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Squaramide-catalysed asymmetric Michael addition/cyclization cascade reaction of 4-arylmethylidene-2,3-dioxopyrrolidines with 2-isothiocyanato-1-indanones

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Palladium-catalyzed asymmetric dearomative alkenylation of indoles through a reductive-Heck reaction

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Highly Diastereoselective Synthesis of Oxindoles Containing Vicinal Quaternary and Tertiary Stereocenters by a Domino Heck/Decarboxylative Alkynylation Sequence

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Quadruple C-H activation coupled to hydrofunctionalization and C-H silylation/borylation enabled by weakly coordinated palladium catalyst

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Dearomative ipso-Cyclization to Spiropseudoindoxyls: An Extendable Approach To Access Indolo[3,2-c]quinolinones and Isocryptolepine

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Palladium-Catalyzed Enantioselective Intramolecular Dearomative Heck Reaction

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Palladium-Catalyzed Asymmetric Intramolecular Dearomative Heck Annulation of Aryl Halides to Furnish Indolines

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Progress in Organocatalytic Dearomatization Reactions Catalyzed by N‐Heterocyclic Carbenes

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Palladium-catalyzed intramolecular tandem dearomatization of indoles for the synthesis of tetracyclic indolines

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Direct Construction of Fused/Bridged 3D Rings via Visible‐Light Induced Dearomative Cycloaddition of Arenes

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Sequential Copper‐Catalyzed Sonogashira Coupling, Hydroamination and Palladium‐Catalyzed Intramolecular Direct Arylation: Synthesis of Azepino‐Fused Isoindolinones

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Recent Advances in the Synthesis of Indolines via Dearomative Annulation of N‐acylindoles

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Salicylaldehyde-Promoted Cobalt-Catalyzed C–H/N–H Annulation of Indolyl Amides with Alkynes: Direct Synthesis of a 5-HT3 Receptor Antagonist Analogue

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Palladium-Catalyzed Dearomative Heck/C–H Activation/[4 + 2] Decarboxylative Cyclization of C2-Tethered Indoles

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Pd-Catalyzed de Novo Assembly of Diversely Substituted Indole-Fused Polyheterocycles

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Palladium-Catalyzed Dearomative Heck/Suzuki Coupling of C2-Deuterated or C2-Nonsubstituted Indoles

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Dearomative 1,4-difunctionalization of naphthalenes via palladium-catalyzed tandem Heck/Suzuki coupling reaction

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TfOH-Catalyzed Cascade C–H/N–H Chemo-/Regioselective Annulation of Indole-2-carboxamides with Benzoquinones for the Construction of Anticancer Tetracyclic Indolo[2,3-c]quinolinones

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Palladium-Catalyzed Dual C(sp2)–H Functionalization of Indole-2-carboxamides Involving a 1,2-Acyl Migration: A Synthesis of Indolo[3,2-c]quinolinones

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Dearomatizing [2+2+1] Spiroannulation of Indoles with Alkynes

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Pd(II)/Lewis Acid Catalyzed Intramolecular Annulation of Indolecarboxamides with Dioxygen through Dual C–H Activation

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Synthesis of Tetracyclic Indolines through Palladium‐Catalyzed Asymmetric Dearomative reaction of Aryl Iodides

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Copper(II)-Catalyzed Domino Synthesis of Indolo[3,2-c]quinolinones via Selective Carbonyl Migration

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Org. Lett., 2019, 21, 867
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Synthesis of N,O-Spiroacetals and α-Arylfurans via Pd-Catalyzed Aerobic Oxidative 2,5-Aminoarylation and α-Arylation of N-[3-(2-Furanyl)propyl]-p-toluenesulfonamides with Boronic Acids

Zhiqiang Wang, Wenkun Luo, Lin Lu and Biaolin Yin

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CuH-Catalyzed Synthesis of 3-Hydroxyindolines and 2-Aryl-3H-indol-3-ones from o-Alkynylnitroarenes, Using Nitro as Both the Nitrogen and Oxygen Source

Hui Peng, Jinhui Ma, Lingfei Duan, Guangwen Zhang and Biaolin Yin

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Annulation of Indole-2-Carboxamides with Bicycloalkenes Catalyzed by Ru(II) at Room Temperature: An Easy Access to β-Carboline-1-one Derivatives under Mild Conditions

Gopal Krushna Das Adhikari, Smruti Ranjan Mohanty, Shyam Kumar Banjare, Namrata Prusty, Gajiram Murmu and Ponneri C. Ravikumar

J. Org. Chem., 2023, 88, 952
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Nickel-Catalyzed Enantioselective Dearomative Heck-Reductive Allylic Defluorination Reaction of Indoles

Yuan-Yuan Hu, Xiao-Qiu Xu, Wei-Chao Deng, Ren-Xiao Liang and Yi-Xia Jia

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Concise Synthesis of Carbocycle‐Fused γ‐Carbolinones via Regio‐/Chemoselective Reaction of Indole‐3‐Carboxamides with Cyclic Diazo Compounds

Chang Gao, Bin Li, Biao Cheng, Qianting Zhou, Xinying Zhang and Xuesen Fan

Adv Synth Catal, 2025, 367
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Palladium-Catalyzed Dearomative Heck/C(sp2)–H Activation/Decarboxylative Cyclization of C2-Tethered Indoles

Shuyi Guo, Wenbo Deng, Xiaochang Xiao, Jingru Xia, Xing Yang, Yun Liang and Yuan Yang

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