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Org. Biomol. Chem., 2017, 15, 1350
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Comparison of the substrate selectivity and biochemical properties of human and bacterial γ-butyrobetaine hydroxylase

Anna M. Rydzik, Ivanhoe K. H. Leung, Grazyna T. Kochan, Nikita D. Loik, Luc Henry, Michael A. McDonough, Timothy D. W. Claridge and Christopher J. Schofield

Org. Biomol. Chem., 2014, 12, 6354
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Substrate scope for trimethyllysine hydroxylase catalysis

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Chem. Commun., 2016, 52, 12849
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Biochemical investigations using mass spectrometry to monitor JMJD6-catalysed hydroxylation of multi-lysine containing bromodomain-derived substrates

Thomas P. Corner, Eidarus Salah, Anthony Tumber, Lennart Brewitz and Christopher J. Schofield

RSC Chem. Biol., 2025, 6, 642
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Fluorine nuclear magnetic resonance-based assay in living mammalian cells

Marina Veronesi, Francesca Giacomina, Elisa Romeo, Beatrice Castellani, Giuliana Ottonello, Chiara Lambruschini, Gianpiero Garau, Rita Scarpelli, Tiziano Bandiera, Daniele Piomelli and Claudio Dalvit

Analytical Biochemistry, 2016, 495, 52
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Ligand-Based Fluorine NMR Screening: Principles and Applications in Drug Discovery Projects

Claudio Dalvit and Anna Vulpetti

J. Med. Chem., 2019, 62, 2218
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Trimethyllysine: From Carnitine Biosynthesis to Epigenetics

Marijn N. Maas, Jordi C. J. Hintzen, Miriam R. B. Porzberg and Jasmin Mecinović

IJMS, 2020, 21, 9451
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Good Partnership between Sulfur and Fluorine: Sulfur-Based Fluorination and Fluoroalkylation Reagents for Organic Synthesis

Chuanfa Ni, Mingyou Hu and Jinbo Hu

Chem. Rev., 2015, 115, 765
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Synthetic Applications of Monofluoromethylsulfonium Salts

Renate Melngaile and Janis Veliks

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NMR studies of the non-haem Fe(II) and 2-oxoglutarate-dependent oxygenases

Naasson M. Mbenza, Praveen G. Vadakkedath, Duncan J. McGillivray and Ivanhoe K.H. Leung

Journal of Inorganic Biochemistry, 2017, 177, 384
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Fluorinated Carnitine Derivatives as Tools to Visualise Carnitine Transport and Metabolism

Richard S. Edwards, Ella‐May Hards, Sofia N. dos Santos, Hannah E. Greenwood, Madeleine E. George, Andrea Emanuelli, Muhammet Tanc, Thomas R. Eykyn and Timothy H. Witney

Advanced Science, 2026, 13
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S‐(Trifluoromethyl)Benzothioate (TFBT): A KF‐Based Reagent for Nucleophilic Trifluoromethylthiolation

Depei Meng, Yichong Lyu, Chuanfa Ni, Min Zhou, Yang Li and Jinbo Hu

Chemistry A European J, 2022, 28
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Oxygenase‐Catalyzed Desymmetrization of N,N‐Dialkyl‐piperidine‐4‐carboxylic Acids

Anna M. Rydzik, Ivanhoe K. H. Leung, Grazyna T. Kochan, Michael A. McDonough, Timothy D. W. Claridge and Christopher J. Schofield

Angewandte Chemie, 2014, 126, 11105
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(R)‐α‐Trifluoromethylalanine as a 19F NMR Probe for the Monitoring of Protease Digestion of Peptides

Emmanuelle Devillers, Evelyne Chelain, Claudio Dalvit, Thierry Brigaud and Julien Pytkowicz

ChemBioChem, 2022, 23
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Fluoromethylcarnitine, a novel inhibitor of trimethylamine levels in trimethylaminuria and trimethylamine N-oxide related disorders

Elena Cini, Giorgia Vinciarelli, Sofia Siciliano, Giorgio Del Castello, Elena Dreassi, Federica Poggialini, Chiara Vagaggini, Maurizio Taddei, Gianfranco Battistuzzi, Andrea Castagnetti, Elisa Viciani, Laura Salvini, Antonina Sidoti, Simona Alibrandi and Giuseppe Giannini

European Journal of Medicinal Chemistry, 2025, 300, 118073
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Optimized Monofluoromethylsulfonium Reagents for Fluoromethylene-Transfer Chemistry

Arturs Sperga, Renate Melngaile, Armands Kazia, Sergey Belyakov and Janis Veliks

J. Org. Chem., 2021, 86, 3196
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Profiling Inhibitor Scaffolds for the Cancer Target Jumonji‐C Domain‐Containing Protein 6

Thomas P. Corner, Eidarus Salah, Anthony Tumber, James P. Holt‐Martyn, Lennart Brewitz and Christopher J. Schofield

ChemMedChem, 2025, 20
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Fluorine NMR functional screening: from purified enzymes to human intact living cells

Claudio Dalvit, Marina Veronesi and Anna Vulpetti

J Biomol NMR, 2020, 74, 613
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Molecular Sensors for NMR-Based Detection

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Chem. Rev., 2019, 119, 195
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Oxygenase‐Catalyzed Desymmetrization of N,N‐Dialkyl‐piperidine‐4‐carboxylic Acids

Anna M. Rydzik, Ivanhoe K. H. Leung, Grazyna T. Kochan, Michael A. McDonough, Timothy D. W. Claridge and Christopher J. Schofield

Angew Chem Int Ed, 2014, 53, 10925
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19F NMR as a tool in chemical biology

Diana Gimenez, Aoife Phelan, Cormac D Murphy and Steven L Cobb

Beilstein J. Org. Chem., 2021, 17, 293
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Direct syntheses of stereoisomers of 3-fluoro GABA and β-fluoroamine analogues of the calcium receptor (CaR) agonists, cinacalcet, tecalcet, fendiline and NPS R-467

Yohann J. G. Renault, Jiayin Diao, David B. Cordes, Katie Leach and David O’Hagan

Med Chem Res, 2023, 32, 1532
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Fluoromethylene Transfer from Diarylfluoromethylsulfonium Salts: Synthesis of Fluorinated Epoxides

Janis Veliks and Armands Kazia

Chemistry A European J, 2019, 25, 3786
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ChemInform Abstract: Fluoromethylated Derivatives of Carnitine biosynthesis Intermediates — Synthesis and Applications.

Anna M. Rydzik, Ivanhoe K. H. Leung, Armin Thalhammer, Grazyna T. Kochan, Timothy D. W. Claridge and Christopher J. Schofield

ChemInform, 2014, 45
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Ejection of structural zinc leads to inhibition of γ-butyrobetaine hydroxylase

Anna M. Rydzik, Jürgen Brem, Weston B. Struwe, Grazyna T. Kochan, Justin L.P. Benesch and Christopher J. Schofield

Bioorganic & Medicinal Chemistry Letters, 2014, 24, 4954
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