Dipyrrolonaphthyridinedione – (still) a mysterious cross-conjugated chromophore

Bartłomiej Sadowski and Daniel T. Gryko

Chem. Sci., 2023, 14, 14020
DOI: 10.1039/D3SC05272A

Chiral spirosiladiphosphines: ligand development and applications in Rh-catalyzed asymmetric hydrosilylation/cyclization of 1,6-enynes with enhanced reactivity

Fei Hou, Minjie Liu, Tong Ru, Zequn Tan, Yingtang Ning and Fen-Er Chen

Chem. Sci., 2023, 14, 4641
DOI: 10.1039/D2SC06349B

Photocatalytic transformation of aliphatic heterocycles and electron-poor alkenes into functionalized heteroarenes

Lorenzo Di Terlizzi, Davide Ravelli and Burkhard König

Green Chem., 2025, 27, 13303
DOI: 10.1039/D5GC04418A

A cascade A3 coupling strategy towards the regioselective synthesis of β-carboline N-fused pyrrole derivatives with pyridine tethers

Vaishali, Chandi C. Malakar and Virender Singh

New J. Chem., 2023, 47, 1186
DOI: 10.1039/D2NJ04620B

Stereoselective access to furan-fused [5.5.0] bicyclic heterocycles enabled by gold-catalyzed asymmetric [8 + 4] cycloaddition

Xunhua Wang, Jianhua Wang and Xiaoxun Li

Org. Chem. Front., 2025, 12, 159
DOI: 10.1039/D4QO01841A

New page to access pyridine derivatives: synthesis from N-propargylamines

Esmail Vessally, Akram Hosseinian, Ladan Edjlali, Ahmadreza Bekhradnia and Mehdi D. Esrafili

RSC Adv., 2016, 6, 71662
DOI: 10.1039/C6RA08720E

Integration of oxidative arylation with sulfonyl migration: one-pot tandem synthesis of densely functionalized (NH)-pyrroles

Joydev K. Laha, Shubhra Sharma, Rohan A. Bhimpuria, Neetu Dayal, Gurudutt Dubey and Prasad V. Bharatam

New J. Chem., 2017, 41, 8791
DOI: 10.1039/C7NJ01709J

Copper-catalyzed tandem annulation of 2-alkynoyl-2′-iodo-1,1′-biphenyls with isocyanoacetates: a rapid access to pyrrole-fused tetracyclic skeletons

Yifan Ouyang, Kaifu Wu, Wei Zhou and Qian Cai

Org. Chem. Front., 2021, 8, 2456
DOI: 10.1039/D0QO01657H

Synthesis, odor characteristics and biological evaluation of N-substituted pyrrolyl chalcones

Jingyi Hu, Xiaoming Ji, Fangyao Su, Qianrui Zhao, Ganlin Zhang, Mingqin Zhao and Miao Lai

Org. Biomol. Chem., 2022, 20, 8747
DOI: 10.1039/D2OB01561G

Base-promoted ring-closing carbonyl–allene metathesis for the synthesis of 2,4-disubstituted pyrroles

Guolin Cheng, Weiwei Lv and Lulu Xue

Green Chem., 2018, 20, 4414
DOI: 10.1039/C8GC01675E

Ribose conversion with amino acids into pyrraline platform chemicals – expeditious synthesis of diverse pyrrole-fused alkaloid compounds

Soohyeon Cho, Lina Gu, Ik Joon IN, Bo Wu, Taehoon Lee, Hakwon Kim and Sangho Koo

RSC Adv., 2021, 11, 31511
DOI: 10.1039/D1RA06110K

Oxidation of pyrrole by dehaloperoxidase-hemoglobin: chemoenzymatic synthesis of pyrrolin-2-ones

Nikolette L. McCombs, Tatyana Smirnova and Reza A. Ghiladi

Catal. Sci. Technol., 2017, 7, 3104
DOI: 10.1039/C7CY00781G

Synthesis of unsymmetrically tetrasubstituted pyrroles and studies of AIEE in pyrrolo[1,2-a]pyrimidine derivatives

Taian Li, Mong-Feng Chiou, Yajun Li, Changqing Ye, Min Su, Mengyu Xue, Xiaobin Yuan, Chuanchuan Wang, Wen-Ming Wan, Daliang Li and Hongli Bao

Chem. Sci., 2022, 13, 5667
DOI: 10.1039/D2SC00837H

1,2 Wagner–Meerwein shift in aza-Nazarov cyclization: Bi(iii)-catalyzed substrate-dependent divergent synthesis of highly substituted pyrroles and indenes

Deepak Datta Gaonkar, Shon Gangai, Krishna Mhaske and Rishikesh Narayan

Org. Chem. Front., 2025, 12, 5027
DOI: 10.1039/D5QO00168D

A transition metal-free [3 + 2] cycloaddition approach for the efficient synthesis of trisubstituted pyrrole derivatives from β-chlorovinyl aldehydes

Jyoti, Vaishali, Shreya Sharma, Diptangshu P. Borthakur, Deepika, Chandi C. Malakar and Virender Singh

Org. Biomol. Chem., 2025, 23, 4735
DOI: 10.1039/D5OB00351B

Direct synthesis of butadiynyl-substituted pyrroles under solvent- and transition metal-free conditions

Denis N. Tomilin, Bartłomiej Pigulski, Nurbey Gulia, Agata Arendt, Lyubov N. Sobenina, Al'bina I. Mikhaleva, Sławomir Szafert and Boris A. Trofimov

RSC Adv., 2015, 5, 73241
DOI: 10.1039/C5RA08820H

Azido-alkynylation of alkenes through radical-polar crossover

Julien Borrel and Jerome Waser

Chem. Sci., 2023, 14, 9452
DOI: 10.1039/D3SC03309K

Silver-catalyzed tandem cycloisomerization/hydroarylation reactions and mechanistic investigations for an efficient access to 1,2-dihydroisoquinolines

Maxime De Abreu, Yue Tang, Etienne Brachet, Mohamed Selkti, Véronique Michelet and Philippe Belmont

Org. Biomol. Chem., 2021, 19, 1037
DOI: 10.1039/D0OB02197K

Novel iron doped calcium oxalates as promising heterogeneous catalysts for one-pot multi-component synthesis of pyranopyrazoles

Kranthi Kumar Gangu, Suresh Maddila, Surya Narayana Maddila and Sreekantha B. Jonnalagadda

RSC Adv., 2017, 7, 423
DOI: 10.1039/C6RA25372E

Solvent-free incorporation of CO2 into 2-oxazolidinones: a review

Sattar Arshadi, Alireza Banaei, Saeideh Ebrahimiasl, Aazam Monfared and Esmail Vessally

RSC Adv., 2019, 9, 19465
DOI: 10.1039/C9RA00551J

Coinage (Au, Ag, Cu) metal-catalyzed (3 + 2) annulation of α-aminoketones and electron-deficient alkynes as a route to 3-EWG-substituted pyrroles

Elena I. Chikunova, Polina F. Kotikova, Dmitry V. Dar'in, Vadim Yu. Kukushkin and Alexey Yu. Dubovtsev

Catal. Sci. Technol., 2024, 14, 5671
DOI: 10.1039/D4CY00660G

Efficient access to 1,3,4-trisubstituted pyrroles via gold-catalysed cycloisomerization of 1,5-diynes

Qiuling Wan, Luoting Xin, Jian Zhang and Xueliang Huang

Org. Biomol. Chem., 2022, 20, 1647
DOI: 10.1039/D1OB02393D

Transition-metal-free and facile synthesis of 3-alkynylpyrrole-2,4-dicarboxylates from methylene isocyanides and propiolaldehyde

Xiaoli Huo, Xiaojuan Chen, Liya Yu, Chong Zhang, Linghui Zeng, Huajian Zhu, Jiaan Shao, Liping Fu and Jiankang Zhang

New J. Chem., 2021, 45, 16430
DOI: 10.1039/D1NJ03596G

Formal nucleophilic pyrrolylmethylationviapalladium-based auto-tandem catalysis: switchable regiodivergent synthesis and remote chirality transfer

Zhi Chen, Yu-Fan Li, Shun-Zhong Tan, Qin Ouyang, Zhi-Chao Chen, Wei Du and Ying-Chun Chen

Chem. Sci., 2022, 13, 12433
DOI: 10.1039/D2SC05210E

Direct catalytic synthesis of β-(C3)-substituted pyrroles: a complementary addition to the Paal–Knorr reaction

Amol Prakash Pawar, Jyothi Yadav, Nisar Ahmad Mir, Eldhose Iype, Krishnan Rangan, Sumati Anthal, Rajni Kant and Indresh Kumar

Chem. Commun., 2021, 57, 251
DOI: 10.1039/D0CC06357F

Catalyst-free direct regiospecific multicomponent synthesis of C3-functionalized pyrroles

Amol Prakash Pawar, Jyothi Yadav, Atul Jankiram Dolas, Eldhose Iype, Krishnan Rangan and Indresh Kumar

Org. Biomol. Chem., 2022, 20, 5747
DOI: 10.1039/D2OB00961G

Samarium(ii) iodide-mediated reactions applied to natural product total synthesis

Majid. M. Heravi and Azadeh Nazari

RSC Adv., 2022, 12, 9944
DOI: 10.1039/D1RA08163B

RhCl(PPh3)3-mediated C–H oxyfunctionalization of pyrrolido-functionalized bisazoaromatic pincers: a combined experimental and theoretical scrutiny of redox-active and spectroscopic properties

Tapas Ghorui, Sima Roy, Shuvam Pramanik and Kausikisankar Pramanik

Dalton Trans., 2016, 45, 5720
DOI: 10.1039/C5DT05044H

Magnetic solid sulfonic acid-enabled direct catalytic production of biomass-derived N-substituted pyrroles

Keping Wang, Mei Wu, Yixuan Liu, Ying Yang and Hu Li

New J. Chem., 2022, 46, 5312
DOI: 10.1039/D1NJ05828B

Iron-catalyzed [3 + 2]-cycloaddition of in situ generated N-ylides with alkynes or olefins: access to multi-substituted/polycyclic pyrrole derivatives

Kai Zhou, Ming Bao, Jingjing Huang, Zhenghui Kang, Xinfang Xu, Wenhao Hu and Yu Qian

Org. Biomol. Chem., 2020, 18, 409
DOI: 10.1039/C9OB02571E

Arylsulfonylmethyl isocyanides: a novel paradigm in organic synthesis

Tanpreet Kaur, Preeti Wadhwa and Anuj Sharma

RSC Adv., 2015, 5, 52769
DOI: 10.1039/C5RA07876H

Divergent copper-catalyzed syntheses of 3-carboxylpyrroles and 3-cyanofurans from O-acetyl oximes and β-ketoesters/nitriles

Wilfrido E. Almaraz-Ortiz, Aldahir Ramos Orea, Oscar Casadiego-Díaz, Agustín Reyes-Salgado, Arturo Mejía-Galindo and Rubén O. Torres-Ochoa

RSC Adv., 2022, 12, 26673
DOI: 10.1039/D2RA04938D

Five-membered heterocycles as promising platforms for molecular logic gate construction

Alexander Ciupa

RSC Adv., 2025, 15, 10565
DOI: 10.1039/D5RA00749F

Ru(ii)-Catalyzed, Cu(ii)-mediated carbene migratory insertion in the synthesis of trisubstituted pyrroles from isoxazoles

Pravin Kumar, Santosh Kumar Keshri and Manmohan Kapur

Org. Biomol. Chem., 2021, 19, 3428
DOI: 10.1039/D1OB00255D

Flow synthesis approaches to privileged scaffolds – recent routes reviewed for green and sustainable aspects

Antonella Ilenia Alfano, Margherita Brindisi and Heiko Lange

Green Chem., 2021, 23, 2233
DOI: 10.1039/D0GC03883K

Intramolecular iron-catalyzed transannulation of furans with O-acetyl oximes: synthesis of functionalized pyrroles

Anton S. Makarov, Alexander A. Fadeev and Maxim G. Uchuskin

Org. Chem. Front., 2021, 8, 6553
DOI: 10.1039/D1QO01281A

Novel 7-(1H-pyrrol-1-yl)spiro[chromeno[4,3-b]quinoline-6,1′-cycloalkanes]: synthesis, cross-coupling reactions, and photophysical properties

Letícia B. Silva, Felipe S. Stefanello, Sarah C. Feitosa, Clarissa P. Frizzo, Marcos A. P. Martins, Nilo Zanatta, Bernardo A. Iglesias and Helio G. Bonacorso

New J. Chem., 2021, 45, 4061
DOI: 10.1039/D0NJ05740A

Zinc(ii)-catalysed cyclocondensation of oxime ethers triggered by polarity inversion: construction of fused pyrroles

Norihiko Takeda, Sora Fujita, Kaho Murakami, Chihiro Honda, Hina Tomoda, Motohiro Yasui, Takahiro Yamada and Masafumi Ueda

Chem. Commun., 2025, 61, 7995
DOI: 10.1039/D5CC01362C

Direct synthesis of 2,3,5-trisubstituted pyrroles via copper-mediated one-pot multicomponent reaction

Jian-Ping He, Zhen-Zhen Zhan, Nan Luo, Ming-Ming Zhang and Guo-Sheng Huang

Org. Biomol. Chem., 2020, 18, 9831
DOI: 10.1039/D0OB01952F

Copper-catalyzed carbene insertion and ester migration for the synthesis of polysubstituted pyrroles

Mingrui Li, Yiming Sun, Yuxing Xie, Yang Yu, Fei Huang and He Huang

Chem. Commun., 2020, 56, 11050
DOI: 10.1039/D0CC04157B

Rh-catalysed divergent synthesis of polysubstituted pyrroles from α,β-unsaturated ketones via selective single or double insertion of isocyanides

Takuya Shimbayashi, Taiyou Ishige and Ken-ichi Fujita

Org. Chem. Front., 2023, 10, 5559
DOI: 10.1039/D3QO01269G

Gold-catalyzed N,O-functionalization of 1,4-diyn-3-ols with N-hydroxyanilines to form highly functionalized pyrrole derivatives

Yu-Chen Hsu, Shu-An Hsieh, Po-Hsuan Li and Rai-Shung Liu

Chem. Commun., 2018, 54, 2114
DOI: 10.1039/C8CC00330K

Advancements in copper-catalyzed thiocyanation: an update

Karthika U. V., Mohan Neetha and Gopinathan Anilkumar

Org. Biomol. Chem., 2025, 23, 9079
DOI: 10.1039/D5OB01120E

Synthesis of pyrrole disulfides via umpolung of β-ketothioamides

Xiangrui Meng, Weisi Guo, Guangming Nan and Ming Li

Org. Biomol. Chem., 2022, 20, 7609
DOI: 10.1039/D2OB01506D

Ammonium niobium oxalate (ANO) as an efficient catalyst in the Paal–Knorr synthesis of N-substituted pyrroles

Luiz H. Dapper, Kethelyn M. da Rosa, Viviane T. Mena, Rodrigo O. M. A. de Souza, Felipe L. N. da Silva, Thiago Anjos, Filipe Penteado and Eder J. Lenardão

RSC Sustainability, 2024, 2, 521
DOI: 10.1039/D3SU00395G

Sequential multicomponent catalytic synthesis of pyrrole-3-carboxaldehydes: evaluation of antibacterial and antifungal activities along with docking studies

Nisar A. Mir, Panduga Ramaraju, Satheeshvarma Vanaparthi, Sachin Choudhary, Rajnish P. Singh, Preetika Sharma, Rajni Kant, Rajpal Singh, Murugesan Sankaranarayanan and Indresh Kumar

New J. Chem., 2020, 44, 16329
DOI: 10.1039/D0NJ03575K

A simple route to tetracyclic oxazepine-fused pyrrolesviametal-free [3+2] annulation between dibenzo[b,f][1,4]oxazepines and aqueous succinaldehyde

Sachin Choudhary, Anoop Singh, Jyothi Yadav, Nisar A. Mir, Sumati Anthal, Rajni Kant and Indresh Kumar

New J. Chem., 2019, 43, 953
DOI: 10.1039/C8NJ04861D

A multi-component synthesis of N-substituted 2-amino-3-cyano pyrroles via ring-opening of nitroepoxides

Xingyu Liu, Zhuang Nie, Jiaan Shao, Wenteng Chen and Yongping Yu

New J. Chem., 2018, 42, 2368
DOI: 10.1039/C7NJ04584K

Conformational rigidity controlled copper catalyzed chemodivergent annulation

Pratap Kumar Mandal, Subhra Kanti Mahato, Neelam, Soumalya Panja, Parikshit Moitra and Amit Kumar Simlandy

Org. Chem. Front., 2026, 13, 1003
DOI: 10.1039/D5QO01518A

Rapid, room-temperature self-organization of polyarylated 1H-pyrroles from acetylenes and nitriles in the KOBut/DMSO system

Elena Yu. Schmidt, Inna V. Tatarinova, Natal'ya A. Lobanova, Igor A. Ushakov, Irina Yu. Bagryanskaya and Boris A. Trofimov

Org. Biomol. Chem., 2023, 21, 7209
DOI: 10.1039/D3OB01311A

Consecutive reactions to construct tricarbonyl compounds and synthetic applications thereof

Diego Madroñero, Cesar A. Mujica-Martinez and Alfredo Vázquez

RSC Adv., 2021, 11, 33235
DOI: 10.1039/D1RA05187C

3-Thiolated pyrroles/pyrrolines: controllable synthesis and usage for the construction of thiolated fluorophores

Jun Tian, Kang-Ning Yuan, Wen Liu, Hong-Hong Chang, Xing Li and Wen-Chao Gao

Chem. Commun., 2021, 57, 1943
DOI: 10.1039/D0CC07988J

Enal-azomethine ylides: application in the synthesis of functionalized pyrroles

Pratap Kumar Mandal, Sandeep Patel and Sreenivas Katukojvala

Org. Biomol. Chem., 2024, 22, 5734
DOI: 10.1039/D4OB00859F

Sequential multicomponent site-selective synthesis of 4-iodo and 5-iodopyrrole-3-carboxaldehydes from a common set of starting materials by tuning the conditions

Sachin Choudhary, Jyothi Yadav, Mamta, Amol Prakash Pawar, Satheeshvarma Vanaparthi, Nisar A. Mir, Eldhose Iype, Ratika Sharma, Rajni Kant and Indresh Kumar

Org. Biomol. Chem., 2020, 18, 1155
DOI: 10.1039/C9OB02501D

A transition metal-free approach towards the regioselective synthesis of β-carboline tethered pyrroles and 2,3-dihydro-1H-pyrroles

