Issue 85, 2016
From the journal:

RSC Advances

Rational design of an efficient one-pot synthesis of 6H-pyrrolo[2,3,4-gh]perimidines in polyphosphoric acid†

Alexander V. Aksenov,*a   Nicolai A. Aksenov,ab   Dmitrii S. Ovcharov,a   Dmitrii A. Aksenov,a   Georgii Griaznov,a   Leonid G. Voskressenskyb  and  Michael Rubin*ac  

* Corresponding authors

a Department of Chemistry, North Caucasus Federal University, 1a Pushkin St., Stavropol 355009, Russian Federation
E-mail: alexaks05@rambler.ru

b Department of Organic Chemistry, People's Friendship University of Russia, 6 Miklukho-Maklaya St., Moscow, Russian Federation

c Department of Chemistry, University of Kansas, 1251 Wescoe Hall Dr., Lawrence, KS 66045-7582, USA
E-mail: mrubin@ku.edu
Fax: +1-785-864-5396
Tel: +1-785-864-5071

Abstract

Several highly efficient one-pot synthetic protocols were developed, enabling polyphosphoric acid-activated nitroalkanes to act as electrophiles in reactions with aminonapthalenes. The featured methods allow for the single step assembly of polyheterocyclic aromatic derivatives of 6H-pyrrolo[2,3,4-gh]perimidine scaffold in high yields.

Graphical abstract: Rational design of an efficient one-pot synthesis of 6H-pyrrolo[2,3,4-gh]perimidines in polyphosphoric acid

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Article information

DOI
https://doi.org/10.1039/C6RA17269E
Article type
Paper
Submitted
05 Jul 2016
Accepted
23 Aug 2016
First published
25 Aug 2016

RSC Adv., 2016,6, 82425-82431

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Rational design of an efficient one-pot synthesis of 6H-pyrrolo[2,3,4-gh]perimidines in polyphosphoric acid

A. V. Aksenov, N. A. Aksenov, D. S. Ovcharov, D. A. Aksenov, G. Griaznov, L. G. Voskressensky and M. Rubin, RSC Adv., 2016, 6, 82425 DOI: 10.1039/C6RA17269E

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