Issue 46, 2015

Regioselective synthesis of 2H-indazoles through Ga/Al- and Al-mediated direct alkylation reactions of indazoles

Abstract

A procedure has been developed for the regioselective, high yielding synthesis of 2H-indazoles that involves direct alkylation of indazoles with various allyl and benzyl bromides, and α-bromocarbonyl compounds.

Graphical abstract: Regioselective synthesis of 2H-indazoles through Ga/Al- and Al-mediated direct alkylation reactions of indazoles

Supplementary files

Article information

Article type
Paper
Submitted
20 Aug 2015
Accepted
29 Sep 2015
First published
29 Sep 2015

Org. Biomol. Chem., 2015,13, 11376-11381

Author version available

Regioselective synthesis of 2H-indazoles through Ga/Al- and Al-mediated direct alkylation reactions of indazoles

M. Lin, H. Liu, W. Lin, C. Kuo and T. Chuang, Org. Biomol. Chem., 2015, 13, 11376 DOI: 10.1039/C5OB01747E

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