Issue 24, 2019, Issue in Progress

Copper-catalyzed synthesis of 2-aminopyridylbenzoxazoles via domino reactions of intermolecular N-arylation and intramolecular O-arylation

Abstract

A simple and general approach to nitrogen-containing heterocycles via copper-catalyzed domino reaction has been developed, and the corresponding 2-aminopyridylbenzoxazole derivatives were obtained in good to excellent yields using the readily available starting materials. This method possesses unique step economy features, and is of high tolerance towards various functional groups in the substrates.

Graphical abstract: Copper-catalyzed synthesis of 2-aminopyridylbenzoxazoles via domino reactions of intermolecular N-arylation and intramolecular O-arylation

Supplementary files

Article information

Article type
Paper
Submitted
13 Mar 2019
Accepted
25 Apr 2019
First published
01 May 2019
This article is Open Access
Creative Commons BY-NC license

RSC Adv., 2019,9, 13414-13417

Copper-catalyzed synthesis of 2-aminopyridylbenzoxazoles via domino reactions of intermolecular N-arylation and intramolecular O-arylation

J. Lu, RSC Adv., 2019, 9, 13414 DOI: 10.1039/C9RA01908A

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