Jump to main content
Jump to site search

Issue 40, 2020
Previous Article Next Article

One-pot access to 2-amino-3-arylbenzofurans: direct entry to polyheterocyclic chemical space

Author affiliations

Abstract

As a means to make new benzofuran-embedded polycyclic structures, we established two efficient one-pot sequential coupling routes to 2-amino-3-arylbenzofurans and 2-amino-3-arylnaphtho[2,1-b]furans. Further ring formation (six- and seven-membered rings) with the resulting amine moiety at the C2 position of benzofurans was realized, leading to further expansion of benzofuran-based chemical space.

Graphical abstract: One-pot access to 2-amino-3-arylbenzofurans: direct entry to polyheterocyclic chemical space

Back to tab navigation

Supplementary files

Article information


Submitted
19 Aug 2020
Accepted
22 Sep 2020
First published
23 Sep 2020

Org. Biomol. Chem., 2020,18, 8119-8140
Article type
Paper

One-pot access to 2-amino-3-arylbenzofurans: direct entry to polyheterocyclic chemical space

S. S. Prasad, D. R. Joshi, J. H. Lee and I. Kim, Org. Biomol. Chem., 2020, 18, 8119
DOI: 10.1039/D0OB01715A

Social activity

Search articles by author

Spotlight

Advertisements