Palladacycle-catalyzed Suzuki–Miyaura reaction of aryl/heteroaryl halides with MIDA boronates in EtOH/H2O or H2O

Yabo Li; Jingran Wang; Zhiwei Wang; Mengmeng Huang; Beiqi Yan; Xiuling Cui; Yusheng Wu; Yangjie Wu

doi:10.1039/C4RA07486F

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Palladacycle-catalyzed Suzuki–Miyaura reaction of aryl/heteroaryl halides with MIDA boronates in EtOH/H₂O or H₂O†

Yabo Li,^a Jingran Wang,^a Zhiwei Wang,^a Mengmeng Huang,*^a Beiqi Yan,^a Xiuling Cui,^a Yusheng Wu*^ab and Yangjie Wu*^a

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* Corresponding authors

^a College of Chemistry and Molecular Engineering, Henan Key Laboratory of Chemical Biology and Organic Chemistry, Key Laboratory of Applied Chemistry of Henan Universities, Zhengzhou University, Zhengzhou, P. R. China
E-mail: wyj@zzu.edu.cn, hmm@zzu.edu.cn
Fax: +86-371-67767993

^b Tetranov Biopharm, LLC, 75 Daxue Road, Zhengzhou, P.R. China
E-mail: yusheng.wu@tetranovglobal.com

Abstract

With good to excellent yields, a series of mono- or diheteroaryl compounds were synthesized via the palladacycle-catalyzed Suzuki–Miyaura reaction of various N-methyliminodiacetic acid (MIDA) boronates with aryl/heteroaryl halides in EtOH/H₂O or H₂O.

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Article information

DOI: https://doi.org/10.1039/C4RA07486F
Article type: Paper
Submitted: 11 May 2014
Accepted: 06 Aug 2014
First published: 07 Aug 2014

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RSC Adv., 2014,4, 36262-36266

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Palladacycle-catalyzed Suzuki–Miyaura reaction of aryl/heteroaryl halides with MIDA boronates in EtOH/H₂O or H₂O

Y. Li, J. Wang, Z. Wang, M. Huang, B. Yan, X. Cui, Y. Wu and Y. Wu, RSC Adv., 2014, 4, 36262 DOI: 10.1039/C4RA07486F

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