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Enantioselective Synthesis of Polycyclic Spiroheterocycles by Chiral Phosphoric Acid Catalyzed Dearomative Cyclization of γ‐Hydroxy Ynamides

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Angew Chem Int Ed, 2026
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Enantioselective Synthesis of Polycyclic Spiroheterocycles by Chiral Phosphoric Acid Catalyzed Dearomative Cyclization of γ‐Hydroxy Ynamides

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Angewandte Chemie, 2026
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Organocatalytic Asymmetric Cascade Bicyclization of 2‐Indolylmethanols with α‐(2‐Indolyl) Propargylic Alcohols to Access Chiral Fluorescent Hexacyclic Bisindoles

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Organocatalytic Enantioselective Nucleophilic Addition of Indole Imine 5-Methides

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Organocatalytic Remote‐Controlled Enantioselective 1,10‐Additions of In Situ Generated Alkynyl 2,4′‐Biphenyl Quinone Methides

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Organocatalytic Enantioselective 1,12‐Addition of Alkynyl Biphenyl Quinone Methides Formed In Situ

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Organocatalytic Dearomatization of β‐Naphthols through a 1,6‐Conjugated Addition of Alkynyl 7‐Methylene‐7H‐indoles Formed In Situ

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Controlling Stereoselectivity with Noncovalent Interactions in Chiral Phosphoric Acid Organocatalysis

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Recent Advances in Organocatalytic Enantioselective Reactions of α‐Functionalized Propargylic Alcohols

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Benzenediazonium Tetrafluoroborate‐Catalyzed Formal [3 + 3] Cyclization of 4‐Hydroxycoumarins With Propargylicalcohols

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Asymmetric Organocatalytic 1,6-Conjugate Addition of Alkynyl 8-Methylenenaphthalen-2(8H)-one Formed In Situ: Synergistic Construction of Axial and Central Chirality

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Organocatalytic Enantioselective Synthesis of Axially Chiral Tetrasubstituted Allenes via Direct 1,8-Addition to In Situ Formed Alkynyl 8-Methylenenaphthalen-2(8H)-ones

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Organocatalytic Stereodivergent Dearomatization and N-Acylation of 2-Amino-3-subsituted Indoles

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Organocatalytic Enantioselective 1,12‐Addition of Alkynyl Biphenyl Quinone Methides Formed In Situ

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Asymmetric Cascade Dearomatization–Cyclization Reaction of Tryptamines with β,γ-Alkynyl-α-imino Esters: Access to Hexahydropyrrolo[2,3-b]indole-Containing Tetrasubstituted α-Amino Allenoates

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Organocatalytic Synthesis of Chiral Tetraarylmethanes from 7‐Indolylmethanols with Thioether as Directing Group

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Organocatalytic Enantioselective Dearomatization of 2,3‐Disubstituted Indoles with α‐(3‐Indolyl)propargylic Alcohols

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Stereoselective Synthesis of Axially Chiral Allenes and Styrenes via Chiral Phosphoric Acid Catalysis: An Overview

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ACS Omega, 2024, 9, 33351
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Beyond 1,4-addition of in-situ generated (aza-)quinone methides and indole imine methides

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Synthesis of Chiral 3H‐Pyrrolo[1,2‐a]indoles Via Organocatalytic Enantioselective Addition of Alkynyl Biphenyl Quinone Methides

Sheng Pan, Xing Wang, Meiwen Liu, Fang Fang, Yan Xia, Pengfei Li and Wenjun Li

ChemCatChem, 2024, 16
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