DOI: 10.1039/A706283D
(Paper)
Reference Section for: Chem. Commun., 1998, 29-30
Aziridination of naphthalene by 3-acetoxyaminoquinazolin-4(3H)-ones
(Note: The full text of this document is currently only available in the PDF Version )
Robert S. Atkinson, Emma Barker, Christopher K. Meades, Robert S. Atkinson, Christopher K. Meades and Hassan A. Albar
Abstract
Reaction of naphthalene with 3-acetoxyaminoquinazolinones 1, 4 or 8 in the presence of hexamethyldisilazane gives the corresponding mono-aziridine as the major (for 1) or exclusive (for 8) product; on heating in benzene, aziridine 5 acts as an aziridinating agent for alkenes.
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