Issue 14, 1995

Docetaxel (taxotere) derivatives: novel NbCl3-based stereoselective approach to 2′-methyldocetaxel

Abstract

The C-2 methylated 2S,3R and 2R,3S side chains of docetaxel have been enantioselectively prepared and esterified with protected 10-deacetylbaccatin III to provide novel analogues of docetaxel.

Article information

Article type
Paper

J. Chem. Soc., Perkin Trans. 1, 1995, 1811-1815

Docetaxel (taxotere) derivatives: novel NbCl3-based stereoselective approach to 2′-methyldocetaxel

J. Denis, A. Fkyerat, Y. Gimbert, C. Coutterez, P. Mantellier, S. Jost and A. E. Greene, J. Chem. Soc., Perkin Trans. 1, 1995, 1811 DOI: 10.1039/P19950001811

To request permission to reproduce material from this article, please go to the Copyright Clearance Center request page.

If you are an author contributing to an RSC publication, you do not need to request permission provided correct acknowledgement is given.

If you are the author of this article, you do not need to request permission to reproduce figures and diagrams provided correct acknowledgement is given. If you want to reproduce the whole article in a third-party publication (excluding your thesis/dissertation for which permission is not required) please go to the Copyright Clearance Center request page.

Read more about how to correctly acknowledge RSC content.

Spotlight

Advertisements