Jump to main content
Jump to site search
PLANNED MAINTENANCE Close the message box

Scheduled maintenance work on Wednesday 22nd May 2019 from 11:00 AM to 1:00 PM (GMT).

During this time our website performance may be temporarily affected. We apologise for any inconvenience this might cause and thank you for your patience.


Issue 70, 2015
Previous Article Next Article

Diastereoselective synthesis of substituted diaziridines from simple ketones and aldehydes

Author affiliations

Abstract

Diastereopure substituted diaziridines from simple ketones, aldehydes and amines are here reported. These important chemical scaffolds are obtained in the presence of a weak inorganic base and hydroxylamine O-sulfonic acid (HOSA). This method introduces three stereocenters in one step to provide a wide variety of substituted diaziridines with high yields and diastereoselectivities.

Graphical abstract: Diastereoselective synthesis of substituted diaziridines from simple ketones and aldehydes

Back to tab navigation

Supplementary files

Publication details

The article was received on 11 Jun 2015, accepted on 20 Jul 2015 and first published on 21 Jul 2015


Article type: Communication
DOI: 10.1039/C5CC04813C
Author version
available:
Download author version (PDF)
Chem. Commun., 2015,51, 13511-13514

  •   Request permissions

    Diastereoselective synthesis of substituted diaziridines from simple ketones and aldehydes

    A. W. Beebe, E. F. Dohmeier and G. Moura-Letts, Chem. Commun., 2015, 51, 13511
    DOI: 10.1039/C5CC04813C

Search articles by author

Spotlight

Advertisements