Manpreet Singh, Avijit Kumar Paul and Virender Singh

New J. Chem., 2020, 44, 12370
DOI: 10.1039/D0NJ02315A

Construction of pyrroles, furans and thiophenes via intramolecular cascade desulfonylative/dehydrogenative cyclization of vinylidenecyclopropanes induced by NXS (X = I or Br)

Zhe Meng, Jun Yan, Chao Ning, Min Shi and Yin Wei

Chem. Sci., 2023, 14, 7648
DOI: 10.1039/D3SC01542D

Copper-catalyzed decarboxylative ethynyl methylene cyclic carbamates with amines: modular synthesis of 3-aminopyrroles

Jiadong Chen and Shengbiao Tang

New J. Chem., 2024, 48, 16996
DOI: 10.1039/D4NJ03137G

Direct synthesis of pentasubstituted pyrroles and hexasubstituted pyrrolines from propargyl sulfonylamides and allenamides

Changqing Ye, Yihang Jiao, Mong-Feng Chiou, Yajun Li and Hongli Bao

Chem. Sci., 2021, 12, 9162
DOI: 10.1039/D1SC02090K

Application of the Cu(i)/TEMPO/O2catalytic system for aerobic oxidative dehydrogenative aromatization of pyrrolidines

Zheng Luo, Yan Liu, Chao Wang, Danjun Fang, Junyu Zhou and Huayou Hu

Green Chem., 2019, 21, 4609
DOI: 10.1039/C9GC01932D

Recent advances in the transition metal-free synthesis of heterocycles from α,β-unsaturated ketones

Kizhakkan Thiruthi Ashitha, Ajay Krishna M. S., Basavaraja D. and Sasidhar B. Somappa

Org. Chem. Front., 2022, 9, 5306
DOI: 10.1039/D2QO00278G

Selective synthesis of functionalized pyrroles from 3-aza-1,5-enynes

Yingying Zhao, Haolong Wang, Xincheng Li, Dongping Wang, Xiaoyi Xin and Boshun Wan

Org. Biomol. Chem., 2016, 14, 526
DOI: 10.1039/C5OB01887K

Synthesis of 2,5-disubstituted pyrroles via dehydrogenative condensation of secondary alcohols and 1,2-amino alcohols by supported platinum catalysts

S. M. A. H. Siddiki, Abeda S. Touchy, Chandan Chaudhari, Kenichi Kon, Takashi Toyao and Ken-ichi Shimizu

Org. Chem. Front., 2016, 3, 846
DOI: 10.1039/C6QO00165C

A synthesis of fuctionalized 2-amino-3-cyano pyrroles from terminal alkynes, sulfonyl azides and phenacylmalononitriles

Issa Yavari, Meysam Ghorbanzadeh and Somayeh Akbarzadeh

Org. Biomol. Chem., 2022, 20, 4352
DOI: 10.1039/D2OB00277A

Synthesis and fungicidal activity of 3,4-dichloroisothiazole based strobilurins as potent fungicide candidates

Lai Chen, Xiao-Feng Guo, Zhi-Jin Fan, Nai-Lou Zhang, Yu-Jie Zhu, Zhi-Ming Zhang, Inna Khazhieva, Morzherin Y. Yurievich, Nataliya P. Belskaya and Vasiliy A. Bakulev

RSC Adv., 2017, 7, 3145
DOI: 10.1039/C6RA25520E

Facile synthesis of 5α-functionalized pyrroles via multicomponent reactions of vicinal tricarbonyl compounds, enamines, and nucleophiles

Hua-li Wan, Zhao-ping Shi and Qiang Sha

Org. Chem. Front., 2024, 11, 5390
DOI: 10.1039/D4QO00951G

Microwave assisted synthesis of five membered nitrogen heterocycles

Gopinadh Meera, K. R. Rohit, Salim Saranya and Gopinathan Anilkumar

RSC Adv., 2020, 10, 36031
DOI: 10.1039/D0RA05150K

Copper-catalyzed three-component annulation toward pyrroles via the cleavage of two C–C bonds in 1,3-dicarbonyls

Gaochen Xu, Luchao Li, Binyan Xu, Zheng Fang, Jindian Duan and Kai Guo

Chem. Commun., 2023, 59, 10636
DOI: 10.1039/D3CC02681G

Regioselective BF3·Et2O-catalyzed C–H functionalization of indoles and pyrrole with reaction of α-diazophosphonates

Yan Cai, Yuming Li, Minxuan Zhang, Jiaxin Fu and Zhiwei Miao

RSC Adv., 2016, 6, 69352
DOI: 10.1039/C6RA15329A

A new avenue to the synthesis of highly substituted pyrroles: synthesis from N-propargylamines

Esmail Vessally

RSC Adv., 2016, 6, 18619
DOI: 10.1039/C5RA20706A

One-pot sequential multicomponent reaction between in situ generated aldimines and succinaldehyde: facile synthesis of substituted pyrrole-3-carbaldehydes and applications towards medicinally important fused heterocycles

Anoop Singh, Nisar A. Mir, Sachin Choudhary, Deepika Singh, Preetika Sharma, Rajni Kant and Indresh Kumar

RSC Adv., 2018, 8, 15448
DOI: 10.1039/C8RA01637B

Transition metal-catalyzed [2 + 2 + 2] cycloaddition of nitrogen-linked 1,6-diynes: a straightforward route to fused pyrrolidine systems

Mirzaagha Babazadeh, Somayeh Soleimani-Amiri, Esmail Vessally, Akram Hosseinian and Ladan Edjlali

RSC Adv., 2017, 7, 43716
DOI: 10.1039/C7RA05398C

Cobalt-catalyzed acceptorless dehydrogenative coupling of aminoalcohols with alcohols: direct access to pyrrole, pyridine and pyrazine derivatives

Siba P. Midya, Vinod G. Landge, Manoj K. Sahoo, Jagannath Rana and Ekambaram Balaraman

Chem. Commun., 2018, 54, 90
DOI: 10.1039/C7CC07427A

Diverse synthesis of pyrrolo/indolo[3,2-c]coumarins as isolamellarin-A scaffolds: a brief update

Khokan Samanta, Prasanta Patra, Gandhi Kumar Kar, Shaishab Kumar Dinda and Dibyendu Shekhar Mahanty

New J. Chem., 2021, 45, 7450
DOI: 10.1039/D0NJ06267G

Tandem sequential catalytic enantioselective synthesis of highly-functionalised tetrahydroindolizine derivatives

Shuyue Zhang, Mark D. Greenhalgh, Alexandra M. Z. Slawin and Andrew D. Smith

Chem. Sci., 2020, 11, 3885
DOI: 10.1039/D0SC00432D

Cp*Ir(iii) complexes catalyzed solvent-free synthesis of quinolines, pyrroles and pyridines via an ADC strategy

Md. Bakibillah, Sahin Reja, Kaushik Sarkar, Deboshmita Mukherjee, Dilip Sarkar, Sumana Roy, Tahani Mazyad Almutairi, Mohammad Shahidul Islam and Rajesh Kumar Das

Org. Biomol. Chem., 2024, 22, 4704
DOI: 10.1039/D4OB00459K

Chiral Au(iii) chelates exhibit unique NCI-60 cytotoxicity profiles and interactions with human serum albumin

Sheldon Sookai, Matthew P. Akerman and Orde Q. Munro

Dalton Trans., 2024, 53, 5089
DOI: 10.1039/D3DT04024K

The reaction of prop-2-ynylsulfonium salts and sulfonyl-protected β-amino ketones to epoxide-fused 2-methylenepyrrolidines and S-containing pyrroles

Tingting Jia, Gongruixue Zeng, Chong Zhang, Linghui Zeng, Wenya Zheng, Siyao Li, Keyi Wu, Jiaan Shao, Jiankang Zhang and Huajian Zhu

Chem. Commun., 2021, 57, 2657
DOI: 10.1039/D0CC07745C

Kinetic resolution of 1-(1-alkynyl)cyclopropyl ketones via gold-catalyzed divergent (4 + 4) cycloadditions: stereoselective access to furan fused eight-membered heterocycles

Xunhua Wang, Ruifeng Lv and Xiaoxun Li

Chem. Sci., 2024, 15, 9361
DOI: 10.1039/D4SC02763A

Synthesis of disulfides tethered pyrroles from β-ketothioamides via a bicyclization/ring-opening/oxidative coupling reaction

Cong-Xiang Li, Rui-Juan Liu, Kun Yin, Li-Rong Wen and Ming Li

Org. Biomol. Chem., 2017, 15, 5820
DOI: 10.1039/C7OB00655A

Visible light-driven metal-free synthesis of highly substituted pyrroles through C–H functionalisation

Theodora W. von Zuben, Guilherme Cariello Silva and Airton G. Salles

Green Chem., 2021, 23, 6361
DOI: 10.1039/D1GC02177J

A hexameric resorcinarene capsule as a hydrogen bonding catalyst in the conjugate addition of pyrroles and indoles to nitroalkenes

Stefania Gambaro, Margherita De Rosa, Annunziata Soriente, Carmen Talotta, Giuseppe Floresta, Antonio Rescifina, Carmine Gaeta and Placido Neri

Org. Chem. Front., 2019, 6, 2339
DOI: 10.1039/C9QO00224C

BF3-promoted reactions of α-amino acetals with alkynes to 2,5-disubstituted pyrroles

Zhi-Yuan Gao, Yu He, Lan-Yang Li, Jie-Sheng Tian and Teck-Peng Loh

Org. Chem. Front., 2022, 9, 3317
DOI: 10.1039/D2QO00405D

Atom-efficient iron-catalyzed cascade synthesis of pyrroles from nitroarenes under low-pressure conditions

Germán López Robledo, Johannes Fessler, Kathrin Junge and Matthias Beller

Chem. Commun., 2026, 62, 2568
DOI: 10.1039/D5CC05916J

A sustainable C–H functionalization of indoles, pyrroles and furans under a blue LED with iodonium ylides

Saibal Sar, Ranajit Das, Dhiraj Barman, Pikaso Latua, Souvik Guha, Ludovic Gremaud and Subhabrata Sen

Org. Biomol. Chem., 2021, 19, 7627
DOI: 10.1039/D1OB01219C

Cycloamination strategies for renewable N-heterocycles

Hu Li, Haixin Guo, Zhen Fang, Taku Michael Aida and Richard Lee Smith

Green Chem., 2020, 22, 582
DOI: 10.1039/C9GC03655E

Synthesis of multisubstituted pyrroles by nickel-catalyzed arylative cyclizations of N-tosyl alkynamides

Simone M. Gillbard, Chieh-Hsu Chung, Somnath Narayan Karad, Heena Panchal, William Lewis and Hon Wai Lam

Chem. Commun., 2018, 54, 11769
DOI: 10.1039/C8CC06649C

Synthesis of fused cyanopyrroles and spirocyclopropanes via addition of N-ylides to chalconimines

Siba Prasad Midya, Elumalai Gopi, Nishikant Satam and Irishi N. N. Namboothiri

Org. Biomol. Chem., 2017, 15, 3616
DOI: 10.1039/C7OB00529F

A fluorescent target-guided Paal–Knorr reaction

Sachin B. Wagh, Vladimir Maslivetc, James J. La Clair and Alexander Kornienko

RSC Adv., 2020, 10, 37035
DOI: 10.1039/D0RA06962K

Enantioselective β-alkylation of pyrroles with the formation of an all-carbon quaternary stereocenter

Qiao Ma, Lei Gong and Eric Meggers

Org. Chem. Front., 2016, 3, 1319
DOI: 10.1039/C6QO00273K

Synthesis of polysubstituted pyrrolesviaisocyanide-based multicomponent reactions as an efficient synthesis tool

Mohammad Taghi Nazeri and Ahmad Shaabani

New J. Chem., 2021, 45, 21967
DOI: 10.1039/D1NJ04514H

An antibiotic agent pyrrolo[1,2-a]pyrazine-1,4-dione,hexahydro isolated from a marine bacteria Bacillus tequilensis MSI45 effectively controls multi-drug resistant Staphylococcus aureus

George Seghal Kiran, Sethu Priyadharsini, Arya Sajayan, Amrudha Ravindran and Joseph Selvin

RSC Adv., 2018, 8, 17837
DOI: 10.1039/C8RA00820E

N-Propargylic β-enaminocarbonyls: powerful and versatile building blocks in organic synthesis

Sattar Arshadi, Esmail Vessally, Ladan Edjlali, Ebrahim Ghorbani-Kalhor and Rahim Hosseinzadeh-Khanmiri

RSC Adv., 2017, 7, 13198
DOI: 10.1039/C7RA00746A

A two-step resin based approach to reveal survivin-selective fluorescent probes

Andrew J. Ambrose, Nhan T. Pham, Jared Sivinski, Larissa Guimarães, Niloufar Mollasalehi, Paula Jimenez, Maria A. Abad, A. Arockia Jeyaprakash, Steven Shave, Letícia V. Costa-Lotufo, James J. La Clair, Manfred Auer and Eli Chapman

RSC Chem. Biol., 2021, 2, 181
DOI: 10.1039/D0CB00122H

Vinylogous hydrazone strategy for the organocatalytic alkylation of heteroaromatic derivatives

Beata Łukasik, Justyna Kowalska, Sebastian Frankowski and Łukasz Albrecht

Chem. Commun., 2021, 57, 6312
DOI: 10.1039/D1CC01923F

Synthesis and practical applications of 2-(2-nitroalkyl)pyrroles

Alessandro Palmieri and Marino Petrini

Org. Biomol. Chem., 2020, 18, 4533
DOI: 10.1039/D0OB00956C

Post-synthetic diversification of pyrrole-fused benzosultams via trans-sulfonylations and reactions on the periphery of pyrrole

Joydev K. Laha, Rohan A. Bhimpuria and Aitha Manoj Kumar

Org. Chem. Front., 2017, 4, 2170
DOI: 10.1039/C7QO00440K

Divergent [3+2] annulations of oxime acetates with thioaurones/aurones leading to benzothiazino-/benzoyl-pyrroles

Chada Raji Reddy, Damodar Enagandhula, Andhavaram Ramaraju, Avula Shivakrishna and Raju Adepu

Chem. Commun., 2025, 61, 10162
DOI: 10.1039/D5CC00956A

Palladium(ii)-catalysed regioselective synthesis of 3,4-disubstituted quinolines and 2,3,5-trisubstituted pyrroles from alkenes via anti-Markovnikov selectivity

Gopal Chandru Senadi, Wan-Ping Hu, Amol Milind Garkhedkar, Siva Senthil Kumar Boominathan and Jeh-Jeng Wang

Chem. Commun., 2015, 51, 13795
DOI: 10.1039/C5CC05196G

Metal-catalyzed reactions of organic nitriles and boronic acids to access diverse functionality

Hirendra Nath Dhara, Amitava Rakshit, Tipu Alam and Bhisma K. Patel

Org. Biomol. Chem., 2022, 20, 4243
DOI: 10.1039/D2OB00288D

Magnetic sulfonated polysaccharides as efficient catalysts for synthesis of isoxazole-5-one derivatives possessing a substituted pyrrole ring, as anti-cancer agents

Zarrin Ghasemi, Afsaneh Hamidian Amale, Sajjad Azizi, Sepideh Valizadeh and Jafar Soleymani

RSC Adv., 2021, 11, 36958
DOI: 10.1039/D1RA06472J

Reactions of pyrrole, imidazole, and pyrazole with ozone: kinetics and mechanisms

Agnes Tekle-Röttering, Sungeun Lim, Erika Reisz, Holger V. Lutze, Mohammad Sajjad Abdighahroudi, Sarah Willach, Winfried Schmidt, Peter R. Tentscher, Daniel Rentsch, Christa S. McArdell, Torsten C. Schmidt and Urs von Gunten

Environ. Sci.: Water Res. Technol., 2020, 6, 976
DOI: 10.1039/C9EW01078E

Cascade synthesis of 2,4-disulfonylpyrroles by the sulfonylation/[2 + 3]-cycloaddition reactions of gem-dibromoalkenes with arylsulfonyl methyl isocyanides

Parvin Salehi, Zahra Tanbakouchian, Noushin Farajinia-Lehi and Morteza Shiri

RSC Adv., 2021, 11, 13292
DOI: 10.1039/D0RA10451E

Recent progress in molecularly tailored organic hole transporting materials for highly efficient perovskite solar cells

Shakil N. Afraj, Arulmozhi Velusamy, Sakshi Sharma, Jolly Jacob, Juan-Pablo Correa-Baena, Ming-Chou Chen and Antonio Facchetti

J. Mater. Chem. C, 2025, 13, 15234
DOI: 10.1039/D5TC01870F

Two-pot synthesis and photophysical studies of 1,6-disubstituted 5-aza-indoles from succinaldehyde and N-aryl propargylic-imines

Satheeshvarma Vanaparthi, Mamta, Jyothi Yadav, Amol Prakash Pawar, Eldhose Iype, Sravendra Rana and Indresh Kumar

Org. Biomol. Chem., 2021, 19, 10601
DOI: 10.1039/D1OB01949J

An isoxazole strategy for the synthesis of alkyl 5-amino-4-cyano-1H-pyrrole-2-carboxylates – versatile building blocks for assembling pyrrolo-fused heterocycles

Anastasiya V. Agafonova, Liya D. Funt, Mikhail S. Novikov and Alexander F. Khlebnikov

Org. Biomol. Chem., 2021, 19, 1976
DOI: 10.1039/D1OB00053E

Asymmetric synthesis of 4,5-dihydropyrrole derivatives via DKR: DROC of activated aziridines with enaminones

Amit K. Sharma, Poulami Mandal, Ranjan Mali, Noimur Rahman, Nilay K. Pal and Manas K. Ghorai

Org. Chem. Front., 2026, 13, 1783
DOI: 10.1039/D5QO01590A

Construction of axially chiral 2-arylpyrroles using catalytic asymmetric Suzuki–Miyaura cross-coupling: an efficient approach to esaxerenone

Ling Jia, Bing Li, Xi Wang, Jinfeng Zhao, Jingping Qu and Yuhan Zhou

Org. Biomol. Chem., 2024, 22, 8749
DOI: 10.1039/D4OB01174K

An organocatalytic method for constructing pyrroles via the cycloisomerisation of Z-1-iodo-4-N-methylbenzenesulfonyl-1,6-enynes

Long Meng, Xiaochen Chi, Xi Sun, Chengqiang Cao, Bing Ai, Qing Liu, Pingping Zhao, Zengdian Zhao, Yunhui Dong and Hui Liu

Org. Biomol. Chem., 2019, 17, 7669
DOI: 10.1039/C9OB01123D

New route to 1,4-oxazepane and 1,4-diazepane derivatives: synthesis from N-propargylamines

