Issue 24, 2015
From the journal:

Chemical Communications

Copper-catalyzed ortho-halogenation of arenes and heteroarenes directed by a removable auxiliary†

Bo Li,a   Bin Liua  and  Bing-Feng Shi*ab  

* Corresponding authors

a Department of Chemistry, Zhejiang University, Hangzhou 310027, China
E-mail: bfshi@zju.edu.cn

b State Key Laboratory of Bioorganic & Natural Products Chemistry, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, Shanghai 200032, China

Abstract

Copper-catalyzed ortho-halogenation of C(sp2)–H bonds directed by a PIP directing group with NXS (X = Cl, Br, I) has been developed. The reaction is scalable and tolerates a broad range of functional groups and heteroarenes, providing an efficient access to halogenated arenes and heteroarenes.

Graphical abstract: Copper-catalyzed ortho-halogenation of arenes and heteroarenes directed by a removable auxiliary

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Article information

DOI
https://doi.org/10.1039/C5CC00531K
Article type
Communication
Submitted
19 Jan 2015
Accepted
16 Feb 2015
First published
17 Feb 2015

Chem. Commun., 2015,51, 5093-5096

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Copper-catalyzed ortho-halogenation of arenes and heteroarenes directed by a removable auxiliary

B. Li, B. Liu and B. Shi, Chem. Commun., 2015, 51, 5093 DOI: 10.1039/C5CC00531K

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