Synthetic strategies for the construction of C3-fluorinated oxindoles

Deeksha, Bittu and Ritesh Singh

Org. Biomol. Chem., 2023, 21, 6456
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Recent advances in stereoselective construction of fluorinated quaternary carbon centers from fluorinated compounds

Zongwei Li, Lin Fan and Guodu Liu

Org. Biomol. Chem., 2024, 22, 4592
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Organocatalytic atroposelective fluorooxindole addition to coumarin Michael acceptors

Maria Bouda, Grace E. Hana, Dea Xhili, Archita Sripada, Jeffery A. Bertke and Christian Wolf

Chem. Commun., 2025, 61, 7883
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Pd-catalyzed enantioselective reductive Heck reaction of mono-fluoro, gem-difluoro, and trifluoromethyl tethered-alkenes

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Chem. Commun., 2025, 61, 11413
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Sustainable and selective Ni-catalyzed allylation of 2-oxindoles and 2-coumaranones in batch and flow chemistry

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Stereoselective Construction of 3-(Aminoalkylidene)oxindoles in One Pot: Development of a Novel, Robust, and Scalable Process for the Multigram-Scale Preparation of Nintedanib

Saroj Maji, Sabyasachi Halder, Ashok Kumar Sharma, Avinash Madhesiya, Tejender S. Thakur and Gautam Panda

Org. Process Res. Dev., 2024, 28, 754
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Base‐Promoted Diastereoselective Addition of 2‐Aryloxy‐2‐Fluoroketones to N‐(tert‐Butylsulfinyl)Imines

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ChemistrySelect, 2024, 9
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Organocatalytic Asymmetric Conjugate Addition of Fluorooxindoles to Quinone Methides

Maria Bouda, Jeffery A. Bertke and Christian Wolf

J. Org. Chem., 2024, 89, 6100
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Lewis Base‐catalyzed β‐Addition of (Arylsulfonyl) fluoromethane Derivatives to Allenoates

Yong‐Liang Liu, Xiao‐Ping Wang and Ya Li

ChemistrySelect, 2022, 7
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Construction of Enantioenriched Quaternary C–Cl Oxindoles through Palladium-Catalyzed Asymmetric Allylic Substitution with Chloroenolates

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J. Org. Chem., 2023, 88, 15298
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DBU-catalyzed selective β-addition of α-fluoro nitroalkanes to allenoates

Li-Wen Ning, Yi-Hu Jin, Ren-Jie Wang, Youcan Zhang and Ya Li

Journal of Fluorine Chemistry, 2024, 274, 110255
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COAP‐Palladium‐Catalyzed Asymmetric Linear Allylic Alkylation of Vinyl Benzoxazinanones for Multifunctional 3,3′‐Disubstituted Oxindole Derivatives

Jun‐Hao Shen, Sheng‐Suo Zhou, Bai‐Lin Wang, Wen‐Kai Liu, Zheng Wang and Xing‐Wang Wang

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Highly Regio‐ and Enantioselective Cu/Pd Co‐Catalyzed Allylic Alkylation of α‐pyridyl‐α‐fluoroesters: Construction of Quaternary C−F Stereocenters

Xinlong Yan, Zongwei Li, Lin Fan, Jiashan Li and Guodu Liu

Chemistry An Asian Journal, 2023, 18
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Enantioseparation and racemization of 3‐fluorooxindoles

Andi Yuan, Sarah E. Steber, Dea Xhili, Eryn Nelson and Christian Wolf

Chirality, 2023, 35, 619
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Sulfone as traceless activating group: Divergent synthesis of α-fluoroamides with C–F quaternary stereocenters

Jieqing Wu, Liying Fu, Renyi Diao, Longjun Nie, Chi Zhang, Yufeng Li and Chao Feng

Green Synthesis and Catalysis, 2025, 6, 96
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Azidobenziodazolones as Azido Sources for the Enantioselective Copper-Catalyzed Azidation of N-Unprotected 3-Trifluoromethylated Oxindoles

Yu-Xuan Chen, Tao Huo, Quan Yin, Ling-Feng Jiang, Xuan Cheng, Hong-Xiang Ma, Yu-Xuan Jiang, Mei-Zhi Sun and Qing-Hai Deng

Org. Lett., 2023, 25, 2739
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Organocatalyzed Asymmetric Michael Addition of 3-Fluorooxindole to Vinylidene Bisphosphonates

Yi-Hu Jin, Xiao-Ping Wang, Li-Wen Ning, Ren-Jie Wang, Ya Li, Youcan Zhang and Ling-Yan Chen

J. Org. Chem., 2024, 89, 8435
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Asymmetric Michael Addition of Benzofuran-Derived Azadienes to 3-Fluorooxindoles Catalyzed by a Chiral Squaramide Catalyst

Shangzhi Wang, Zhonglin Wei, Jungang Cao, Dapeng Liang, Yingjie Lin and Haifeng Duan

J. Org. Chem., 2025, 90, 10869
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Chiral Acyl Radicals Generated by Visible Light Enable Stereoselective Access to 3,3-Disubstituted Oxindoles: Application toward the Synthesis of (–)- and (+)-Physovenine

Josef Späth, Meghan J. Oddy, Roger Hunter and Wade F. Petersen

Synthesis, 2023, 55, 1736
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Diastereoselective addition of 2-alkoxy-2-fluoroacetate to N-(tert‑butylsulfinyl)imines: Synthesis of α-alkoxy-α-fluoro-β-amino acids

Jie Wei, Li-Wen Ning and Ya Li

Journal of Fluorine Chemistry, 2023, 268, 110118
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