Esmail Vessally, Akram Hosseinian, Ladan Edjlali, Ahmadreza Bekhradnia and Mehdi D. Esrafili

RSC Adv., 2016, 6, 99781
DOI: 10.1039/C6RA20718A

Catalytic Friedel–Crafts Alkylative Desymmetrization of Cyclohexa-2,5-dienones: Access to Linear and Bridged Polycyclic Pyrroles and 3-Arylpyrroles

Raj Kumar Patel, Anil Chauhan, Priyankar Jha, Ruchir Kant and Ravindra Kumar

Org. Lett., 2022, 24, 5422
DOI: 10.1021/acs.orglett.2c02135

Vibrations of pyrrole, N-substituted pyrroles, and their cations

Alexander R. Davies, David J. Kemp and Timothy G. Wright

Journal of Molecular Spectroscopy, 2021, 376, 111410
DOI: 10.1016/j.jms.2020.111410

Inhibition of Pro-inflammatory Enzymes and Growth of an Induced Rheumatoid Arthritis Synovial Fibroblast by Bruguiera cylindrica

Ibrahim M.S. Eldeen, Jochen Ringe and Noraznawati Ismail

International J. of Pharmacology, 2019, 15, 916
DOI: 10.3923/ijp.2019.916.925

Synthesis of Furans and Pyrroles from 2‐Alkoxy‐2,3‐dihydrofurans Through a Nucleophilic Substitution‐Triggered Heteroaromatization

Changhui Liu, Li Zhou, Wenbo Huang, Man Wang and Yanlong Gu

Adv Synth Catal, 2016, 358, 900
DOI: 10.1002/adsc.201500993

Foliar Applications of Bacillus subtilis HA1 Culture Filtrate Enhance Tomato Growth and Induce Systemic Resistance against Tobacco mosaic virus Infection

Hamada El-Gendi, Abdulaziz A. Al-Askar, Lóránt Király, Marwa A. Samy, Hassan Moawad and Ahmed Abdelkhalek

Horticulturae, 2022, 8, 301
DOI: 10.3390/horticulturae8040301

A novel trifluoromethyl 2-phosphonopyrrole analogue inhibits human cancer cell migration and growth by cell cycle arrest at G1 phase and apoptosis

Paulina Olszewska, Dariusz Cal, Piotr Zagórski and Elżbieta Mikiciuk-Olasik

European Journal of Pharmacology, 2020, 871, 172943
DOI: 10.1016/j.ejphar.2020.172943

Catalytic Application of Ionic Liquids for the Green Synthesis of Aromatic Five-Membered Nitrogen Heterocycles

Jaya Dwivedi, Shivangi Jaiswal, Devesh U. Kapoor and Swapnil Sharma

Catalysts, 2025, 15, 931
DOI: 10.3390/catal15100931

1-Methylimidazole as an Organic Catalyst for [3+3]-Cyclodimerization of Acylethynylpyrroles to Bis(acylmethylidene)dipyrrolo[1,2-a:1′,2′-d]pyrazines

Kseniya V. Belyaeva, Lina P. Nikitina, Veronika S. Gen’, Denis N. Tomilin, Lyubov N. Sobenina, Andrei V. Afonin, Ludmila A. Oparina and Boris A. Trofimov

Catalysts, 2022, 12, 1604
DOI: 10.3390/catal12121604

Antimicrobial potential of Streptomyces sp. NP73 isolated from the forest soil of Northeast India against multi-drug resistant Escherichia coli

Aditya Narayan Konwar, Surajit Basak, Kangkon Saikia, Shalini Gurumayum, Nitya Panthi, Jagat Chandra Borah and Debajit Thakur

Letters in Applied Microbiology, 2024, 77
DOI: 10.1093/lambio/ovae086

Synthesis of 2-Arylpyrroles via an Optimized Palladium Coupling

Gunner B. Mitchem and Aaron L. Odom

Synthesis, 2025, 57, 1733
DOI: 10.1055/s-0043-1775453

Trichloromethylthiolation of N‐Heterocycles: Practical and Completely Regioselective

Johannes B. Ernst, Andreas Rühling, Birgit Wibbeling and Frank Glorius

Chemistry A European J, 2016, 22, 4400
DOI: 10.1002/chem.201600377

Chemical Reactivity and Skin Sensitization Studies on a Series of Chloro- and Fluoropyrroles—A Computational Approach

Jaganathan Padmanabhan, Zeeshan Arif, Prakrity Singh and Ramakrishnan Parthasarathi

ACS Omega, 2021, 6, 21514
DOI: 10.1021/acsomega.1c02436

Synthesis of Pyrroles through Rhodium(III)-Catalyzed Reactions of Allylamines and Alkenes

Dong-Su Kim, Yong-Sik Seo and Chul-Ho Jun

Org. Lett., 2015, 17, 3842
DOI: 10.1021/acs.orglett.5b01811

Visible Light‐Induced, Metal‐Free Denitrative [3+2] Cycloaddition for Trisubstituted Pyrrole Synthesis

Bhupal S. Karki, Lalita Devi, Ayushi Pokhriyal, Ruchir Kant and Namrata Rastogi

Chemistry An Asian Journal, 2019, 14, 4793
DOI: 10.1002/asia.201901068

Mn(II) Promoted Divergent‐Convergent Domino Reaction Giving Dinuclear Tetrasubstituted Pyrrole Complex

Jin Cai, Bing Zhao, Qi Zhang, Ao‐Hua Wang, Jia‐Hao Zhang, Bin Liu and Ming‐Hua Zeng

Chemistry A European J, 2024, 30
DOI: 10.1002/chem.202303553

Rational modification of semaxanib and sunitinib for developing a tumor growth inhibitor targeting ATP binding site of tyrosine kinase

Jagroop Kaur, Baljit Kaur and Palwinder Singh

Bioorganic & Medicinal Chemistry Letters, 2018, 28, 129
DOI: 10.1016/j.bmcl.2017.11.049

β‐Trifluoromethyl α,β‐unsaturated Ketones: Efficient Building Blocks for Diverse Trifluoromethylated Molecules

Bharatkumar Chaudhary, Neeraj Kulkarni, Nehanaz Saiyed, Meenakshi Chaurasia, Surbhi Desai, Sagar Potkule and Satyasheel Sharma

Adv Synth Catal, 2020, 362, 4794
DOI: 10.1002/adsc.202001018

Coupled Natural Fusion Enzymes in a Novel Biocatalytic Cascade Convert Fatty Acids to Amines

Shona M. Richardson, Piera M. Marchetti, Michael A. Herrera and Dominic J. Campopiano

ACS Catal., 2022, 12, 12701
DOI: 10.1021/acscatal.2c02954

B(C6F5)3-Catalyzed Dehydrogenation of Pyrrolidines to Form Pyrroles

Ana Alvarez-Montoya, Joseph P. Gillions, Laura Winfrey, Rebecca R. Hawker, Kuldip Singh, Fabrizio Ortu, Yukang Fu, Yang Li and Alexander P. Pulis

ACS Catal., 2024, 14, 4856
DOI: 10.1021/acscatal.3c05444

Sulfonyl Azoles in the Synthesis of 3-Functionalized Azole Derivatives

Alessandro Palmieri and Marino Petrini

The Chemical Record, 2016, 16, 1353
DOI: 10.1002/tcr.201500291

In silico, Synthesis and Biological Investigations of Pyrrolo[3,4-C]Pyrrole Hydroxamic Acid Derivatives as Potential Anticancer Agents

Luis Bahena, Carlos Cervantes, Karla J Soto-Arredondo, Minerva Martínez-Alfaro, Natanael Zarco, Marco A. García-Revilla, Yolanda Alcaraz-Contreras, Lourdes Palma Tirado, Miguel A. Vázquez and Juvencio Robles

J. Mex. Chem. Soc., 2018, 61
DOI: 10.29356/jmcs.v61i4.460

Construction of Polyheterocyclic Compounds by Lewis Acid Mediated Intramolecular [3+2] Cycloaddition Reaction

Pooja Dahiya, Anoop Yadav, Rajnish Budhwan and Rama Krishna Peddinti

Eur J Org Chem, 2023, 26
DOI: 10.1002/ejoc.202300251

Recent Advancements in Pyrrole Synthesis

Satish Chandra Philkhana, Fatimat O. Badmus, Isaac C. Dos Reis and Rendy Kartika

Synthesis, 2021, 53, 1531
DOI: 10.1055/s-0040-1706713

Experimental Evidence of Synergistic Interactions in Pyrrole–Phenol Complexes at Low Temperatures under Isolated Conditions

Shubhra Sarkar, N. Ramanathan and K. Sundararajan

J. Phys. Chem. A, 2018, 122, 9073
DOI: 10.1021/acs.jpca.8b09076

The Synthesis of Multisubstituted Pyrroles via a Copper-Catalyzed Tandem Three-Component Reaction

Xue-Qing Mou, Zheng-Liang Xu, Li Xu, Shao-Hua Wang, Bang-Hong Zhang, Di Zhang, Jie Wang, Wei-Ting Liu and Wen Bao

Org. Lett., 2016, 18, 4032
DOI: 10.1021/acs.orglett.6b01883

Pyrrole-2,5-dione analogs as a promising antioxidant agents: microwave-assisted synthesis, bio-evaluation, SAR analysis and DFT studies/interpretation

Guda Mallikarjuna Reddy, Alexandre Camilo and Jarem Raul Garcia

Bioorganic Chemistry, 2021, 106, 104465
DOI: 10.1016/j.bioorg.2020.104465

Synthesis of Methyl-Protected (±)-Chlorizidine A

Jyoti P. Mahajan and Santosh B. Mhaske

Org. Lett., 2017, 19, 2774
DOI: 10.1021/acs.orglett.7b01090

Comparative Transcriptome Profiling Reveals Potential Candidate Genes, Transcription Factors, and Biosynthetic Pathways for Phosphite Response in Potato (Solanum tuberosum L.)

Richard Dormatey, Tianyuan Qin, Yihao Wang, Benjamin Karikari, Simon Dontoro Dekomah, Youfang Fan, Zhenzhen Bi, Panfeng Yao, Kazim Ali, Chao Sun and Jiangping Bai

Genes, 2022, 13, 1379
DOI: 10.3390/genes13081379

Biological Activities and GC-MS Analysis of Aloe vera and Opuntia ficus-indica Extracts

Afaf Alghamdi, Wafa Alshehri, Bayan Sajer, Mada Ashkan, Ruba Ashy, Rukaia Gashgari, Haifa Hakmi and Muhammad Zia-Ul-Haq

Journal of Chemistry, 2023, 2023, 1
DOI: 10.1155/2023/6504505

Reaction of 1‐Phenacylidene pyrrolo[3,2,1‐ij]quinolin‐2‐ones with Cyclic/Acyclic Enaminones and the Anticoagulant Activity of Synthesized Pyrrole‐Quinoline Derivatives

Anna A. Skoptsova, Alexander S. Shestakov, Irina V. Ledenyova, Nadezhda V. Stolpovskaya, Nadezhda A. Podoplelova, Mikhail A. Panteleev, Boris V. Paponov, Oleg E. Sidorenko, Khidmet S. Shikhaliev and Nadezhda P. Novichikhina

ChemistrySelect, 2022, 7
DOI: 10.1002/slct.202200730

Microwave-Assisted Synthesis of 1-(5-Substituted-4-hydroxy-2-methyl-1H-pyrrol-3-yl)ethan-1-ones from 2-Amino Acid-Derived Enamine-Type Schiff Bases

Diego Quiroga, Sergio Torres-Cortés and Ericsson Coy-Barrera

Molbank, 2025, 2025, M1975
DOI: 10.3390/M1975

Gold(I)-Catalyzed Synthesis of 3-Sulfenyl Pyrroles and Indoles by a Regioselective Annulation of Alkynyl Thioethers

Peter E. Simm, Prakash Sekar, Jeffery Richardson and Paul W. Davies

ACS Catal., 2021, 11, 6357
DOI: 10.1021/acscatal.1c01457

SYNTHESIS OF DEUTERIUM-LABELED PYRROLYLCARNOSINE

V. P. Shevchenko, I. Yu. Nagaev, T. N. Fedorova and N. F. Myasoedov

Doklady Rossijskoj akademii nauk. Nauki o žizni, 2023, 508, 23
DOI: 10.31857/S2686738922700020

Microwave‐assisted Four‐component Cascade Reaction: One‐pot Rapid Access in the Metal‐free Synthesis of Fully Substituted Pyrroles

Zhou Zhang, Jingpeng Li, Zhuoyu Wang, Mengxi Xie, Xiansong Xia and Chao Huang

ChemistrySelect, 2023, 8
DOI: 10.1002/slct.202302666

Current Trends in Pyrrole and Porphyrin-Derived Nanoscale Materials for Biomedical Applications

Parinaz Fathi and Dipanjan Pan

Nanomedicine (Lond.), 2020, 15, 2493
DOI: 10.2217/nnm-2020-0125

Synthesis of Pyrroles through the CuH-Catalyzed Coupling of Enynes and Nitriles

Yujing Zhou, Lin Zhou, Luke T. Jesikiewicz, Peng Liu and Stephen L. Buchwald

J. Am. Chem. Soc., 2020, 142, 9908
DOI: 10.1021/jacs.0c03859

Design, synthesis, and pharmacological evaluation of indazole carboxamides of N-substituted pyrrole derivatives as soybean lipoxygenase inhibitors

Vasiliki Lavrentaki, Antonios Kousaxidis, Panagiotis Theodosis-Nobelos, Georgios Papagiouvannis, Konstantinos Koutsopoulos and Ioannis Nicolaou

Mol Divers, 2024, 28, 3757
DOI: 10.1007/s11030-023-10775-8

Hexafluoroisopropanol as solvent and promotor in the Paal-Knorr synthesis of N-substituted diaryl pyrroles

Robert H.E. Schirmacher, Daniel Rösch and Franziska Thomas

Tetrahedron, 2021, 83, 131985
DOI: 10.1016/j.tet.2021.131985

Catalytic Degradation of Pyrrole in Aqueous Solution by Cu/SBA-15

Shweta Garg, Vimal Chandra Srivastava, Seema Singh and Tapas Kumar Mandal

International Journal of Chemical Reactor Engineering, 2015, 13, 437
DOI: 10.1515/ijcre-2015-0074

Synthesis of New Thiazole Derivatives Bearing Thiazolidin-4(5H)-One Structure and Evaluation of Their Antimicrobial Activity

Asaf Evrim Evren, Leyla Yurttaş and Hülya Karaca Gencer

Braz. J. Pharm. Sci., 2022, 58
DOI: 10.1590/s2175-97902022e19248

Plant Juice Catalysed Synthesis of Substituted Pyrrole through Paal Knorr Reaction

Anis Ahmed Sheikh, Ummul Khair Asema and Abdul Ahad

Int J Sci Res Sci Eng Technol, 2024, 11, 53
DOI: 10.32628/IJSRSET2411586

Synthesis of 3-Aroyl-4-heteroarylpyrrole Derivatives by the Van Leusen Method

Jorge Trilleras, Jairo Quiroga and Angelina Hormaza

Molbank, 2022, 2022, M1341
DOI: 10.3390/M1341

Solubility Determination and Model Evaluation of Triethylamine Hydrochloride in Three Binary Mixed Solvents

Zhe Zhang, Fang Zong, Junfeng Teng, Lili Wang, Xin Jin and Shuguang Xiang

J Solution Chem, 2024, 53, 1353
DOI: 10.1007/s10953-024-01379-3

Magnesium(II) porphyrazine with peripherally overloaded pyrrolyl substituents – Synthesis, optical and electrochemical characterization

Wojciech Szczolko, Tomasz Koczorowski, Pawel Bakun, Michal Kryjewski, Mateusz Grajewski, Lukasz Popenda and Tomasz Goslinski

Journal of Molecular Structure, 2024, 1318, 139356
DOI: 10.1016/j.molstruc.2024.139356

Towards Rare-Functionalized N-Alkenyl-1H-pyrroles via Regioselectively Metalated N-Isopropenyl-1H-pyrroles

Ol'ga A. Tarasova, Marina A. Maximova, Alexander I. Albanov, Nina A. Nedolya and Boris A. Trofimov

Synthesis, 2022, 54, 2516
DOI: 10.1055/a-1736-4200

Characterization of a mercury tolerant strain of Staphylococcus arlettae from Darjeeling hills with an account of its antibiotic resistance pattern and metabolome

Sukanya Acharyya, Sumedha Saha, Soumya Majumder and Malay Bhattacharya

Arch Microbiol, 2021, 203, 5745
DOI: 10.1007/s00203-021-02563-5

Substituted Pyrrololactams via Ring Expansion of Spiro-2H-pyrroles from Intermolecular Alkyne–Isocyanide Click Reactions

Jimil George, Hun Young Kim and Kyungsoo Oh

Org. Lett., 2017, 19, 628
DOI: 10.1021/acs.orglett.6b03786

Neurotoxicity, Neuroprotection, In Vitro MAOA/MAOB Inhibitory Activity Assessment, Molecular Docking, and Permeability Assay Studies of Newly Synthesized Hydrazones Containing a Pyrrole Ring

Maya Georgieva, Emilio Mateev, Iva Valkova, Hristina Kuteva, Diana Tzankova, Denitsa Stefanova, Yordan Yordanov, Karolina Lybomirova, Alexander Zlatkov, Virginia Tzankova and Magdalena Kondeva-Burdina

Molecules, 2024, 29, 4338
DOI: 10.3390/molecules29184338

Synthesis of π-conjugated systems bearing thiophene and pyrrole heterocycles through palladium catalyzed cross-coupling reactions

M. Cidália R. Castro and M. Manuela M. Raposo

Tetrahedron, 2016, 72, 1881
DOI: 10.1016/j.tet.2016.02.054

Recent Advances on MIL‐101 Catalyzed Multicomponent Synthesis of N‐ and O‐Containing Heterocyclic Scaffolds

Sudarshana Sarmah, Pooja Paul, Munmee Goswami and Rishanlang Nongkhlaw

ChemistrySelect, 2025, 10
DOI: 10.1002/slct.202500418

Coumarin hybrid derivatives as promising leads to treat tuberculosis: Recent developments and critical aspects of structural design to exhibit anti-tubercular activity

Dinesh S. Reddy, Manasa Kongot and Amit Kumar

Tuberculosis, 2021, 127, 102050
DOI: 10.1016/j.tube.2020.102050

Pyrrole–Aminopyrimidine Ensembles: Cycloaddition of Guanidine to Acylethynylpyrroles

