Substrate-controlled [4+1] and [3+2] annulations of ninhydrin-derived Morita–Baylis–Hillman carbonates to access polysubstituted furans and cyclopentenes

Kai-Kai Wang, Yan-Li Li, Ya-Fei Li, Wei-Wei Yao, Lan-Xin Li, Xiao-Long He and Rongxiang Chen

Chem. Commun., 2024, 60, 3717
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Base-Mediated Tandem [3 + 2] Cycloaddition/Ring Openning Reaction of Arylhydrazonoyl Chlorides with Arylnitroso Compounds for Synthesis of Substituted Diazene Oxides

Yi Li, Weinan Xu, Xidan Lei, Jiangbo Xi, Jing Zou, Gang Wang and Zhao-Lin He

J. Org. Chem., 2023, 88, 14200
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Strategies and Methods for the Synthesis of 2‐Pyrazolines: Recent Developments (2012–2022)

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Adv Synth Catal, 2023, 365, 1934
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Lewis Base Controlled (4+3) and (4+2) Annulations of MBH Carbonates with Benzofuran‐Derived Azadienes: Access to Highly Substituted Benzofuro[3,2‐b]Azepines and Spirotetrahydroquinolines

Kai‐Kai Wang, Ya‐Fei Li, Lan‐Xin Li, Wei‐Wei Yao, Yan‐Li Li, Ran Bi, Feng Li, Xiao‐Long He and Rongxiang Chen

Adv Synth Catal, 2024, 366, 4521
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Synthesis of polysubstituted spiroazepines via [4 + 3] annulation reaction of ninhydrin-derived Morita−Baylis−Hillman carbonates with 1‑heterodienes

Kai-Kai Wang, Ya-Fei Li, Ran Bi, Qing Xu, Wen-Jin Li, Liang-Man Wu, Xiao-Ran Wang, Xue-Hao Wang, Aili Sun and Rongxiang Chen

Journal of Molecular Structure, 2025, 1330, 141478
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Dearomative [4 + 2] cycloaddition of 3‐nitroindoles with ortho‐amino Morita−Baylis−Hillman carbonates to forge indole‐fused quinolines

Kai‐Kai Wang, Yan‐Li Li, Lan‐Xin Li, Wei‐Wei Yao, Ya‐Fei Li, Wen‐Fei Wang, Rongxiang Chen, Yi‐Fan Hu and Aili Sun

Journal of Heterocyclic Chem, 2024, 61, 528
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Recent Advances in the Chemistry of Morita–Baylis–Hillman (MBH) Carbonates: A Review

Rabia Ashraf, Ameer Fawad Zahoor, Sajjad Ahmad, Syed Makhdoom Hussain, Bushra Parveen, Samreen Gul Khan, Usman Nazeer, Asim Mansha, Aijaz Rasool Chaudhry and Ahmad Irfan

Journal of Heterocyclic Chem, 2025
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Iodine‐Mediated One‐Pot Synthesis of 1,4,5‐Substituted Pyrazoles from MBH Acetates via Allyl Hydrazone Intermediate

Dipak J. Dahatonde, Aritra Ghosh, Adilakshmi Vutla and Sanjay Batra

Eur J Org Chem, 2023, 26
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Advances in the Synthesis of Heterocycles with Two and Three Heteroatoms using Hydrazonoyl Halides

Nargiza R. Yamaletdinova and Rail R. Gataullin

Helvetica Chimica Acta, 2024, 107
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DMAP‐promoted [4+2]/[3+3] Annulation Cascade Reaction of Morita–Baylis–Hillman Carbonates with Conjugated Imines to Access Functionalized Benzo[c][2,7]naphthyridine Skeletons

Kai‐Kai Wang, Ran Bi, Ya‐Fei Li, Yue‐Yao Ma, Wen‐Jin Li, Bo‐Wen Zhang, Jun‐Yuan Yan, Xiao‐Long He and Rongxiang Chen

Adv Synth Catal, 2025, 367
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Convenient Synthetic Protocols for Diverse Functionalized Dihydrobenzofuran-Fused Spiro-indanedione-oxindole Scaffolds

Jing Sun, Xueyan Liu, Qiu Sun, Ying Han and Chao-Guo Yan

J. Org. Chem., 2023, 88, 11562
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Facile synthesis of spiro-heterocycles through one-pot multicomponent [3 + 3] cross 1,3-dipolar cycloaddition reactions

Guo-Yang Ma, Ya-Fei Li, Qing Xu, Yue-Yao Ma, Ya-Wen Li, Guo-Qiang Gong, Ning Zhang, Tan Dang and Kai-Kai Wang

Tetrahedron, 2024, 168, 134328
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Substrate-Controlled Diversity-Oriented Synthesis of Novel Polycyclic Frameworks via [4 + 2] and [3 + 2] Annulations of Ninhydrin-Derived MBH Adducts with 3,4-Dihydroisoquinolines

Kaikai Wang, Wenwen Zhou, Jun Jia, Junwei Ye, Mengxin Yuan, Jie Yang, Yonghua Qi and Rongxiang Chen

Molecules, 2023, 28, 6761
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Design, synthesis and molecular modeling of new Pyrazolyl-Benzimidazolone hybrids targeting breast Cancer

Mohamed Adardour, Al-Hassan M. Mustafa, Mehdi Oubahmane, Marouane Ait Lahcen, Emad M. Seif, Manal Abdel Fattah Ezzat, Elena Zaballos-García, Joel T. Mague, Ismail Hdoufane, Driss Cherqaoui, Oliver H. Krämer, Wolfgang Sippl, Hany S. Ibrahim and Abdesselam Baouid

Bioorganic Chemistry, 2025, 157, 108269
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Recent highlights in the synthesis and biological significance of pyrazole derivatives

Ziad Moussa, Mani Ramanathan, Shaikha Mohammad Alharmoozi, Shahad Ali Saeed Alkaabi, Salamah Hamdan Mohammed Al Aryani, Saleh A. Ahmed and Harbi Tomah Al-Masri

Heliyon, 2024, 10, e38894
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Synthesis of functionalized spiro[indanone-benzazepine] scaffolds via [4 + 3] annulation reaction of N-(o-chloromethyl)aryl amides with ninhydrin-derived Morita−Baylis−Hillman carbonates

Kai-Kai Wang, Jun-Wei Ye, Jun Jia, Ya-Fei Li, Wei-Wei Yao, Lan-Xin Li, Su-Miao Zhao, Yan Xu and Rongxiang Chen

Tetrahedron, 2024, 150, 133772
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