Issue 21, 2007

Stereocontrolled synthesis of substituted N-arenesulfonyl azetidines from γ-(phenylseleno)alkyl arylsulfonamides

Abstract

Different synthetic methodologies for the stereocontrolled synthesis of substituted azetidines are reported. The approach utilizes an optimized oxidation reaction of γ-(phenylseleno)alkyl arylsulfonamides, followed by the intramolecular substitution of the resulting phenylselenonyl group by the nitrogen atom.

Graphical abstract: Stereocontrolled synthesis of substituted N-arenesulfonyl azetidines from γ-(phenylseleno)alkyl arylsulfonamides

Article information

Article type
Paper
Submitted
21 Aug 2007
Accepted
05 Sep 2007
First published
21 Sep 2007

Org. Biomol. Chem., 2007,5, 3510-3519

Stereocontrolled synthesis of substituted N-arenesulfonyl azetidines from γ-(phenylseleno)alkyl arylsulfonamides

M. Tiecco, L. Testaferri, A. Temperini, R. Terlizzi, L. Bagnoli, F. Marini and C. Santi, Org. Biomol. Chem., 2007, 5, 3510 DOI: 10.1039/B712861D

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