Olga V. Petrova, Arsalan B. Budaev, Elena F. Sagitova, Igor A. Ushakov, Lyubov N. Sobenina, Andrey V. Ivanov and Boris A. Trofimov

Molecules, 2021, 26, 1692
DOI: 10.3390/molecules26061692

Palladium Catalyzed, Multicomponent Synthesis of Fused-Ring Pyrroles from Aryl Iodides, Carbon Monoxide, and Alkyne-Tethered Imines

Neda Firoozi, Gerardo M. Torres and Bruce A. Arndtsen

J. Org. Chem., 2016, 81, 11145
DOI: 10.1021/acs.joc.6b02102

A Simple and Direct Synthesis of Pentasubstituted Pyrroles via [3+4] Annulation and Their In Vitro Evaluation as Thrombolytic Agents and Cytotoxicity Studies on L929 Cells

Biguvu Balachandra and Sivakumar Shanmugam

ChemistrySelect, 2018, 3, 2037
DOI: 10.1002/slct.201702476

Skeletal Editing of (Hetero)Arenes Using Carbenes

Zhaohong Liu, Paramasivam Sivaguru, Yongquan Ning, Yong Wu and Xihe Bi

Chemistry A European J, 2023, 29
DOI: 10.1002/chem.202301227

Enzyme-Triggered Synthesis and Functionalization of Five-Membered Nitrogen Atom(s) Containing Heterocycles

Shivangi Jaiswal, Annu Bhardwaj, Jaya Dwivedi and Swapnil Sharma

Catal Surv Asia, 2026, 30, 1
DOI: 10.1007/s10563-025-09467-0

2‐Amino‐5‐(cyanomethylsulfanyl)‐1H‐pyrroles from Propargylamines, Isothiocyanates, and Bromoacetonitrile by One‐Pot Synthetic Protocol

Olga A. Tarasova, Nina A. Nedolya, Alexander I. Albanov and Boris A. Trofimov

ChemistrySelect, 2020, 5, 5726
DOI: 10.1002/slct.202000577

Harnessing the Reactivity of Alkyne by Cu‐Catalyst: Assembly of Highly Functionalized Five‐Membered N‐Heterocycles

Md Kalimullah, Divakar Chaudhary and Rakesh K. Saunthwal

Adv Synth Catal, 2025, 367
DOI: 10.1002/adsc.70170

Microwave-assisted green synthesis and structural characterization of N-aryl pyrrole derivatives via Mn-catalyzed Clauson-Kaas reaction: DFT, NMR correlation, and bioactivity evaluation

Meera Gopinadh, K.S. Sunish and Sobhi Daniel

Results in Chemistry, 2026, 21, 103049
DOI: 10.1016/j.rechem.2026.103049

Azanorbornadienes as Thiol-Reactive Cleavable Linkers

Lucrezia De Pascalis, Srinivas Tekkam and M.G. Finn

Org. Lett., 2020, 22, 6248
DOI: 10.1021/acs.orglett.0c01912

Regioselective Brønsted Acid-Catalyzed Annulation of Cyclopropane Aldehydes with N′-Aryl Anthranil Hydrazides: Domino Construction of Tetrahydropyrrolo[1,2-a]quinazolin-5(1H)ones

Priyanka Singh, Navpreet Kaur and Prabal Banerjee

J. Org. Chem., 2020, 85, 3393
DOI: 10.1021/acs.joc.9b03170

Introduction of marine-derivedStreptomycessp. UTMC 1334 as a source of pyrrole derivatives with anti-acetylcholinesterase activity

F. Almasi, F. Mohammadipanah, H.-R. Adhami and J. Hamedi

J Appl Microbiol, 2018, 125, 1370
DOI: 10.1111/jam.14043

Novel Bifunctional Mesoporous Catalysts Based on Preyssler Heteropolyacids for Green Pyrrole Derivative Synthesis

Omar Portilla-Zúñiga, Ángel Sathicq, José Martínez, Hugo Rojas, Eduardo De Geronimo, Rafael Luque and Gustavo P. Romanelli

Catalysts, 2018, 8, 419
DOI: 10.3390/catal8100419

Synthesis and pyrolysis of various novel pyrrole ester fragrance precursors

Pengyu Li, Haiying Tian, Lu Han, Huaiqi Li, Yuhang Ji, Jinchu Yang, Miao Lai, Wenjuan Chu and Xiaoming Ji

Flavour & Fragrance J, 2023, 38, 285
DOI: 10.1002/ffj.3747

Ag(I)-Mediated Annulation of 2-(2-Enynyl)pyridines and Propargyl Amines to Access 1-(2H-Pyrrol-3-yl)indolizines

Feng Li, Qing Yang, Ming-Yue Liu, Pei-Xuan An, Ya-Long Du and Yan-Bo Wang

J. Org. Chem., 2024, 89, 304
DOI: 10.1021/acs.joc.3c02024

Synthesis of Multisubstituted Heterocyclic and Aromatic Compounds Using Catalyst-Controlled Site-Selective Reactions

Miyuki Yamaguchi

Chem. Pharm. Bull., 2026, 74, 132
DOI: 10.1248/cpb.c25-00640

In situ hemisynthesis of new meso -substituted dipyrromethanes using natural aldehydes: in vitro anticholinesterase activity and in silico study

Ramzi Maadadi, Chafai Boukentoucha, Ismahene Bazine, Rafik Menacer, Chawki Bensouici, Leonid Pevzner, Mikhail Petrov, Alexander Stepakov, Anthony Abou Dib and Dominique Harakat

Natural Product Research, 2026, 1
DOI: 10.1080/14786419.2026.2648132

Palladium‐Catalysed Norbornene‐Mediated Regioselective Direct C−H Glycosylation of Free (N−H) Pyrrole Derivatives

Neha Singh Chauhan and Pintu Kumar Mandal

Adv Synth Catal, 2024, 366, 1291
DOI: 10.1002/adsc.202301356

Access to Fused Pyrroles from Cyclic 1,3-Dienyl Boronic Esters and Arylnitroso Compounds

Benjamin François, Ludovic Eberlin, Fabienne Berrée, Andrew Whiting and Bertrand Carboni

J. Org. Chem., 2020, 85, 5173
DOI: 10.1021/acs.joc.9b03214

Iodine‐Promoted One‐pot Synthesis of Highly Substituted 4‐Aminopyrroles and Bis‐4‐aminopyrrole from Aryl Methyl Ketones, Arylamines, and Enamines

Hitesh B. Jalani, Jyotirling R. Mali, Hyejun Park, Jae Kyun Lee, Kiho Lee, Kyeong Lee and Yongseok Choi

Adv Synth Catal, 2018, 360, 4073
DOI: 10.1002/adsc.201800899

Measurement, correlation, and analysis of the solubility of triethylamine hydrochloride in ten pure solvents

Junfeng Teng, Fang Zong, Zhe Zhang, Lili Wang, Xiaoyan Sun and Shuguang Xiang

Journal of Molecular Liquids, 2023, 390, 123040
DOI: 10.1016/j.molliq.2023.123040

Iodine-Promoted Ring-Opening α,β-Difunctionalization of Cyclopropanols with Enaminones: A Selective Route to 2,4-Diacylpyrroles

Jun-Long Zhan, Jiang-Shan Wei, Sheng-Ling Yuan, Yuan-Fei Cui, Meng-Shuang Zhang, Chun-Xiao Xie, Yu-Ting Huang, Qiang Meng, Lin Zhu and Yunhe Lv

Org. Lett., 2025, 27, 10246
DOI: 10.1021/acs.orglett.5c03405

Sustainable Pathways to Pyrroles through Iron‐Catalyzed N‐Heterocyclization from Unsaturated Diols and Primary Amines

Tao Yan and Katalin Barta

ChemSusChem, 2016, 9, 2321
DOI: 10.1002/cssc.201600607

Synthesis of polyfunctionalized pyrroles bearing C-2 α-azido side-chains and displacement of the α-azido group by various nucleophiles

Naomi Kishii, Morie Shimadu, Shun Maruyama, Sayuri Tou, Ikuo Sasaki and Hideyuki Sugimura

Tetrahedron Letters, 2018, 59, 776
DOI: 10.1016/j.tetlet.2018.01.049

Tandem Asymmetric Cycloaromatization/ Intramolecular Pictet‐Spengler‐Type Reaction. An Entry to Polycyclic Pyrroles

Daniel Gaviña, Marcos Escolano, Fernando Rabasa‐Alcañiz, Santiago Díaz‐Oltra, María Sánchez‐Roselló and Carlos del Pozo

Adv Synth Catal, 2022, 364, 2982
DOI: 10.1002/adsc.202200399

One-pot synthesis of new bis(2,4′-bipyridine), bis(pyrrole), and bis(benzo[f]chromene) derivatives: Antimicrobial evaluation, molecular docking, DFT, and ADME profiling

Nabila A. Kheder, Syed Tasqeeruddin, Naglaa S. Mahmoud, Mostafa A.A. Mahmoud and Ismail A. Elhaty

Journal of Molecular Structure, 2026, 1350, 144065
DOI: 10.1016/j.molstruc.2025.144065

Visible-Light-Accelerated Pd-Catalyzed Cascade Addition/Cyclization of Arylboronic Acids to γ- and β-Ketodinitriles for the Construction of 3-Cyanopyridines and 3-Cyanopyrrole Analogues

Amitava Rakshit, Prashant Kumar, Tipu Alam, Hirendranath Dhara and Bhisma K. Patel

J. Org. Chem., 2020, 85, 12482
DOI: 10.1021/acs.joc.0c01703

Quantum Chemical Studies on the Prototropic and Acid/Base Equilibria for 2-Aminopyrrole in Vacuo—Role of CH Tautomers in the Design of Strong Brønsted Imino N-Bases

Ewa Daniela Raczyńska, Pierre-Charles Maria and Jean-François Gal

Molecules, 2025, 30, 2112
DOI: 10.3390/molecules30102112

Ultrafast decay dynamics of N-ethylpyrrole excited to the S1 electronic state: A femtosecond time-resolved photoelectron imaging study

Wen-peng Yuan, Bai-hui Feng, Dong-yuan Yang, Yan-jun Min, Sheng-rui Yu, Guo-rong Wu and Xue-ming Yang

Chinese Journal of Chemical Physics, 2021, 34, 386
DOI: 10.1063/1674-0068/cjcp2104060

The Reactions of p-Tosylmethyl Isocyanide with Aldehydes in the Synthesis of Heterocyclic Compounds: A Review

Nadezhda V. Vchislo, Victoria G. Fedoseeva and Ekaterina A. Verochkina

MROC, 2023, 20, 372
DOI: 10.2174/1570193X19999220523113243

Umpolung Reactivity of Ynamides: An Unconventional [1,3]‐Sulfonyl and [1,5]‐Sulfinyl Migration Cascade

B. Prabagar, Rajendra K. Mallick, Rangu Prasad, Vincent Gandon and Akhila K. Sahoo

Angew Chem Int Ed, 2019, 58, 2365
DOI: 10.1002/anie.201813143

Molecular docking study and molecular dynamics simulation of ethyl 3,5‐diphenyl‐1H‐pyrrole‐2‐carboxylate and (Z)‐ethyl‐2‐(3‐oxo‐1,3‐diphenylprop‐1‐enylamino)acetate

Malahat Kurbanova, Abel Maharramov, Aytan Safarova, Sajjad Ahmad and Youness El Bakri

J Biochem & Molecular Tox, 2022, 36
DOI: 10.1002/jbt.23013

Silver and Copper‐Catalyzed Cycloaddition Reactions of Isocyanide Esters

Fatemeh Doraghi, Parsa Baghershahi, Farzad Gilaninezhad, Negar Mehdi Zadeh Darban, Navid Dastyafteh, Milad Noori and Mohammad Mahdavi

Adv Synth Catal, 2025, 367
DOI: 10.1002/adsc.202400994

5-Arylpyrrolidine-2-carboxylic Acid Derivatives as Precursors in the Synthesis of Sulphonyl-substituted Pyrroles

S. G. Kostryukov, V. A. Kalyazin, P. S. Petrov, E. V. Bezrukova and N. V. Somov

Russ J Org Chem, 2024, 60, 281
DOI: 10.1134/S1070428024020143

α,β-Unsaturated aldehydes in the synthesis of pyrroles (microreview)

Natalia A. Keiko and Nadezhda V. Vchislo

Chem Heterocycl Comp, 2017, 53, 498
DOI: 10.1007/s10593-017-2082-0

Development of a Novel Method for Activation of Isotope Exchange

V. P. Shevchenko, I. Yu. Nagaev, K. V. Shevchenko and N. F. Myasoedov

Radiochemistry, 2023, 65, 442
DOI: 10.1134/S1066362223040069

Acid-Catalyzed Multicomponent Rearrangements via 2-((Quinoxalin-3(4H)-on-2-yl)(aryl)methylene)malononitriles, Generated In Situ, for Divergent Synthesis of Pyrroles with Different Substitution Patterns

Vakhid A. Mamedov, Elena A. Khafizova, Nataliya E. Algaeva, Shamil K. Latypov and Oleg G. Sinyashin

J. Org. Chem., 2020, 85, 9887
DOI: 10.1021/acs.joc.0c01180

Ruthenium(II)‐ and Copper(II)‐Mediated Synthesis of Trisubstituted Pyrroles from Isoxazoles and Acrylate Esters

Pravin Kumar and Manmohan Kapur

Asian J Org Chem, 2020, 9, 1065
DOI: 10.1002/ajoc.202000176

Transition Metal-Free Cyclization of N-Boc-N-propargylenamines

Takayasu Yamauchi, Yuya Chikayuki, Yasuaki Kouno, Shiori Yonekawa, Haruka Ishikawa, Yoko Waki, Hiroyoshi Teramoto, Shigeru Sasaki and Kimio Higashiyama

HETEROCYCLES, 2020, 100, 719
DOI: 10.3987/COM-20-14206

One-Pot Synthesis of 3-Substituted 2-Arylpyrrole in Aqueous Media via Addition–Annulation of Arylboronic Acid and Substituted Aliphatic Nitriles

Md Yousuf and Susanta Adhikari

Org. Lett., 2017, 19, 2214
DOI: 10.1021/acs.orglett.7b00490

Design, Synthesis, and Antifungal Activities of Phenylpyrrole Analogues Based on Alkaloid Lycogalic Acid

Shuaiheng Zhang, Zhenghong Zhou, Tienan Wang and Aidang Lu

Molecules, 2024, 29, 3150
DOI: 10.3390/molecules29133150

Pyrrole: An Essential Framework in the Development of Therapeutic Agents and Insightful Analysis of Structure‐Active Relationships

Bhaskar Sahu, Rakesh Sahu, Bina Gidwani and Achal Mishra

ChemistrySelect, 2024, 9
DOI: 10.1002/slct.202401604

Graphene oxide: a novel acid catalyst for the synthesis of 2,5-dimethyl-N-phenyl pyrrole by the Paal–Knorr condensation

Chun-yan Chen, Xiao-ya Guo, Guang-qiang Lu, Christian Marcus Pedersen, Yan Qiao, Xiang-lin Hou and Ying-xiong Wang

New Carbon Materials, 2017, 32, 160
DOI: 10.1016/S1872-5805(17)60013-6

Molecular Editing of 5-Alkynyl-1,2,3-triazines via a Silver-Mediated Skeletal Remodeling Approach: Solvent-Controlled Switchable Synthesis of Functionalized Pyrroles and Furans

Hsiang-Wen Chen, Wan-Hsuan Liu, Chia-Hao Chang and Jiun-Jie Shie

J. Org. Chem., 2025, 90, 15191
DOI: 10.1021/acs.joc.5c01536

Ring-Chain Tautomerism. I: Synthetic Applications of Heterocycles with One Heteroatom (A Review)

M. Abdel-Megid, T. E. Ali, A. E. Rashad and A. H. Shamroukh

Russ J Org Chem, 2024, 60, 1328
DOI: 10.1134/S107042802407025X

Pyrolysis of spent rapeseed meal: A circular economy example for waste valorization

Riccardo Gallorini, Sara Aquilia, Claudia Bello, Francesco Ciardelli, Michele Pinna, Anna Maria Papini and Luca Rosi

Journal of Analytical and Applied Pyrolysis, 2023, 174, 106138
DOI: 10.1016/j.jaap.2023.106138

Photoredox Catalysis by 21‐Thiaporphyrins: A Green and Efficient Approach for C−N Borylation and C−H Arylation

Anu Janaagal, Apoorv Kushwaha, Pranjali Jhaldiyal, T. J. Dhilip Kumar and Iti Gupta

Chemistry A European J, 2024, 30
DOI: 10.1002/chem.202401623

Iron(iii) chloride-catalyzed mechanochemical cascade synthesis of highly-substituted pyrrolyl indoles

Anindita Mukherjee, Dmitry S. Kopchuk, Sougata Santra, Adinath Majee, Grigory V. Zyryanov and Oleg N. Chupakhin

Mendeleev Communications, 2022, 32, 624
DOI: 10.1016/j.mencom.2022.09.018

Microwave‐activated Synthesis of Pyrroles: A Short Review

Anuradha Sharma and Poonam Piplani

Journal of Heterocyclic Chem, 2017, 54, 27
DOI: 10.1002/jhet.2550

Microwave: A Green Contrivance for the Synthesis of N-Heterocyclic Compounds

Trimurti L. Lambat, Paavan Kavi Param Gaitry Chopra and Sami H. Mahmood

COC, 2020, 24, 2527
DOI: 10.2174/1385272824999200622114919

Synthesis of New Spiroindolinopyrrolidines

S. V. Borisova and V. V. Sorokin

Russ J Gen Chem, 2022, 92, 10
DOI: 10.1134/S1070363222010030

Structural, physico-chemical landscapes, ground state and excited state properties in different solvent atmosphere of Avapritinib and its ultrasensitive detection using SERS/GERS on self-assembly formation with graphene quantum dots

Ali Alsalme, T. Pooventhiran, Nabil Al-Zaqri, D. Jagadeeswara Rao and Renjith Thomas

Journal of Molecular Liquids, 2021, 322, 114555
DOI: 10.1016/j.molliq.2020.114555

A Cascade Reaction for the Synthesis of Multisubstituted Pyrroles from Unsymmetrical 2‐Ene‐1,4‐diones Using Indoles and Ammonium Formate

Wen‐Jing Nan, Ruo‐Fei Lin, Ming‐Li Yuan, Yang‐Yi Li, Wen‐Ming Shu and An‐Xin Wu

ChemistrySelect, 2025, 10
DOI: 10.1002/slct.202503157

Synthesis of fluorinated 3-pyrrolines and pyrroles via [3+2] annulation of N-aryl fluorinated imines with allenoates catalyzed by phosphine

