Issue 48, 2014
From the journal:

Organic & Biomolecular Chemistry

A facile approach to spirocyclic 2-azido indolines via azidation of indoles with ceric ammonium nitrate†

Jing Li,a   Mao Liu,a   Qi Li,a   Hua Tiana  and  Yian Shi*abc  

* Corresponding authors

a Beijing National Laboratory for Molecular Sciences, CAS Key Laboratory of Molecular Recognition and Function, Institute of Chemistry, Chinese Academy of Sciences, Beijing 10090, China

b State Key Laboratory of Coordination Chemistry, Center for Multimolecular Organic Chemistry, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing 210093, China

c Department of Chemistry, Colorado State University, Fort Collins, Colorado 80523, USA
E-mail: yian@lamar.colostate.edu
Fax: +001-970-4911801
Tel: +001-970-4917424

Abstract

This paper describes azidation of indoles with NaN3 and ceric ammonium nitrate (CAN), giving a variety of spirocyclic 2-azido indolines in good yields and moderate diastereoselectivities.

Graphical abstract: A facile approach to spirocyclic 2-azido indolines via azidation of indoles with ceric ammonium nitrate

About
Cited by
Related
Download options Please wait...

Supplementary files

Article information

DOI
https://doi.org/10.1039/C4OB01549E
Article type
Communication
Submitted
22 Jul 2014
Accepted
01 Oct 2014
First published
30 Oct 2014

Org. Biomol. Chem., 2014,12, 9769-9772

Author version available

Download author version (PDF)

Permissions

Request permissions

A facile approach to spirocyclic 2-azido indolines via azidation of indoles with ceric ammonium nitrate

J. Li, M. Liu, Q. Li, H. Tian and Y. Shi, Org. Biomol. Chem., 2014, 12, 9769 DOI: 10.1039/C4OB01549E

To request permission to reproduce material from this article, please go to the Copyright Clearance Center request page.

If you are an author contributing to an RSC publication, you do not need to request permission provided correct acknowledgement is given.

If you are the author of this article, you do not need to request permission to reproduce figures and diagrams provided correct acknowledgement is given. If you want to reproduce the whole article in a third-party publication (excluding your thesis/dissertation for which permission is not required) please go to the Copyright Clearance Center request page.

Read more about how to correctly acknowledge RSC content.

Social activity

Spotlight

Advertisements