Issue 15, 2002
From the journal:

Chemical Communications

Synthesis of the kappa-agonist CJ-15,161 via a palladium-catalyzed cross-coupling reaction

Arun Ghosh,*a   Janice E. Sieser,a   Stéphane Carona  and  Timothy J. N. Watsona  

* Corresponding authors

a Chemical Research and Development, Pfizer Global Research and Development, Eastern Point Road, P.O. Box 8013, Groton, CT, USA
E-mail: Arun_Ghosh@groton.pfizer.com

Abstract

Syntheses of CJ-15,161 (1) involving intermolecular N-arylation of an appropriately functionalized diamine, obtained from the precursor α-amino acids or, more conveniently, from the corresponding 1,2-amino alcohols via 1,2,3-oxathiazolidine-2,2-dioxide 22, are reported.

Graphical abstract: Synthesis of the kappa-agonist CJ-15,161 via a palladium-catalyzed cross-coupling reaction

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Article information

DOI
https://doi.org/10.1039/B204844B
Article type
Communication
Submitted
20 May 2002
Accepted
19 Jun 2002
First published
03 Jul 2002

Chem. Commun., 2002, 1644-1645

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Synthesis of the kappa-agonist CJ-15,161 via a palladium-catalyzed cross-coupling reaction

A. Ghosh, J. E. Sieser, S. Caron and T. J. N. Watson, Chem. Commun., 2002, 1644 DOI: 10.1039/B204844B

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