Zhentong Zhu, Yuwei Guo, Xiaojun Wang, Fanhong Wu and Yongming Wu

Journal of Fluorine Chemistry, 2017, 195, 102
DOI: 10.1016/j.jfluchem.2016.12.010

Xiapyrroles A–F: N-Alkylpyrrole Alkaloids from the Marine-Derived Actinomycete Streptomyces xiamenensis 1310KO-148

Min Ah Lee, Jong Soon Kang, Yeo Dae Yoon, Hwa-Sun Lee, Chang-Su Heo, Sun Joo Park and Hee Jae Shin

J. Nat. Prod., 2025, 88, 797
DOI: 10.1021/acs.jnatprod.4c01491

Pyrroles as Privileged Scaffolds in the Search for New Potential HIV Inhibitors

Maria da Conceição Avelino Dias Bianco, Debora Inacio Leite Firmino Marinho, Lucas Villas Boas Hoelz, Monica Macedo Bastos and Nubia Boechat

Pharmaceuticals, 2021, 14, 893
DOI: 10.3390/ph14090893

HFIP-mediated multicomponent reactions for the synthesis of fluorescent quinoline-fused pyrroles

Rohit Kumar, Swadhin Swaraj Acharya, Prabhas Bhaumick, Tasneem Parvin and Lokman H. Choudhury

Tetrahedron, 2023, 132, 133250
DOI: 10.1016/j.tet.2023.133250

Cu-NPs@COF: A potential heterogeneous catalyst for CO2 fixation to produce 2-oxazolidinones as well as benzimidazoles under moderate reaction conditions

Resmin Khatun, Surajit Biswas, Imdadul Haque Biswas, Sk Riyajuddin, Najirul Haque, Kaushik Ghosh and Sk Manirul Islam

Journal of CO2 Utilization, 2020, 40, 101180
DOI: 10.1016/j.jcou.2020.101180

Simple and Efficient “One‐Pot” Synthesis of Diphenylaryl (Heteroaryl) Methanols from Benzene

Irena S. Akhrem, Dzhul'etta V. Avetisyan, Lyudmila V. Afanas'eva and Oleg I. Artyushin

ChemistrySelect, 2020, 5, 7835
DOI: 10.1002/slct.201904255

Chiral counteranion controlled chemoselectivity in gold catalysed hydroamination/enantioselective formal 1,3-allylic alcohol isomerisation of β-amino-1,4-enynols

Lorenzo Carli, Anyawan Tapdara, Jianwen Jin, Yichao Zhao and Philip Wai Hong Chan

Tetrahedron Chem, 2023, 7, 100043
DOI: 10.1016/j.tchem.2023.100043

Xanthine oxidase inhibitory activity of new pyrrole carboxamide derivatives: In vitro and in silico studies

İbrahim Evren Kıbrız, Mustafa Saçmacı, İsmail Yıldırım, Samir Abbas Ali Noma, Tuğba Taşkın Tok and Burhan Ateş

Archiv der Pharmazie, 2018, 351
DOI: 10.1002/ardp.201800165

Electronic, vibrational, and torsional couplings in N-methylpyrrole: Ground, first excited, and cation states

Alexander R. Davies, David J. Kemp and Timothy G. Wright

The Journal of Chemical Physics, 2021, 154
DOI: 10.1063/5.0050654

Synthesis of Highly Substituted 3-Acylpyrroles by a Four-Component Sonogashira Alkynylation–Amine Addition–Nitroalkene Michael Addition–Cyclocondensation

G. Hendrik Schmitz, Panagiota Lampiri and Thomas J. J. Müller

Synlett, 2023, 34, 1781
DOI: 10.1055/a-2077-4955

Design and Synthesis of 4-(2-Pyrrolyl)-4-phenylheptane Derivatives as Estrogen Receptor Antagonists

Genichiro Tsuji, Yosuke Demizu, Miyako Naganuma, Hidetomo Yokoo, Takashi Misawa and Kenji Matsuno

HETEROCYCLES, 2020, 101, 429
DOI: 10.3987/COM-19-14121

Mechanistic Insights into Thiazolidinones as Anticholinesterase Agents: 3D QSAR Pharmacophore Modeling, Molecular Docking, MD Simulations, and DFT Studies for Alzheimer’s Therapy

T. J. Sindhu, Jainey P. James, C. Zakiya Fathima, Bijo Mathew and Sunil Kumar

J. Comput. Biophys. Chem., 2025, 24, 1415
DOI: 10.1142/S2737416525500309

A New Facet of Azatriene Reactivity: A Short Cut to 5‐Amino‐3‐methyl‐4‐(1H‐pyrrol‐1‐yl)thiophene‐2‐carboxylates and 5‐Amino‐3‐methyl‐4‐(1H‐pyrrol‐1‐yl)thiophene‐2‐carbonitriles

Nina A. Nedolya, Olga A. Tarasova, Alexander I. Albanov and Boris A. Trofimov

Eur J Org Chem, 2018, 2018, 1953
DOI: 10.1002/ejoc.201800268

Palladium-carbene catalyzed direct arylation of five-membered heteroaromatics

Murat Kaloğlu, Nazan Kaloğlu, İlkay Yıldırım, Namık Özdemir and İsmail Özdemir

Journal of Molecular Structure, 2020, 1206, 127668
DOI: 10.1016/j.molstruc.2019.127668

Oxidative Aza-Annulation of Enynyl Azides to 2-Keto/Formyl-1H-pyrroles

Chada Raji Reddy, Sujatarani A. Panda and Andhavaram Ramaraju

J. Org. Chem., 2017, 82, 944
DOI: 10.1021/acs.joc.6b02468

Synthesis, odor characteristics and thermal behaviors of pyrrole esters

Jingyi Hu, Meng Zhou, Mengxiao Li, Zizhen Chen, Mingqin Zhao, Xiaoming Ji and Miao Lai

Journal of Saudi Chemical Society, 2023, 27, 101600
DOI: 10.1016/j.jscs.2023.101600

A Practical Synthesis of Densely Functionalized Pyrroles via a Three-Component Cascade Reaction between Carbohydrates, Oxoacetonitriles, and Ammonium Acetate

Mengxin Xia, Mallikharjuna Rao Lambu, Madhu Babu Tatina and Zaher M. A. Judeh

J. Org. Chem., 2021, 86, 837
DOI: 10.1021/acs.joc.0c02381

From Acylethynylpyrroles to Pyrrolo[1,2-a]pyrazines in One Step

E. F. Sagitova, L. N. Sobenina and B. A. Trofimov

Russ J Org Chem, 2020, 56, 225
DOI: 10.1134/S1070428020020082

Modular Domino Process toward Highly Functionalized Pyrroles via Pd-Catalyzed [4 + 1] Annulation under Mild Conditions

Linhong Zuo, Yulian Yang and Wusheng Guo

Org. Lett., 2021, 23, 2013
DOI: 10.1021/acs.orglett.1c00148

Induction of Systemic Resistance to Tobacco mosaic virus in Tomato through Foliar Application of Bacillus amyloliquefaciens Strain TBorg1 Culture Filtrate

Ahmed Abdelkhalek, Dalia G. Aseel, Lóránt Király, András Künstler, Hassan Moawad and Abdulaziz A. Al-Askar

Viruses, 2022, 14, 1830
DOI: 10.3390/v14081830

Synthesis and Applications of Nitrogen-Containing Heterocycles as Antiviral Agents

Tuyen N. Tran and Maged Henary

Molecules, 2022, 27, 2700
DOI: 10.3390/molecules27092700

Synthesis, Characterization, and Evaluation of Tetrazole Derivatives with Pyrrole‐2,5‐Dione Moieties as Urease Inhibitors: Exploring Structure‐Activity Relationships and Computational Insights

Dara Muhammed Aziz and Sangar Ali Hassan

ChemistrySelect, 2024, 9
DOI: 10.1002/slct.202401259

Recent Advances in Biocatalytic Dearomative Spirocyclization Reactions

Xiaorui Chen, Changtong Zhu, Luyun Ji, Changmei Liu, Yan Zhang, Yijian Rao and Zhenbo Yuan

Catalysts, 2025, 15, 673
DOI: 10.3390/catal15070673

Iodine-Catalyzed Regioselective Synthesis of Multisubstiuted Pyrrole Polyheterocycles Free from Rotamers and Keto–Enol Tautomers

Nitika Sharma and Rama Krishna Peddinti

J. Org. Chem., 2017, 82, 9360
DOI: 10.1021/acs.joc.7b01538

Synthesis of N-alkoxycarbonyl Pyrroles from O-Substituted Carbamates: A Synthetically Enabling Pyrrole Protection Strategy

Jodie L. Hann, Catherine L. Lyall, Gabriele Kociok-Köhn and Simon E. Lewis

J. Org. Chem., 2023, 88, 13584
DOI: 10.1021/acs.joc.3c01257

Investigation of Biogenic Silver nanoparticles Concentrations Impact on Novel Benzofuran Derivative and Their Electrochemical Study

Shivaprasadagouda Patil, Mahanthesh Basanagouda, Sudhir M. Hiremath, Aishwarya Nadgir, Malatesh S Pujar, Raghavendra K. Sali, S. Christopher Jeyaseelan and Ashok H. Sidarai

BioNanoSci., 2023, 13, 744
DOI: 10.1007/s12668-023-01092-3

4,11-Dimethyl-2,13-di-m-tolyltribenzo[b,e,g][1,4]dioxocine-7,8-dicarbonitrile

Dmitry Erzunov, Vyacheslav Baklagin, Vladimir Bukhalin, Igor Abramov, Kyrill Yu. Suponitsky and Arthur Vashurin

Molbank, 2025, 2025, M2059
DOI: 10.3390/M2059

Facile Preparation of 2-Aryl-3-iodopyrroles with N-Tosyl 4-Aryl-3-butyn-1-ylamines, I2, and tBuOK

Hideo Togo, Kaho Shibasaki and Hiroki Naruto

HETEROCYCLES, 2021, 102, 1091
DOI: 10.3987/COM-21-14443

Synthesis of Pyrrole via a Silver-Catalyzed 1,3-Dipolar Cycloaddition/Oxidative Dehydrogenative Aromatization Tandem Reaction

Yan Liu, Huayou Hu, Xiang Wang, Sanjun Zhi, Yuhe Kan and Chao Wang

J. Org. Chem., 2017, 82, 4194
DOI: 10.1021/acs.joc.7b00180

Scalable Synthesis of Silacyclohexanones and Ready Access to Silicon Building Blocks

Eagala Ramesh, Laxman D. Nandawadekar, Ramana Sreenivasa Rao and D. Srinivasa Reddy

Org. Lett., 2023, 25, 6881
DOI: 10.1021/acs.orglett.3c02561

Porous SB-Cu1 two-dimensional metal-organic framework: The green catalyst towards C N bond-forming reactions

Sepideh Bagheri, Naghmeh Esfanidiary and Juho Yliniemi

Colloids and Surfaces A: Physicochemical and Engineering Aspects, 2022, 637, 128202
DOI: 10.1016/j.colsurfa.2021.128202

Cascade Assembly of 4,5,6,7-Tetrahydroindole from Cyclohexanone Oxime and Acetylene in the KOH/DMSO Superbase Medium: A Quantum Chemical Study

Alexander S. Bobkov, Nadezhda M. Vitkovskaya and Boris A. Trofimov

J. Org. Chem., 2020, 85, 6463
DOI: 10.1021/acs.joc.0c00353

Metal-free greener method for the synthesis of densely functionalized pyrroles via a one-pot three-component reaction

Maryam Fatahpour, Nourallah Hazeri, Malek Taher Maghsoodlou and Mojtaba Lashkari

J IRAN CHEM SOC, 2019, 16, 111
DOI: 10.1007/s13738-018-1486-9

ChemInform Abstract: Pyrrole: A Resourceful Small Molecule in Key Medicinal Hetero‐Aromatics

Varun Bhardwaj, Divya Gumber, Vikrant Abbot, Saurabh Dhiman and Poonam Sharma

ChemInform, 2015, 46
DOI: 10.1002/chin.201518314

Synthesis of pyrroles via ruthenium-catalyzed nitrogen-transfer [2 + 2 + 1] cycloaddition of α,ω-diynes using sulfoximines as nitrene surrogates

Kazuma Matsui, Masatoshi Shibuya and Yoshihiko Yamamoto

Commun Chem, 2018, 1
DOI: 10.1038/s42004-018-0022-2

Nitroalkenes as Latent 1,2-Biselectrophiles – A Multicatalytic Approach for the Synthesis of 1,4-Diketones and Their Application in a Four-Step One-Pot Reaction to Polysubstituted Pyrroles

Patrick J. W. Fuchs and Kirsten Zeitler

J. Org. Chem., 2017, 82, 7796
DOI: 10.1021/acs.joc.7b00830

Oxidative N-heterocyclic carbene (NHC) catalysis for the rapid access to functionalized pyrrolo-oxazinones

Arghya Ghosh, Shilpa Barik, Soumen Barik, Sayan Shee and Akkattu T. Biju

Tetrahedron, 2021, 94, 132330
DOI: 10.1016/j.tet.2021.132330

Synthesis of 1 H -Pyrazolo[1,2- b ]Phthalazine-5,10-Dione and 1 H -Pyrazolo[1,2- a ]Pyridazine-5,8-Dione Derivatives by Bovine Serum Albumin in Water

Alireza Farahanipour, Hossein Bavandi, Mansour Shahedi and Zohreh Habibi

Polycyclic Aromatic Compounds, 2023, 43, 7042
DOI: 10.1080/10406638.2022.2128829

Asymmetric hydrogenation of α-pyrrolyl terminal alkenes: An easy access to enantioenriched pyrroles bearing a C2 Me-substituted stereogenic center

Ao Zhou, Nianxin Rong, Haokun Zhuang and Qin Yin

Green Synthesis and Catalysis, 2025
DOI: 10.1016/j.gresc.2025.04.003

Substituent-Dependent Divergent Synthesis of 2-(3-Amino-2,4-dicyanophenyl)pyrroles, Pyrrolyldienols and 3-Amino-1-acylethylidene-2-cyanopyrrolizines via Reaction of Acylethynylpyrroles with Malononitrile

Maxim D. Gotsko, Ivan V. Saliy, Igor A. Ushakov, Lyubov N. Sobenina and Boris A. Trofimov

Molecules, 2022, 27, 8528
DOI: 10.3390/molecules27238528

FeCl3‐Catalyzed Formal [3+2] Cyclodimerization of 4‐Carbonyl‐1,2‐diaza‐1,3‐dienes

Giacomo Mari, Matteo Corrieri, Lucia De Crescentini, Gianfranco Favi, Stefania Santeusanio and Fabio Mantellini

Eur J Org Chem, 2021, 2021, 5202
DOI: 10.1002/ejoc.202101046

1-Methoxypyrrole-2-carboxamide—A new pyrrole compound isolated from Streptomyces griseocarneus SWW368

Watsapon Wattanasuepsin, Bungonsiri Intra, Jirayut Euanorasetr, Yoshihiro Watanabe, Ratchanee Mingma, Wataru Fukasawa, Mihoko Mori, Atsuko Matsumoto, Kazuro Shiomi and Watanalai Panbangred

J. Gen. Appl. Microbiol., 2017, 63, 207
DOI: 10.2323/jgam.2016.10.006

Synthesis of Pyrrolopyrazinones by Construction of the Pyrrole Ring onto an Intact Diketopiperazine

Susanna K. Maisto, Angela P. Leersnyder, Gwyneth L. Pudner and Jonathan R. Scheerer

J. Org. Chem., 2020, 85, 9264
DOI: 10.1021/acs.joc.0c01263

Crystal structure and Hirshfeld surface analysis of (2Z)-3-oxo-N-phenyl-2-[(1H-pyrrol-2-yl)methylidene]butanamide monohydrate

Ayten S. Safarova, Ali N. Khalilov, Mehmet Akkurt, Ivan Brito, Ajaya Bhattarai, Farid N. Naghiyev and Ibrahim G. Mamedov

Acta Crystallogr E Cryst Commun, 2023, 79, 1142
DOI: 10.1107/S2056989023009799

Synthesis of Polycyclic Pyrrolopyridine Derivatives via Multicomponent Synthesis of 1,5‐Diketones

Ujjain Chaurasia and Tasneem Parvin

ChemistrySelect, 2024, 9
DOI: 10.1002/slct.202304938

Silver-Catalyzed [3 + 2] Cyclization Reaction of α-Azidovinyl Acids with RCF2-Imidoyl Sulfoxonium Ylides: Synthesis of Polyfluoroalkyl-Substituted 2H-Pyrrole Derivatives

Ruihan Jiang, Hongyu Wang, Lixue Su, Xiubin Bu, Ming Yang, Xiaobo Yang and Yu-Long Zhao

J. Org. Chem., 2026, 91, 2193
DOI: 10.1021/acs.joc.5c02888

New Pyrrole-Chalcone Hybrids Against Acetylcholinesterase: Synthesis, In Vitro, and Computational Studies

Dadan Ridwanuloh, Ade Danova, Elvira Hermawati, Warinthorn Chavasiri, Ihsanawati Ihsanawati and Anita Alni

J. Multidiscip. Appl. Nat. Sci., 2026
DOI: 10.47352/jmans.2774-3047.375

A Mild Method for the Direct Fluorination of Pyrroles by Using a Lipophilic Anionic Phase‐Transfer Catalyst

Kenichi Hiramatsu and Hirokazu Tamamura

Eur J Org Chem, 2016, 2016, 3491
DOI: 10.1002/ejoc.201600570

A Critical Review on Advances in the Multicomponent Synthesis of Pyrroles

Iqbal Azad, Firoj Hassan, Mohammad `Saquib, Naseem Ahmad, Abdul Rahman Khan, Abdillah G.Al-Sehemi and Malik Nasibullah

Orient. J. Chem, 2018, 34, 1670
DOI: 10.13005/ojc/340401

Modular Access to Tetrasubstituted N−H Pyrroles by Catalytic 1,3‐Dipolar Cycloaddition of Azomethine Ylides and α,β‐Ynones

Qian Huang, Zi‐Han Li, Zhen‐Ni Zhao, Bo‐Ting Chen, Feng‐Kai He and Yi‐Yong Huang

Eur J Org Chem, 2024, 27
DOI: 10.1002/ejoc.202400437

Organocatalytic Cascade β-Functionalization/Aromatization of Pyrrolidines via Double Hydride Transfer

Lan Zhou, Xiao-De An, Shuo Yang, Xian-Jiang Li, Chang-Lun Shao, Qing Liu and Jian Xiao

