adv., 2016, 6, 20637 DOI: 10.1039/C6RA00163G

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