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Issue 14, 2002
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Synthesis and biological evaluation of phospholane and dihydrophosphole analogues of the glutamate receptor agonist AP4

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Abstract

The syntheses and preliminary pharmacological characterisation of two novel cyclic phosphinic acid-containing amino acids designed as conformationally restricted analogues of the metabotropic glutamate receptor agonist AP4 (1) are reported.

Graphical abstract: Synthesis and biological evaluation of phospholane and dihydrophosphole analogues of the glutamate receptor agonist AP4

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Article information


Submitted
20 May 2002
Accepted
06 Jun 2002
First published
18 Jun 2002

J. Chem. Soc., Perkin Trans. 1, 2002, 1625-1627
Article type
Communication

Synthesis and biological evaluation of phospholane and dihydrophosphole analogues of the glutamate receptor agonist AP4

S. J. Conway, J. C. Miller, A. D. Bond, B. P. Clark and D. E. Jane, J. Chem. Soc., Perkin Trans. 1, 2002, 1625
DOI: 10.1039/B204891D

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