Org. Lett., 2020, 22, 776
DOI: 10.1021/acs.orglett.9b03918

Fermentation: A Boon for Production of Bioactive Compounds by Processing of Food Industries Wastes (By-Products)

Pardeep Kumar Sadh, Suresh Kumar, Prince Chawla and Joginder Singh Duhan

Molecules, 2018, 23, 2560
DOI: 10.3390/molecules23102560

Modular Synthesis of Highly Substituted 3-Azapyrroles by Rh(II)-Catalyzed N–H Bond Insertion and Cyclodehydration

Matthew B. Williams and Alistair Boyer

J. Org. Chem., 2022, 87, 16139
DOI: 10.1021/acs.joc.2c00434

Ascorbic acid as a multifunctional hydrogen bonding catalyst for Paal–Knorr synthesis of N-substituted mono- and bis-pyrroles: experimental and theoretical aspects

Amin Ghaemi, Hossein Reza Darabi, Kioumars Aghapoor, Farshid Mohsenzadeh, Hani Sayahi, Hossein Taherzadeh, Maryam Farajpour Mojdehi, Yadollah Balavar and Hossein Farhangian

Res Chem Intermed, 2023, 49, 4087
DOI: 10.1007/s11164-023-05072-w

Catalyst-Free Annulation of Acylethynylpyrroles with 1-Pyrrolines: A Straightforward Access to Tetrahydrodipyrrolo[1,2-a:1′,2′-c]imidazoles

Ludmila A. Oparina, Kseniya V. Belyaeva, Nikita A. Kolyvanov, Igor A. Ushakov, Maxim D. Gotsko, Lyubov’ N. Sobenina, Alexander V. Vashchenko and Boris A. Trofimov

J. Org. Chem., 2022, 87, 9518
DOI: 10.1021/acs.joc.2c00476

Benzimidazole-functionalized PEPPSI type Pd(II)NHC complexes bearing nitrophenylethyl and hidroxyphenylethyl group: Synthesis, characterization, crystal structure and it's catalytic activity on direct arylation reaction

Tuba Çağlılar, Ayten Behçet, Duygu Barut Celepci, Aydın Aktaş, Yetkin Gök and Muhittin Aygün

Journal of Molecular Structure, 2021, 1246, 131137
DOI: 10.1016/j.molstruc.2021.131137

Pyrrole-containing hybrids as potential anticancer agents: An insight into current developments and structure-activity relationships

Li Long, Han Zhang, ZhiHui Zhou, Lei Duan, Dang Fan, Ran Wang, Shan Xu, Dan Qiao and Wufu Zhu

European Journal of Medicinal Chemistry, 2024, 273, 116470
DOI: 10.1016/j.ejmech.2024.116470

Catalytic Enantioselective Hetero-[6+4] and -[6+2] Cycloadditions for the Construction of Condensed Polycyclic Pyrroles, Imidazoles, and Pyrazoles

Giulio Bertuzzi, Mathias Kirk Thøgersen, Maxime Giardinetti, Andreu Vidal-Albalat, Adam Simon, K. N. Houk and Karl Anker Jørgensen

J. Am. Chem. Soc., 2019, 141, 3288
DOI: 10.1021/jacs.8b13659

Copper-Promoted Regioselective Synthesis of Polysubstituted Pyrroles from Aldehydes, Amines, and Nitroalkenes via 1,2-Phenyl/Alkyl Migration

Dimitrios Andreou, Michael G. Kallitsakis, Edward Loukopoulos, Catherine Gabriel, George E. Kostakis and Ioannis N. Lykakis

J. Org. Chem., 2018, 83, 2104
DOI: 10.1021/acs.joc.7b03051

Nanocrystalline ZnO: A Competent and Reusable Catalyst for the Preparation of Pharmacology Relevant Heterocycles in the Aqueous Medium

Moumita Saha and Asish R. Das

CGC, 2020, 7, 53
DOI: 10.2174/2213346107666200218122718

Synthesis of Dihydropyrrolizine and Tetrahydroindolizine Scaffolds from Pyrroles by Titanocene(III) Catalysis

Sven Hildebrandt and Andreas Gansäuer

Angewandte Chemie, 2016, 128, 9871
DOI: 10.1002/ange.201603985

Total synthesis of (±) aspidostomide B, C, regioisomeric N-methyl aspidostomide D and their derivatives

Mulla Althafh Hussain and Faiz Ahmed Khan

Tetrahedron Letters, 2019, 60, 151040
DOI: 10.1016/j.tetlet.2019.151040

Direct Multicomponent Synthesis of C3-Arylated Pyrroles under Catalyst-Free Conditions

Amol Prakash Pawar, Reena Jangir, Atul Jankiram Dolas, Yadav Kacharu Nagare, Krishnan Rangan, Eldhose Iype and Indresh Kumar

Synthesis, 2025, 57, 380
DOI: 10.1055/a-2380-3855

Experimental and Theoretical Investigation of Triethylamine Hydrochloride Solubility in Acetonitrile–Dimethyl Carbonate Mixtures

Junfeng Teng, Fang Zong, Lili Wang, Xiaoyan Sun and Shuguang Xiang

J Solution Chem, 2025, 54, 817
DOI: 10.1007/s10953-025-01444-5

Synthesis of Substituted Pyrrolo[2,3‐c]Pyrazol‐4‐Ylacetic Acids via Acid‐Catalyzed Rearrangement of Aroyl‐Containing Pyrazolo[3,4‐b]Pyridin‐6‐Ones

Ekaterina N. Kudryavtseva, Anna A. Zholtovskaya and Boris V. Lichitsky

Journal of Heterocyclic Chem, 2026
DOI: 10.1002/jhet.70182

Dendritic Amine on Mesoporous Silica: First Organo Base Catalyst for Paal Knorr Reaction under Solvent Free Condition, A green approach

K. A. Jisha and K. Sreekumar

Catal Lett, 2017, 147, 964
DOI: 10.1007/s10562-017-1975-y

Photoabsorption and Photoionization Cross-Sections and Asymmetry Parameters of Pyrrole in the Vacuum-Ultraviolet Energy Range

Mariana B. M. S. Medeiros, Josenilton N. Sousa, Manuela S. Arruda, Milton M. Fujimoto, Manoel G. P. Homem, Helder K. Tanaka, Bruno Credidio, Ricardo R. T. Marinho and Frederico V. Prudente

ACS Phys. Chem Au, 2025, 5, 254
DOI: 10.1021/acsphyschemau.4c00101

Recent advances in the construction of axially chiral arylpyrroles

Yang-Bo Chen, Ye-Nan Yang, Xuan-Zhu Huo, Long-Wu Ye and Bo Zhou

Sci. China Chem., 2023, 66, 2480
DOI: 10.1007/s11426-023-1671-y

Synthesis and Rh-catalyzed reductive cyclization of 1,6-enynes and 1,6-diynes containing alkynylboronate termini

Christopher J. Pell and Oleg V. Ozerov

Journal of Organometallic Chemistry, 2020, 912, 121143
DOI: 10.1016/j.jorganchem.2020.121143

Recent developments by zinc based reagents/catalysts promoted organic transformations

Shaik Ghouse, Chinnabattigalla Sreenivasulu, Dakoju Ravi Kishore and Gedu Satyanarayana

Tetrahedron, 2022, 105, 132580
DOI: 10.1016/j.tet.2021.132580

A short review on the synthesis of pyrrolo[3,4-c]coumarins an isolamellarin-B scaffolds

Prasanta Patra

Synthetic Communications, 2022, 52, 1999
DOI: 10.1080/00397911.2022.2119413

Gold‐Catalyzed Cyclization of Yndiamides with Isoxazoles via α‐Imino Gold Fischer Carbenes

Zixuan Tong, Philip J. Smith, Helena D. Pickford, Kirsten E. Christensen and Edward A. Anderson

Chemistry A European J, 2023, 29
DOI: 10.1002/chem.202302821

Heterocyclic and heteropolycyclic moieties in organic hole transport materials for perovskite solar cells: Design, synthesis, and performance

Shakil N. Afraj, Arulmozhi Velusamy, Ming-Chou Chen, Marwa Abd-Ellah and Ahmed L. Abdelhady

Coordination Chemistry Reviews, 2025, 532, 216500
DOI: 10.1016/j.ccr.2025.216500

Proteinase resistance of carnosine, pyrrolylcarnosine, and salicylcarnosine

K. V. Shevchenko, I. Yu. Nagaev, O. I. Kulikova, S. L. Stvolinsky, V. P. Shevchenko and N. F. Myasoedov

RUBI, 2024, 50
DOI: 10.31857/S0132342324020042

Microwave‐Assisted Synthesis of N‐Substituted‐2,5‐dihydro‐1H‐pyrroles and N‐Substituted‐1H‐pyrroles in Water

Thiago M. De Souza, Lothar W. Bieber, Ricardo L. Longo and Ivani Malvestiti

ChemistrySelect, 2018, 3, 34
DOI: 10.1002/slct.201702325

Visible Light‐Induced [3+2] Annulation Reaction of Alkenes with Vinyl Azides: Direct Synthesis of Functionalized Pyrroles

Ming Yang, Xin‐Yu Wang, Jie Wang and Yu‐Long Zhao

Chin. J. Chem., 2024, 42, 151
DOI: 10.1002/cjoc.202300498

Reactivity of terminal imido complexes of group 4–6 metals: Stoichiometric and catalytic reactions involving cycloaddition with unsaturated organic molecules

Kento Kawakita, Bernard F. Parker, Yuya Kakiuchi, Hayato Tsurugi, Kazushi Mashima, John Arnold and Ian A. Tonks

Coordination Chemistry Reviews, 2020, 407, 213118
DOI: 10.1016/j.ccr.2019.213118

Identification of antibacterial metabolites produced by a marine bacterium Halobacillus marinus HMALI004

Sardar Ali, Runlin Cai, Hao Feng, Jianmin Xie, Yueling Zhang and Hui Wang

Journal of Applied Microbiology, 2022, 133, 3030
DOI: 10.1111/jam.15764

Synthesis of 3-[(4-Nitrophenyl)thio]-Substituted 4-Methylene-1-pyrrolines from N-Propargylic β-Enaminones

Esra Korkmaz and Metin Zora

J. Org. Chem., 2020, 85, 4937
DOI: 10.1021/acs.joc.0c00109

Marine Pyrrole Alkaloids

Kevin Seipp, Leander Geske and Till Opatz

Marine Drugs, 2021, 19, 514
DOI: 10.3390/md19090514

[3+2] Cycloaddition of Tosylmethyl Isocyanide with Styrylisoxazoles: Facile Access to Polysubstituted 3-(Isoxazol-5-yl)pyrroles

Xueming Zhang, Xianxiu Xu and Dawei Zhang

Molecules, 2017, 22, 1131
DOI: 10.3390/molecules22071131

Efficient [Cu(NHC)]‐Catalyzed Multicomponent Synthesis of Pyrroles

Tuan Thanh Dang and Abdul Majeed Seayad

Chemistry An Asian Journal, 2017, 12, 2383
DOI: 10.1002/asia.201701045

Solvent Free Synthesis of N-Substituted Pyrrole Derivatives Catalyzed by Silica Sulfuric Acid

A. J. Khammas, C. Yolacan and F. Aydogan

Russ J Gen Chem, 2018, 88, 2680
DOI: 10.1134/S1070363218120332

New pentasubstituted pyrrole hybrid atorvastatin–quinoline derivatives with antiplasmodial activity

Rita C.C. Carvalho, Wagner A. Martins, Tayara P. Silva, Carlos R. Kaiser, Mônica M. Bastos, Luiz C.S. Pinheiro, Antoniana U. Krettli and Núbia Boechat

Bioorganic & Medicinal Chemistry Letters, 2016, 26, 1881
DOI: 10.1016/j.bmcl.2016.03.027

Synthesis and evaluation of novel spiro derivatives for pyrrolopyrimidines as anti-hyperglycemia promising compounds

Samar Said Fatahala, Shahenda Mahgub, Heba Taha and Rania Helmy Abd-El Hameed

Journal of Enzyme Inhibition and Medicinal Chemistry, 2018, 33, 809
DOI: 10.1080/14756366.2018.1461854

Combining NMR and MS to Describe Pyrrole-2-Carbaldehydes in Wheat Bran of Radiation

Yun-Seo Kil, Ananda Baral, Byeong-Seon Jeong, Pekka Laatikainen, Yang Liu, Ah-Reum Han, Min-Jeong Hong, Jin-Baek Kim, Hyukjae Choi, Pil-Hoon Park and Joo-Won Nam

J. Agric. Food Chem., 2022, 70, 13002
DOI: 10.1021/acs.jafc.2c04771

Mass Spectra of New Heterocycles: XXII. Electron Impact and Chemical Ionization of 1-Alkyl(cycloalkyl, alkoxyalkyl)-5-[(alkyl, allyl, benzyl)sulfanyl]-1H-pyrrol-2-amines

L. V. Klyba, N. A. Nedolya, E. R. Sanzheeva and O. A. Tarasova

Russ J Org Chem, 2021, 57, 347
DOI: 10.1134/S1070428021030040

Efficient One-Pot, Three-Step Synthesis of 1,2,3,5-Tetrasubstituted Pyrroles via Aza-Michael Addition of Methyl 3-Iminoacrylates

Michiyasu Nakao, Shigeki Sano, Ken Horikoshi and Syuji Kitaike

HETEROCYCLES, 2023, 106, 1397
DOI: 10.3987/COM-23-14876

Volatile Nitrogenous Compounds from Bacteria: Source of Novel Bioactive Compounds

Camilla A. S. Valença, Ana A. T. Barbosa, Eliana B. Souto, Elina B. Caramão and Sona Jain

Chemistry & Biodiversity, 2021, 18
DOI: 10.1002/cbdv.202100549

Access to Pyrrolocoumarins through DBU‐Mediated Coupling of 2‐Oxo‐2H‐chromene‐3‐carbaldehydes and Phenacyl Azides

Lodsna Borkotoky, Satheesh Borra and Ram Awatar Maurya

Eur J Org Chem, 2022, 2022
DOI: 10.1002/ejoc.202101237

Elucidation of Chalkophomycin Biosynthesis Reveals N-Hydroxypyrrole-Forming Enzymes

Anne Marie Crooke, Anika K. Chand, Zheng Cui and Emily P. Balskus

J. Am. Chem. Soc., 2024, 146, 16268
DOI: 10.1021/jacs.4c04712

First‐Row Transition‐Metal Catalyzed Acceptorless Dehydrogenation and Related Reactions: A Personal Account

Murugan Subaramanian, Ganesan Sivakumar and Ekambaram Balaraman

The Chemical Record, 2021, 21, 3839
DOI: 10.1002/tcr.202100165

Examination of Triazolinedione-Derived Dihydropyrrole Hybrid Compounds: ER Stress-Related Apoptosis in Breast Cancer Cells, Molecular Docking, and ADMET Analysis

Seda Mesci, Arif Ayar, Burak Yazgan, Melek Gul and Tuba Yıldırım

MC, 2025, 21, 707
DOI: 10.2174/0115734064328727240911112815

Silver-Catalyzed Domino Reaction of CF3-Substituted N-Allenamides with Primary Amines for the Construction of 2-Amido-5-fluoropyrroles

Maxime Hourtoule and Laurence Miesch

Org. Lett., 2023, 25, 1727
DOI: 10.1021/acs.orglett.3c00401

Effect of Temperature during Preactivation of 5% Pd/C and 5% Pd/Al2O3 with Deuterium Gas on the Isotope Exchange between Deuterium Water and an Organic Compound

V. P. Shevchenko, I. Yu. Nagaev, K. V. Shevchenko, L. A. Andreeva and N. F. Myasoedov

Radiochemistry, 2025, 67, 89
DOI: 10.1134/S1066362225010126

Synthesis of 1,4‐Diketones from β‐Oxo Esters and Enol Acetates by Cerium‐Catalyzed Oxidative Umpolung Reaction

Irina Geibel and Jens Christoffers

Eur J Org Chem, 2016, 2016, 918
DOI: 10.1002/ejoc.201600057

Torsions of N-methylpyrrole and its cation

Alexander R. Davies, David J. Kemp and Timothy G. Wright

Chemical Physics Letters, 2021, 763, 138227
DOI: 10.1016/j.cplett.2020.138227

Recent Advances for the Synthesis of N‐Unsubstituted Pyrroles

Ilya V. Efimov, Larisa N. Kulikova, Almira R. Miftyakhova, Maria D. Matveeva and Leonid G. Voskressensky

ChemistrySelect, 2021, 6, 13740
DOI: 10.1002/slct.202103486

Deprotection and Functionalization of Protective N‐Heterocycles Under Mild Conditions

Wenjing Liu, Zixuan Tan, Qianyu Zhang and Feng Zhao

Eur J Org Chem, 2025, 28
DOI: 10.1002/ejoc.202500165

Structural Determination of Ruthenium Complexes Containing Bi-Dentate Pyrrole-Ketone Ligands

Ya-Wen Tsai, Yun-Fan Chen, Yong-Jie Li, Kuan-Hung Chen, Chia-Her Lin and Jui-Hsien Huang

Molecules, 2018, 23, 159
DOI: 10.3390/molecules23010159

Iodine‐Catalyzed Synthesis of Pyrrolo(2,3‐c)coumarin Derivatives Using 3‐Aminocoumarins, Arylglyoxals and 4‐Hydroxycoumarin through One‐Pot Three‐Component Reaction

Md. Belal and Abu T. Khan

ChemistrySelect, 2018, 3, 2431
DOI: 10.1002/slct.201702629

One‐Pot Synthesis of Polysubstituted Pyrroles via Sequential Ketenimine Formation/Ag(I)‐Catalyzed Alkyne Cycloisomerisation Starting from Ylide Adducts

Jun Xiong, Zhi‐Ying Mu, Gang Yao, Jia‐An Zhang, Qi‐Xun Feng, Hui‐Ting He, Yong‐Long Pang, Hang Shi and Ming‐Wu Ding

Chin. J. Chem., 2021, 39, 1553
DOI: 10.1002/cjoc.202000639

Practical Synthesis of Pharmaceutically Relevant Pyrroles from α,β‐Unsaturated Aldehydes and Phenacyl Azides

Lodsna Borkotoky and Ram Awatar Maurya

Eur J Org Chem, 2023, 26
DOI: 10.1002/ejoc.202300822

New Derivative of Pyrrole and Carnosine: Synthesis, Physicochemical Properties, and Biological Acivity

