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Issue 125, 2015
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Synthesis of isatins by the palladium-catalyzed intramolecular acylation of unactivated aryl C(sp2)–H bonds

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Abstract

Synthesis of isatins from formyl-N-arylformamides is achieved via PdCl2-catalyzed intramolecular acylation. This method shows the possibility of Pd-catalyzed aryl C(sp2)–H bond activation on the synthesis of isatins, affording an array of isatins in good yields. Yet this protocol is operationally simple and atom economical.

Graphical abstract: Synthesis of isatins by the palladium-catalyzed intramolecular acylation of unactivated aryl C(sp2)–H bonds

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Publication details

The article was received on 11 Nov 2015, accepted on 16 Nov 2015 and first published on 27 Nov 2015


Article type: Communication
DOI: 10.1039/C5RA23837D
Citation: RSC Adv., 2015,5, 103280-103283

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    Synthesis of isatins by the palladium-catalyzed intramolecular acylation of unactivated aryl C(sp2)–H bonds

    J. Li, Y. Zheng, X. Yu, S. Lv, Q. Wang, L. Hai and Y. Wu, RSC Adv., 2015, 5, 103280
    DOI: 10.1039/C5RA23837D

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