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Issue 83, 2020
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Boronic acid-mediated ring-opening and Ni-catalyzed arylation of 1-arylcyclopropyl tosylates

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Abstract

Herein, we describe a protocol for the ring-opening arylation of 1-arylcyclopropyl tosylates, in which boronic acids promote ring-opening and a Ni catalyst facilitates arylation in high regioselectivity. A number of 2-arylated allyl derivatives are synthesized, which are relevant motifs found in biologically active molecules.

Graphical abstract: Boronic acid-mediated ring-opening and Ni-catalyzed arylation of 1-arylcyclopropyl tosylates

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Article information


Submitted
02 Sep 2020
Accepted
30 Sep 2020
First published
30 Sep 2020

Chem. Commun., 2020,56, 12538-12541
Article type
Communication

Boronic acid-mediated ring-opening and Ni-catalyzed arylation of 1-arylcyclopropyl tosylates

L. R. Mills, J. J. Monteith and S. A. L. Rousseaux, Chem. Commun., 2020, 56, 12538
DOI: 10.1039/D0CC05895E

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