T. N. Fedorova, O. I. Kulikova, V. A. Migulin, O. A. Muzychuk, D. A. Abaimov and S. L. Stvolinsky

Pharm Chem J, 2024, 58, 617
DOI: 10.1007/s11094-024-03185-z

Depolymerization of tubulin as the main molecular mechanism of the cytotoxic and antitumor activity of pyrrole-containing heterocyclic compounds

A. R. Galembikova, P. D. Dunaev, T. V. Ivoilova, A. I. Gilyazova, A. E. Galyautdinova, E. G. Mikheeva, S. S. Zykova, N. M. Igidov, P. B. Kopnin and S. V. Boichuk

Advances in Molecular Oncology, 2024, 11, 130
DOI: 10.17650/2313-805X-2024-11-2-130-146

Functionalized Bipyrroles and Pyrrolyl-Aminopyrones from Acylethynylpyrroles and Diethyl Aminomalonate

Maxim D. Gotsko, Ivan V. Saliy, Lyubov N. Sobenina, Igor A. Ushakov, Victoriya V. Kireeva and Boris A. Trofimov

Synthesis, 2022, 54, 1134
DOI: 10.1055/a-1681-4164

Novel N-Arylaminophosphonates Bearing a Pyrrole Moiety and Their Ecotoxicological Properties

Jarosław Lewkowski, Marta Morawska, Anna Kaczmarek, Diana Rogacz and Piotr Rychter

Molecules, 2017, 22, 1132
DOI: 10.3390/molecules22071132

Multicomponent Methanolysis Reaction for the Synthesis Pyrrole and Pyrolizine Derivatives via Intermolecular (3 + 2) Cycloaddition

Prashishkumar K. Shirsat, Navnath B. Khomane, Prakash R. Mali, Raghavender Reddy Maddi, Jagadeesh Babu Nanubolu and Harshadas M. Meshram

ChemistrySelect, 2017, 2, 11218
DOI: 10.1002/slct.201702729

Nickel-catalyzed formal [3 + 2]-cycloaddition of 2H-azirines with 1,3-dicarbonyl compounds for the synthesis of pyrroles

Mi-Na Zhao, Gui-Wan Ning, De-Suo Yang, Peng Gao, Ming-Jin Fan and Li-Fang Zhao

Tetrahedron Letters, 2020, 61, 152319
DOI: 10.1016/j.tetlet.2020.152319

Microwave-assisted multicomponent reactions in heterocyclic chemistry and mechanistic aspects

Shivani Gulati, Stephy Elza John and Nagula Shankaraiah

Beilstein J. Org. Chem., 2021, 17, 819
DOI: 10.3762/bjoc.17.71

Phytotoxicity, cytotoxicity, and in vivo antifungal efficacy of chitosan nanobiocomposites on prokaryotic and eukaryotic cells

Alma Carolina Gálvez-Iriqui, Joel Said García-Romo, Mario Onofre Cortez-Rocha, Armando Burgos-Hernández, María Guadalupe Burboa-Zazueta, Ana Guadalupe Luque-Alcaraz, Montserrat Calderón-Santoyo, Waldo Manuel Argüelles-Monal and Maribel Plascencia-Jatomea

Environ Sci Pollut Res, 2021, 28, 3051
DOI: 10.1007/s11356-020-10716-0

Synthesis of new indolylpyrrole derivatives via a four-component domino reaction between arylglyoxals, acetylacetone, indole and aliphatic amines in aqueous media

Fereshteh Mousavizadeh, Mahdiyeh Talebizadeh and Mohammad Anary-Abbasinejad

Tetrahedron Letters, 2018, 59, 2970
DOI: 10.1016/j.tetlet.2018.06.043

Arylation and Alkyne Insertion to C-Acylimines: Rapid Access to 2-Trifluoromethylated and Other Fully Substituted Pyrroles in One Pot

Srinivasarao Yaragorla, Arun Doma and Rajeshwari Tangellapally

Synthesis, 2023, 55, 1298
DOI: 10.1055/s-0042-1751407

Synthesis, Characterization, Antimicrobial and Anticancer Activity of New Bidentate Schiff Base Ligand and their Transition Metal(II) Complexes

S. Arulmozhi, G. Sasikumar, A. Subramani, A. Sudha and S.J. Askar Ali

Asian J. Chem., 2021, 33, 1488
DOI: 10.14233/ajchem.2021.23171

Direct Synthesis of Pyrroles by Dehydrogenative Coupling of Diols and Amines Catalyzed by Cobalt Pincer Complexes

Prosenjit Daw, Subrata Chakraborty, Jai Anand Garg, Yehoshoa Ben‐David and David Milstein

Angew Chem Int Ed, 2016, 55, 14373
DOI: 10.1002/anie.201607742

β-Cyclodextrin as an Efficient and Recyclable Supramolecular Catalyst for the Synthesis of Heterocyclic Compounds

Mohsen Abbasi

Journal of the Chinese Chemical Society, 2017, 64, 896
DOI: 10.1002/jccs.201600887

3,4-Dihydro-2H-pyrrole-2-carbonitriles: Useful Intermediates in the Synthesis of Fused Pyrroles and 2,2′-Bipyrroles

Marco M. Nebe, Murat Kucukdisli and Till Opatz

J. Org. Chem., 2016, 81, 4112
DOI: 10.1021/acs.joc.6b00393

Synthesis and spectroscopic properties of rotamers in the series of 2-(fluoroaryl)-4-substituted pyrroles

Almira R. Miftyakhova, Maria D. Matveeva, Dmitry I. Zhilyaev, Oleg S. Eltsov, Giovanni Talarico, Alexander F. Smol'yakov, Leonid G. Voskressensky and Ilya V. Efimov

Journal of Fluorine Chemistry, 2021, 249, 109863
DOI: 10.1016/j.jfluchem.2021.109863

Evaluating Pigments as a Biosignature: Abiotic/Prebiotic Synthesis of Pigments and Pigment Mimics in Planetary Environments

Laura E. Rodriguez, Jessica M. Weber and Laura M. Barge

Astrobiology, 2024, 24, 767
DOI: 10.1089/ast.2023.0006

Quantum Mechanical Spectral Analysis and Aldose Reductase Inhibition Evaluation of Synthetic New Pyrrolopyrazinones

Yun-Seo Kil, Junhyeung Park, Byeong-Seon Jeong, Punam Thapa, Young Jun Ok, Hyukjae Choi, Jee-Heon Jeong and Joo-Won Nam

ACS Omega, 2025, 10, 13185
DOI: 10.1021/acsomega.4c10696

Copper-Catalyzed Oxidative Cyclization of Maleimides with Amines and Alkyne Esters: Direct Access to Fully Substituted Dihydropyrroles and Pyrrole Derivatives

Jia-Nan Zhu, Lei-Lei Chen, Run-Xiang Zhou, Bo Li, Zhi-Yu Shao and Sheng-Yin Zhao

Org. Lett., 2017, 19, 6044
DOI: 10.1021/acs.orglett.7b02670

Modular Synthesis of Tetrasubstituted Pyrroles through a Four-Component Cyclization Strategy Using Ammonium Salt as the Nitrogen Source

Chunlan Zhou, Haolin Zheng, Ya Chen, Guojiang Mao and Guo-Jun Deng

J. Org. Chem., 2023, 88, 1533
DOI: 10.1021/acs.joc.2c02556

Synthesis of symmetrical and unsymmetrical 1,3-diheteroarylbenzenes through palladium-catalyzed direct arylation of benzene-1,3-disulfonyl dichloride and 3-bromobenzenesulfonyl chlorides

Imane Idris, Fazia Derridj, Safia Djebbar, Jean-François Soulé and Henri Doucet

Tetrahedron, 2015, 71, 9617
DOI: 10.1016/j.tet.2015.10.082

Complexities of the Interaction of NiII, PdII and PtII Pyrrole‐Imine Chelates with Human Serum Albumin**

Sheldon Sookai and Orde Q. Munro

ChemistryEurope, 2023, 1
DOI: 10.1002/ceur.202300012

Understanding nonlinear molecular responses in highly inhomogeneous electric fields: Insights from imidazole and pyrrole

G. F. Quinteiro Rosen, V. Manzoni, R. M. Gester, A. R. Cunha, G. I. Pagola and P. F. Provasi

The Journal of Chemical Physics, 2025, 162
DOI: 10.1063/5.0253042

A new pyrrole based small molecule from Tinospora cordifolia induces apoptosis in MDA-MB-231 breast cancer cells via ROS mediated mitochondrial damage and restoration of p53 activity

K.C. Rashmi, M. Harsha Raj, Manoj Paul, Kesturu S. Girish, Bharathi P. Salimath and H.S. Aparna

Chemico-Biological Interactions, 2019, 299, 120
DOI: 10.1016/j.cbi.2018.12.005

Copper-Catalyzed One-Pot Cascade Reactions of CF3CHN2, Nitriles, and Alkenes: Chemo- and Regioselective Access to 2-(Trifluoromethyl)pyrroles

Chun-Hui Zhang, Zhi-Yuan Tao, Fa-Guang Zhang, Jing Nie and Jun-An Ma

J. Org. Chem., 2025, 90, 10369
DOI: 10.1021/acs.joc.5c01067

Regioselective Synthesis of Highly Functionalized 2H-Pyrroles via Dearomative Chlorination of 1H-Pyrroles

Victoria E. Shambalova, Roman V. Larkovich, Alexander S. Aldoshin, Konstantin A. Lyssenko, Mikhail S. Nechaev and Valentine G. Nenajdenko

J. Org. Chem., 2024, 89, 11394
DOI: 10.1021/acs.joc.4c01099

Diversity‐Oriented Synthesis of Complex Pyrrole‐Based Architectures from Very Simple Starting Materials

Marco Leonardi, Verónica Estévez, Mercedes Villacampa and J. Carlos Menéndez

Adv Synth Catal, 2019, 361, 2054
DOI: 10.1002/adsc.201900044

Recent Strides in the Transition Metal-Free Cross-Coupling of Haloacetylenes with Electron-Rich Heterocycles in Solid Media

Lyubov’ N. Sobenina and Boris A. Trofimov

Molecules, 2020, 25, 2490
DOI: 10.3390/molecules25112490

PrVO4/SnD NPs as a Nanocatalyst for Carbon Dioxide Fixation to Synthesis Benzimidazoles and 2-Oxazolidinones

Zemin He, Ping Yu, Yuzhen Zhao, Huimin Zhang, Yongming Zhang, Xiaoxi Kang, Haiquan Zhang and Seyed Mohsen Sadeghzadeh

Catal Lett, 2021, 151, 1623
DOI: 10.1007/s10562-020-03410-w

In silico and in vitro assessment of anti-Trypanosoma cruzi efficacy, genotoxicity and pharmacokinetics of pentasubstituted pyrrolic Atorvastatin-aminoquinoline hybrid compounds

Carlos Fernando Araujo-Lima, Rita de Cássia Castro Carvalho, Raiza Brandão Peres, Ludmila Ferreira de Almeida Fiuza, Bárbara Verena Dias Galvão, Frederico S. Castelo-Branco, Mônica Macedo Bastos, Nubia Boechat, Israel Felzenszwalb and Maria de Nazaré Correia Soeiro

Acta Tropica, 2023, 242, 106924
DOI: 10.1016/j.actatropica.2023.106924

Finding of antibiotic compounds pyrrolo [1,2-a]pyrazine-1,4-dione, hexahydro and Cyclo(prolyl-tyrosyl) isolated from the degradation of epoxy

V. Vikram and N. Hariram

Environmental Technology, 2025, 46, 2064
DOI: 10.1080/09593330.2024.2419560

Direct and Selective 3-Amidation of Indoles Using Electrophilic N-[(Benzenesulfonyl)oxy]amides

Gerardo X. Ortiz, Brett N. Hemric and Qiu Wang

Org. Lett., 2017, 19, 1314
DOI: 10.1021/acs.orglett.7b00358

Regioselective Olefination of 3‐Substituted Five‐Membered Heteroarenes

Hao Chen, Mirxan Farizyan and Manuel van Gemmeren

Eur J Org Chem, 2020, 2020, 6318
DOI: 10.1002/ejoc.202000659

Single‐Electron‐Transfer‐Initiated Sequential Direct Arylation Reaction of Pyrrole with Aryl Diazonium Salts

Eiji Yamaguchi, Yayoi Kashima and Akichika Itoh

Asian J Org Chem, 2019, 8, 324
DOI: 10.1002/ajoc.201800738

Ab initio kinetic mechanism of OH-initiated atmospheric oxidation of pyrrole

Tam V.-T. Mai, Hieu T. Nguyen and Lam K. Huynh

Chemosphere, 2021, 263, 127850
DOI: 10.1016/j.chemosphere.2020.127850

Organocatalytic Enantioselective Friedel‐Crafts Alkylation Reactions of Pyrroles

Daniel Gaviña, Marcos Escolano, Javier Torres, Gloria Alzuet‐Piña, María Sánchez‐Roselló and Carlos del Pozo

Adv Synth Catal, 2021, 363, 3439
DOI: 10.1002/adsc.202100313

Copper Catalyzed Heteroannelation Reaction between 4‐Thiazolidinones and O‐Acetyl Oximes to Synthesize 2,5‐Diphenyl‐3‐(Pyrimidin‐2‐yl)‐3,4‐Dihydro‐2H‐Pyrrolo‐[2,3‐d]‐Thiazole

Parth P. Patel and Kishor H. Chikhalia

ChemistrySelect, 2024, 9
DOI: 10.1002/slct.202402137

An efficient and facile access to highly functionalized pyrrole derivatives

Meng Gao, Wenting Zhao, Hongyi Zhao, Ziyun Lin, Dongfeng Zhang and Haihong Huang

Beilstein J. Org. Chem., 2018, 14, 884
DOI: 10.3762/bjoc.14.75

Fused Pyrroles in Cholestane and Norcholestane Side Chains: Acaricidal and Plant Growth-Promoting Effects

María G. De los Santos, Marcos Cua-Basulto, Anallely Huepalcalco, Wendy Delit, Jesús Sandoval-Ramírez, Adolfo López-Torres, Esaú Ruiz-Sánchez and María A. Fernández-Herrera

Molecules, 2022, 27, 8466
DOI: 10.3390/molecules27238466

Mass Spectra of New Heterocycles: XXIII. Electron Impact and Chemical Ionization Study of 5-[(Cyanomethyl)sulfanyl]- and 5-[(1,3-Dioxolan-2-ylmethyl)sulfanyl]-1H-pyrrol-2-amines

L. V. Klyba, N. A. Nedolya, E. R. Sanzheeva and O. A. Tarasova

Russ J Org Chem, 2021, 57, 1901
DOI: 10.1134/S1070428021120022

Sterically Controlled C−H Olefination of Heteroarenes

Hao Chen, Mirxan Farizyan, Francesca Ghiringhelli and Manuel van Gemmeren

Angewandte Chemie, 2020, 132, 12311
DOI: 10.1002/ange.202004521

Nano ordered polyacrylonitrile-grafted chitosan as a robust biopolymeric catalyst for efficient synthesis of highly substituted pyrrole derivatives

Mahsa Zohrehvand, Niloufar Nashibi, Mohammad G. Dekamin and Afshin Sarvary

Sci Rep, 2025, 15
DOI: 10.1038/s41598-025-05504-0

Synthesis of Polysubstituted Pyrroles via Silver-Catalyzed Oxidative Radical Addition of Cyclopropanols to Imines

Yulu Zhou, Mingchang Wu, Yi Liu, Cungui Cheng and Gangguo Zhu

Org. Lett., 2020, 22, 7542
DOI: 10.1021/acs.orglett.0c02735

Recent advances in the tandem annulation of 1,3-enynes to functionalized pyridine and pyrrole derivatives

Yi Liu, Puying Luo, Yang Fu, Tianxin Hao, Xuan Liu, Qiuping Ding and Yiyuan Peng

Beilstein J. Org. Chem., 2021, 17, 2462
DOI: 10.3762/bjoc.17.163

tert-Butyl Nitrite Promoted Oxidative Intermolecular Sulfonamination of Alkynes to Synthesize Substituted Sulfonyl Pyrroles from the Alkynylamines and Sulfinic Acids

Zhenjie Qi, Yong Jiang, Yanyan Wang and Rulong Yan

J. Org. Chem., 2018, 83, 8636
DOI: 10.1021/acs.joc.8b00741

Synthesis of 2-trifluoromethylated 3-pyrrolines/pyrrolidines via [3+2] cycloaddition of azomethine ylides with the participation of 3,3,3-trifluoroalanine

Qian Liu, Isao Yoshikawa and Kazuaki Kudo

Journal of Fluorine Chemistry, 2022, 264, 110061
DOI: 10.1016/j.jfluchem.2022.110061

Synthesis and Thermodynamic Parameters of Phase Transitions of 3-(1-R-5-Phenyl-1H-Pyrrol-2-yl)propanoic Acid Derivatives

Dmytro Shevchenko, Yuriy Horak, Nadiia Tyschenko, Dariia Kichura, Mykola Obushak and Iryna Sobechko

ChChT, 2025, 19, 403
DOI: 10.23939/chcht19.03.403

Domino Reaction for the Synthesis of Polysubstituted Pyrroles and Lamellarin R

Jih Ru Hwu, Animesh Roy, Avijit Panja, Wen-Chieh Huang, Yu-Chen Hu, Kui-Thong Tan, Chun-Cheng Lin, Kuo-Chu Hwang, Ming-Hua Hsu and Shwu-Chen Tsay

J. Org. Chem., 2020, 85, 9835
DOI: 10.1021/acs.joc.0c01134

Synthesis of Diverse Pentasubstituted Pyrroles by a Gold(I)-Catalyzed Cascade Rearrangement-Cyclization of Tertiary Enamide

Wenzhong Li, Ran Shi, Sen Chen, Xuesi Zhang, Wei Peng, Si Chen, Jiazhu Li, Xin-Ming Xu, Yan-Ping Zhu and Xueyuan Wang

J. Org. Chem., 2022, 87, 3014
DOI: 10.1021/acs.joc.1c02837

Synthesis of Densely Functionalized Pyrroles via Photoinduced C-Insertion into N-Alkylenamines: Sequential C(sp2)–H/C(sp3)–H Activation with Bromine Radicals

Chuan-Hua Qu, Su-Ya Liu, Shan-Shan Chen, Nian Wang, Ying Cheng, Shi-You Xue, Xue-Ying Yang, Wen-Bin Zong, Yuan Zhou, Li-Min Zhang, Xiang-Yi Zeng, Qin-Mao Li, Lan-Bin He, Xiao Yan and Gui-Ting Song

Org. Lett., 2025, 27, 11264
DOI: 10.1021/acs.orglett.5c03559

Potassium Acetate-Catalyzed Double Decarboxylative Transannulation To Access Highly Functionalized Pyrroles

