Jump to main content
Jump to site search

Issue 14, 2012
Previous Article Next Article

Copper-catalysed addition of α-alkyl azaarenes to ethyl glyoxylate via direct C(sp3)–H activation

Author affiliations

Abstract

A novel protocol for the copper-catalysed direct C(sp3)–H bond functionalisation of 2-alkyl azaarenes to C[double bond, length as m-dash]O double bonds has been developed, which expands the scope of C(sp3)–H bond activation reactions and provides new access to medicinally important azaarene derivatives.

Graphical abstract: Copper-catalysed addition of α-alkyl azaarenes to ethyl glyoxylate via direct C(sp3)–H activation

Back to tab navigation

Supplementary files

Publication details

The article was received on 04 Apr 2012, accepted on 09 May 2012 and first published on 14 May 2012


Article type: Communication
DOI: 10.1039/C2RA20627G
Citation: RSC Adv., 2012,2, 5968-5971
  •   Request permissions

    Copper-catalysed addition of α-alkyl azaarenes to ethyl glyoxylate via direct C(sp3)–H activation

    J. Jin, H. Niu, G. Qu, H. Guo and J. S. Fossey, RSC Adv., 2012, 2, 5968
    DOI: 10.1039/C2RA20627G

Search articles by author

Spotlight

Advertisements