Issue 3, 2011
From the journal:

Chemical Communications

A general and mild domino approach to substituted 1-aminoindoles†

Nis Halland,*a   Marc Nazaré,a   Jorge Alonso,a   Omar R'kyeka  and  Andreas Lindenschmidt*a  

* Corresponding authors

a Sanofi-Aventis Deutschland GmbH, Industriepark Höchst Building G875, D-65926 Frankfurt am Main, Germany
E-mail: nis.halland@sanofi-aventis.com
Fax: +49 69305 21618
Tel: +49 69305 36193

Abstract

A versatile and efficient palladium catalyzed domino reaction leading to a broad range of substituted 1-aminoindoles has been developed. The title compounds were prepared from 2-halo-phenylacetylenes and simple hydrazines in good to excellent yields in just a few hours under mild conditions.

Graphical abstract: A general and mild domino approach to substituted 1-aminoindoles

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Article information

DOI
https://doi.org/10.1039/C0CC03584J
Article type
Communication
Submitted
31 Aug 2010
Accepted
25 Oct 2010
First published
12 Nov 2010

Chem. Commun., 2011,47, 1042-1044

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A general and mild domino approach to substituted 1-aminoindoles

N. Halland, M. Nazaré, J. Alonso, O. R'kyek and A. Lindenschmidt, Chem. Commun., 2011, 47, 1042 DOI: 10.1039/C0CC03584J

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