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Eugene S. Gutman, Thomas C. Irvin, J. Brian Morgan, Rodell C. Barrientos, Oscar B. Torres, Zoltan Beck, Gary R. Matyas, Arthur E. Jacobson and Kenner C. Rice

RSC Chem. Biol., 2021, 2, 835
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Vaccines for substance abuse treatment: new approaches in the immunotherapy of addictions

M. A. Myagkova and V. S. Morozova

Russ Chem Bull, 2018, 67, 1781
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Design, Synthesis, and In Vivo Evaluation of C1-Linked 4,5-Epoxymorphinan Haptens for Heroin Vaccines

Agnieszka Sulima, Fuying Li, Jeffrey Brian Morgan, Phong Truong, Joshua F. G. Antoline, Therese Oertel, Rodell C. Barrientos, Oscar B. Torres, Zoltan Beck, Gregory H. Imler, Jeffrey R. Deschamps, Gary R. Matyas, Arthur E. Jacobson and Kenner C. Rice

Molecules, 2022, 27, 1553
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Efficacy, but Not Antibody Titer or Affinity, of a Heroin Hapten Conjugate Vaccine Correlates with Increasing Hapten Densities on Tetanus Toxoid, but Not on CRM197Carriers

Rashmi Jalah, Oscar B. Torres, Alexander V. Mayorov, Fuying Li, Joshua F. G. Antoline, Arthur E. Jacobson, Kenner C. Rice, Jeffrey R. Deschamps, Zoltan Beck, Carl R. Alving and Gary R. Matyas

Bioconjugate Chem., 2015, 26, 1041
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Opioid-Based Haptens: Development of Immunotherapy

Sándor Hosztafi, Anna Rita Galambos, István Köteles, Dávid Á Karádi, Susanna Fürst and Mahmoud Al-Khrasani

IJMS, 2024, 25, 7781
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Synthesis of 1-Chloronaloxone and 2-Chloronaloxone

James Brailey-Partridge, John S. Carey, Christopher J. Lovell and George M. Taylor

Org. Process Res. Dev., 2021, 25, 2502
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A simple nonradioactive method for the determination of the binding affinities of antibodies induced by hapten bioconjugates for drugs of abuse

Oscar B. Torres, Joshua F. G. Antoline, Fuying Li, Rashmi Jalah, Arthur E. Jacobson, Kenner C. Rice, Carl R. Alving and Gary R. Matyas

Anal Bioanal Chem, 2016, 408, 1191
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Conjugate Vaccine Immunotherapy for Substance Use Disorder

Paul T. Bremer and Kim D. Janda

Pharmacological Reviews, 2017, 69, 298
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Biologics to treat substance use disorders: Current status and new directions

Marco Pravetoni

Human Vaccines & Immunotherapeutics, 2016, 12, 3005
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Endogenous Opiates and Behavior: 2015

Richard J. Bodnar

Peptides, 2017, 88, 126
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A Stable Heroin Analogue That Can Serve as a Vaccine Hapten to Induce Antibodies That Block the Effects of Heroin and Its Metabolites in Rodents and That Cross-React Immunologically with Related Drugs of Abuse

Agnieszka Sulima, Rashmi Jalah, Joshua F. G. Antoline, Oscar B. Torres, Gregory H. Imler, Jeffrey R. Deschamps, Zoltan Beck, Carl R. Alving, Arthur E. Jacobson, Kenner C. Rice and Gary R. Matyas

J. Med. Chem., 2018, 61, 329
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Synthesis of 3‐O‐Carboxyalkyl Morphine Derivatives and Characterization of Their Acid‐Base Properties

István Köteles, Károly Mazák, Gergő Tóth, Péter Horváth, Eszter Kiss, Boglárka Tűz and Sándor Hosztafi

Chemistry & Biodiversity, 2021, 18
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The development of opioid vaccines as a novel strategy for the treatment of opioid use disorder and overdose prevention

Mustafa Tuncturk, Shikha Kushwaha, Robin M Heider, Tyler Oesterle, Richard Weinshilboum and Ming-Fen Ho

International Journal of Neuropsychopharmacology, 2025, 28
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Synthesis of Potential Haptens with Morphine Skeleton and Determination of Protonation Constants

István Köteles, Károly Mazák, Gergő Tóth, Boglárka Tűz and Sándor Hosztafi

Molecules, 2020, 25, 4009
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Synthesis of a deuterated 6‐AmHap internal standard for the determination of hapten density in a heroin vaccine drug product

Mariia Makarova, Rodell C. Barrientos, Oscar B. Torres, Gary R. Matyas, Arthur E. Jacobson, Agnieszka Sulima and Kenner C. Rice

Labelled Comp Radiopharmac, 2020, 63, 564
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The morphine/heroin vaccine decreased the heroin-induced antinociceptive and reinforcing effects in three inbred strains mouse

Susana Barbosa-Méndez, Maura Matus-Ortega, Ricardo Hernández-Miramontes and Alberto Salazar-Juárez

International Immunopharmacology, 2021, 98, 107887
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The M3-TT Vaccine Decreases the Antinociceptive Effects of Morphine and Heroin in Mice

Susana Barbosa-Méndez, Maura Matus-Ortega, Ricardo Hernández Miramontes and Alberto Salazar-Juárez

Int J Ment Health Addiction, 2023, 21, 783
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A Rapid Method for Direct Quantification of Antibody Binding-Site Concentration in Serum

Erwin G. Abucayon, Connor Whalen, Oscar B. Torres, Alexander J. Duval, Agnieszka Sulima, Joshua F. G. Antoline, Therese Oertel, Rodell C. Barrientos, Arthur E. Jacobson, Kenner C. Rice and Gary R. Matyas

ACS Omega, 2022, 7, 26812
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Anti-Strychnine Immunoconjugate Reduces the Effects of Strychnine-Induced Toxicity in Mice

Carly Baehr, Andrew J. Kassick, Jennifer Vigliaturo, Diego Luengas, Aaron Khaimraj, Marco Pravetoni, Saadyah E. Averick and Michael D. Raleigh

ACS Chem. Neurosci., 2023, 14, 1291
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