Issue 74, 2013

Oxidation of 2-arylindoles for synthesis of 2-arylbenzoxazinones with oxone as the sole oxidant

Abstract

A novel and efficient method for the oxidation of 2-arylindoles to synthesize 2-arylbenzoxazinones utilizing oxone as the sole oxidant has been developed. The reaction tolerates a wide range of functional groups and allows quick and atom-economical assembly of a variety of valuable 2-arylbenzoxazinones in high yields.

Graphical abstract: Oxidation of 2-arylindoles for synthesis of 2-arylbenzoxazinones with oxone as the sole oxidant

Supplementary files

Article information

Article type
Communication
Submitted
05 Jun 2013
Accepted
17 Jul 2013
First published
17 Jul 2013

Chem. Commun., 2013,49, 8196-8198

Oxidation of 2-arylindoles for synthesis of 2-arylbenzoxazinones with oxone as the sole oxidant

X. Lian, H. Lei, X. Quan, Z. Ren, Y. Wang and Z. Guan, Chem. Commun., 2013, 49, 8196 DOI: 10.1039/C3CC44215B

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