Jun-Kuan Li, Biying Zhou, Yu-Chen Tian, Chunman Jia, Xiao-Song Xue, Fa-Guang Zhang and Jun-An Ma

Org. Lett., 2020, 22, 9585
DOI: 10.1021/acs.orglett.0c03621

Organo-photoredox-Catalyzed Selective Mono- and Bis-C–H Alkylation of Electron-Rich (Hetero)Arenes

Shyamal Pramanik, Partha Pratim Mondal and Soumitra Maity

J. Org. Chem., 2023, 88, 15256
DOI: 10.1021/acs.joc.3c01757

Design, Synthesis, Biological Evaluation and SARs of Anthranilic Diamide Derivatives Containing Pyrrole Moieties

Yangyang Zhao, Huangong Li, Pengwei Sun, Li Gao, Sha Zhou, Lixia Xiong, Na Yang, Yuxin Li and Zhengming Li

Chem. Res. Chin. Univ., 2020, 36, 1168
DOI: 10.1007/s40242-020-0237-5

Copper-Catalyzed Cycloisomerization of Cyclopropenylimine for Synthesis of Pyrroles

Keiji Konishi, Norihiko Takeda, Motohiro Yasui, Haruo Matsuzaki, Okiko Miyata and Masafumi Ueda

J. Org. Chem., 2019, 84, 14320
DOI: 10.1021/acs.joc.9b02178

Bacillus licheniformis strain POT1 mediated polyphenol biosynthetic pathways genes activation and systemic resistance in potato plants against Alfalfa mosaic virus

Ahmed Abdelkhalek, Abdulaziz A. Al-Askar and Said I. Behiry

Sci Rep, 2020, 10
DOI: 10.1038/s41598-020-72676-2

Regioselective Alkenylation of Five-Membered Heteroarenes via a Dual 1,3-Sulfur Rearrangement

Jia Li, Mingming Mao, Kang Dong, Rui-Peng Li, Xi Chen and Shouchu Tang

Org. Lett., 2023, 25, 4782
DOI: 10.1021/acs.orglett.3c01357

Synthesis, Hydrolytic Stability and In Vivo Biological Study of Bioconjugates of the Tetrapeptides FELL Containing Pyrrole Moiety

Boryana Borisova, Stanislava Vladimirova, Hristina Nocheva, Marie Laronze-Cochard, Stéphane Gérard, Stoyko Petrin and Dancho Danalev

Biomedicines, 2023, 11, 3265
DOI: 10.3390/biomedicines11123265

Synthesis of 2-phosphonoheterocycles via base-promoted 5-endo cyclization

Ameni Bousbia, Mohamed Lamine Benkhoud, Laurent El-Kaïm and Sébastien Prévost

Tetrahedron Letters, 2021, 64, 152742
DOI: 10.1016/j.tetlet.2020.152742

Spectroscopic and Computational pH Study of NiII and PdII Pyrrole-Imine Chelates with Human Serum Albumin

Sheldon Sookai, Matthew Lee Bracken and Monika Nowakowska

Molecules, 2023, 28, 7466
DOI: 10.3390/molecules28227466

Synthesis of N‐ureido Pyrrole Derivatives Through Gold‐Catalysed Reaction: Solvent and Catalyst Effect

Volkan Taşdemir

ChemistrySelect, 2024, 9
DOI: 10.1002/slct.202304123

Identification of Noncompetitive Inhibitors of Cytosolic 5′-Nucleotidase II Using a Fragment-Based Approach

Zsuzsanna Marton, Rémi Guillon, Isabelle Krimm, Preeti, Rahila Rahimova, David Egron, Lars P. Jordheim, Nushin Aghajari, Charles Dumontet, Christian Périgaud, Corinne Lionne, Suzanne Peyrottes and Laurent Chaloin

J. Med. Chem., 2015, 58, 9680
DOI: 10.1021/acs.jmedchem.5b01616

Isocyanide-Based Multicomponent Reactions in Water: Advanced Green Tools for the Synthesis of Heterocyclic Compounds

Tahereh Nasiriani, Siamak Javanbakht, Mohammad Taghi Nazeri, Hassan Farhid, Vida Khodkari and Ahmad Shaabani

Top Curr Chem (Z), 2022, 380
DOI: 10.1007/s41061-022-00403-8

Dative Directing Group Effects in Ti-Catalyzed [2+2+1] Pyrrole Synthesis: Chemo- and Regioselective Alkyne Heterocoupling

Hsin-Chun Chiu, Xin Yi See and Ian A. Tonks

ACS Catal., 2019, 9, 216
DOI: 10.1021/acscatal.8b04669

Multifunctional 2‐ and 3‐Fluoropyrroles

Darren Heeran and Graham Sandford

Eur J Org Chem, 2019, 2019, 2339
DOI: 10.1002/ejoc.201900185

Synthesis of multisubstituted pyrroles by ligand-controlled site-selective arylation and their transformation into multiarylated pyrrolines and pyrrolidines

Miyuki Yamaguchi, Sakiko Fujiwara, Yukiko Mori, Hideyuki Konishi and Kei Manabe

Tetrahedron, 2022, 123, 132962
DOI: 10.1016/j.tet.2022.132962

Electrochemical Organoselenium Catalysis for the Selective Activation of Alkynes: Easy Access to Carbonyl-pyrroles/oxazoles from N-Propargyl Enamines/Amides

Mrinmay Baidya, Jhilik Dutta and Suman De Sarkar

Org. Lett., 2023, 25, 3812
DOI: 10.1021/acs.orglett.3c01355

Surface modification of nanocellulose using polypyrrole for the adsorptive removal of Congo red dye and chromium in binary mixture

Tasrin Shahnaz, Mohamed Madhar Fazil S., Padmanaban V.C. and Selvaraju Narayanasamy

International Journal of Biological Macromolecules, 2020, 151, 322
DOI: 10.1016/j.ijbiomac.2020.02.181

Novel preparation of 2,5-diarylpyrroles from aromatic nitriles with 3-arylpropylmagnesium bromides, 1,3-diiodo-5,5-dimethylhydantoin, and BuOK

Momoko Nakamura, Kazuhiro Yoshida and Hideo Togo

Tetrahedron, 2022, 112, 132709
DOI: 10.1016/j.tet.2022.132709

Synthesis of 6-(1H-Pyrrol-1-yl)azolo[1,5-a]pyrimidin-7-amines by the Clauson–Kaas Reaction

V. V. Fedotov, S. V. Aminov, A. O. Neymash, D. A. Gazizov, A. S. Kultyshev, O. S. Eltsov, P. A. Slepukhin, E. N. Ulomskiy and V. L. Rusinov

Russ J Org Chem, 2025, 61, 660
DOI: 10.1134/S1070428025601062

The Gold‐Catalyzed Hydroarylation of Alkynes with Electron‐Rich Heteroarenes – A Kinetic Investigation and New Synthetic Possibilities

Jasmin Schießl, Matthias Rudolph and A. Stephen K. Hashmi

Adv Synth Catal, 2017, 359, 639
DOI: 10.1002/adsc.201600940

Umpolung Reactivity of Ynamides: An Unconventional [1,3]‐Sulfonyl and [1,5]‐Sulfinyl Migration Cascade

B. Prabagar, Rajendra K. Mallick, Rangu Prasad, Vincent Gandon and Akhila K. Sahoo

Angewandte Chemie, 2019, 131, 2387
DOI: 10.1002/ange.201813143

Ultrasound-Promoted One-Pot Synthesis of Mono- or Bis-Substituted Organylselanyl Pyrroles

Thiago J. Peglow, Gabriel P. da Costa, Luis Fernando B. Duarte, Márcio S. Silva, Thiago Barcellos, Gelson Perin and Diego Alves

J. Org. Chem., 2019, 84, 5471
DOI: 10.1021/acs.joc.9b00405

Chiral Brønsted Acid and Gold Catalyzed Enantioselective Synthesis of 1,8‐Dihydroindeno[2,1‐b]pyrroles

Jianwen Jin, Yichao Zhao, Ella Min Ling Sze, Prasath Kothandaraman and Philip Wai Hong Chan

Adv Synth Catal, 2018, 360, 4744
DOI: 10.1002/adsc.201801178

The intricacies of the stacking interaction in a pyrrole–pyrrole system

Tomasz Sierański

Struct Chem, 2016, 27, 1107
DOI: 10.1007/s11224-015-0732-3

A green method for the synthesis of pyrrole derivatives using arylglyoxals, 1,3-diketones and enaminoketones in water or water–ethanol mixture as solvent

Mohammad Anary-Abbasinejada, Frershteh Nezhad-Shshrokhabadi and Marziyeh Mohammadi

Mol Divers, 2020, 24, 1205
DOI: 10.1007/s11030-019-09984-x

Synthesis of new 3-cyanoacetamide pyrrole and 3-acetonitrile pyrrole derivatives

Mohammad Bayat, Shima Nasri and Behrouz Notash

Tetrahedron, 2017, 73, 1522
DOI: 10.1016/j.tet.2017.02.005

Deuterium Analogs of Pharmaceuticals

V. P. Shevchenko, I. Yu. Nagaev, K. V. Shevchenko, L. A. Andreeva and N. F. Myasoedov

Pharm Chem J, 2026, 59, 1134
DOI: 10.1007/s11094-026-03504-6

Humin-sulfuric acid as a novel recoverable biocatalyst for pyrrole synthesis in water

Mandana Armin, Abbas Ali Jafari and Beheshteh Arjmandzadeh

BMC Chemistry, 2024, 18
DOI: 10.1186/s13065-024-01269-1

Site‐Selective Oxidative C4 Alkenylation of (NH)‐Pyrroles Bearing an Electron‐Withdrawing C2 Group

Joydev K. Laha, Rohan A. Bhimpuria and Gajanan B. Mule

ChemCatChem, 2017, 9, 1092
DOI: 10.1002/cctc.201601468

Comprehensive Review of Dihydro‐2H‐pyrrol‐2‐one Derivatives

Benjamin Siddiqui, Chandra Shekhar Yadav, Mohd Faiyyaz, Mohd Akil, Firoj Hassan, Aneez Ahmad, Naseem Ahmad, Abdul Rahman Khan and Iqbal Azad

ChemistrySelect, 2025, 10
DOI: 10.1002/slct.202401807

Surface-enhanced Raman scattering and quantum chemical studies of 2-trifluoroacetylpyrrole chemisorbed on colloidal silver and gold nanoparticles: A comparative study

R. Premkumar, Shamima Hussain, T. Mathavan, K. Anitha and A. Milton Franklin Benial

Journal of Molecular Liquids, 2019, 290, 111209
DOI: 10.1016/j.molliq.2019.111209

A New Strategy for the Synthesis of 4‐Propargyl‐Substituted 1H‐Pyrroles from N‐(5‐phenyl‐2,4‐pentadiynyl) β‐Enaminones

Elif Serel Yilmaz and Metin Zora

ChemistrySelect, 2019, 4, 11043
DOI: 10.1002/slct.201902759

Dehydrative condensation of β-aminoalcohols with CO2: An environmentally benign access to 2-oxazolidinone derivatives

Sepideh Farshbaf, Leila Zare Fekri, Mohammad Nikpassand, Robab Mohammadi and Esmail Vessally

Journal of CO2 Utilization, 2018, 25, 194
DOI: 10.1016/j.jcou.2018.03.020

A facile heterogeneous catalytic approach for one-pot synthesis of fused benzoxazinones using Cuβ zeolite and Evaluation of biological activities

Suchitha Dasu, Krishna Sai Gajula, Vasu Amrutham, Murali Boosa, Ramulamma Madasu, Madhuri Lekkala, Sai Balaji Andugulapati and Narender Nama

Tetrahedron, 2024, 156, 133931
DOI: 10.1016/j.tet.2024.133931

Antibacterial activity of new silatrane pyrrole-2-carboxamide hybrids

Sergei N. Adamovich, Evgeny Kh. Sadykov, Igor A. Ushakov, Elizaveta N. Oborina and Lydmila A. Belovezhets

Mendeleev Communications, 2021, 31, 204
DOI: 10.1016/j.mencom.2021.03.019

Novel chloropyridazine sulfonamides as aromatase inhibitors and apoptotic inducers in breast cancer

Sally S. Zahran, Mostafa G.M. El-Gazzar, Marwa G. El-Gazzar and Mostafa M. Ghorab

Bioorganic Chemistry, 2025, 160, 108470
DOI: 10.1016/j.bioorg.2025.108470

The application of azoarenes in the synthesis of nitrogen-containing heterocycles

Azim Ziyaei Halimehjani, Nima Sadeghzadeh and Sina Moghaddam

Tetrahedron, 2025, 171, 134428
DOI: 10.1016/j.tet.2024.134428

Catalytic activity of supra molecular self-assembled Nickel (II) coordination complex in synthesis of indeno-pyrimidine derivatives

Kranthi Kumar Gangu, Suresh Maddila, Saratchandra Babu Mukkamala and Sreekantha B. Jonnalagadda

Polyhedron, 2019, 158, 464
DOI: 10.1016/j.poly.2018.11.041

A General Synthetic Route to Isomeric Pyrrolo[1,2-x][1,4]diazepinones

Elena Y. Zelina, Tatyana A. Nevolina, Ludmila N. Sorotskaja, Dmitry A. Skvortsov, Igor V. Trushkov and Maxim G. Uchuskin

J. Org. Chem., 2018, 83, 11747
DOI: 10.1021/acs.joc.8b01669

Optical Rotation Calculations for a Set of Pyrrole Compounds

Shokouh Haghdani, Odd R. Gautun, Henrik Koch and Per-Olof Åstrand

J. Phys. Chem. A, 2016, 120, 7351
DOI: 10.1021/acs.jpca.6b07004

Synthesis of novel pyrroles and fused pyrroles as antifungal and antibacterial agents

Rania Helmy Abd El-Hameed, Amira Ibrahim Sayed, Shima Mahmoud Ali, Mohamed A. Mosa, Zainab M. Khoder and Samar Said Fatahala

Journal of Enzyme Inhibition and Medicinal Chemistry, 2021, 36, 2183
DOI: 10.1080/14756366.2021.1984904

TBAI‐Catalyzed, TBHP‐Mediated Modular Three‐Component Cascade Towards Highly Functionalized Pyrrole via [3+2] Annulation

Karthiyayini Gnanaoli, Deepan Babu Rajkumar, Keerthana Gopal, B. Saritha and C. Uma Maheswari

Eur J Org Chem, 2024, 27
DOI: 10.1002/ejoc.202400197

External Oxidant‐Free Oxidative Tandem Cyclization: NaI‐Catalyzed Thiolation for the Synthesis of 3‐Thiosubstituted Pyrroles

Bingxiang Yuan, Yong Jiang, Zhenjie Qi, Xin Guan, Ting Wang and Rulong Yan

Adv Synth Catal, 2019, 361, 5112
DOI: 10.1002/adsc.201900620

Synthesis, docking, SAR and ADMET evaluation of novel pyrrolo[3,4-c]pyrazole-4,6-dione derivatives

Yasser H. Zaki, Magdi E. A. Zaki, Basant Farag and Sobhi M. Gomha

Sci Rep, 2026, 16
DOI: 10.1038/s41598-025-33678-0

Synthesis of Polysubstituted Pyrroles through the Tandem 1,3‐Addition/5‐endo‐dig Cyclization of 1‐(1‐Alkynyl)cyclopropyl Imines

Aurelija Urbanaitė and Inga Čikotienė

Eur J Org Chem, 2016, 2016, 5294
DOI: 10.1002/ejoc.201600985

Copper catalysed regioselective synthesis of pyrimidine substituted Indolizino[8,7-b]indole derivatives via cascade A3 annulation

Sunit Kumar, Rakesh Kumar, Chandi C. Malakar and Virender Singh

Tetrahedron, 2023, 142, 133547
DOI: 10.1016/j.tet.2023.133547

Synthesis of trisubstituted pyrroles via cycloamination of substituted 2-acetyl-1,4-diketones

Yashi Dwivedi, Priya Tiwari, Gitika Guliani, Subrata Barick and Sandeep Chandrashekharappa

Journal of Molecular Structure, 2026, 1351, 144166
DOI: 10.1016/j.molstruc.2025.144166

One-pot three-component reaction of ninhydrin, 1,3-dicarbonyl compounds, and primary amines to afford indeno[1,2-b]pyrrol-4(1H)-ones

Hossein Karami, Zinatossadat Hossaini, Maryam Sabbaghan and Faramarz Rostami-Charati

Chem Heterocycl Comp, 2018, 54, 1040
DOI: 10.1007/s10593-018-2388-6

An efficient one pot three‐component domino reaction for the synthesis of 1,3,4‐trisubstituted pyrroles

Sundaravel Vivek Kumar, Sivasubramanian Muthusaravanan, Shanmugam Muthusubramanian and Subbu Perumal

ChemistrySelect, 2016, 1, 675
DOI: 10.1002/slct.201600108

Assembly of 1,2,3,4-Tetrahydropyrrolo[1,2-a]pyrazines via the Domino Reaction of 2-Imidazolines and Terminal Electron-Deficient Alkynes

Nikita E. Golantsov, Alexandra S. Golubenkova, Alexey A. Festa, Alexey V. Varlamov and Leonid G. Voskressensky

J. Org. Chem., 2022, 87, 3242
DOI: 10.1021/acs.joc.1c02930

Synthesis of polysubstituted pyrroles via a gold(I)-catalyzed tandem three-component reaction at room temperature

Li Li, Qi Chen, Xiaonan Xiong, Chuang Zhang, Jingjing Qian, Jie Shi, Qiong An and Ming Zhang

Chinese Chemical Letters, 2018, 29, 1893
DOI: 10.1016/j.cclet.2018.09.004

Photocatalyst‐Free Visible‐Light Enabled Synthesis of Substituted Pyrroles from α‐Keto Vinyl Azides

Satheesh Borra, Lodsna Borkotoky, Uma Devi Newar, Babulal Das and Ram Awatar Maurya

Adv Synth Catal, 2020, 362, 3364
DOI: 10.1002/adsc.202000562

Sustainable Synthesis of N-Substituted Pyrroles via Fe-Catalyzed One-Pot Multicomponent Reaction

Santana Chakraborty, Arijit Singha Mohapatra and Nanda D. Paul

Org. Lett., 2026, 28, 3808
DOI: 10.1021/acs.orglett.6c00539

Metal-free cascade reactions of aldehydes and primary amines for the synthesis of 1,3,4-trisubstituted pyrroles

Yong Gao, Changfeng Hu, Jie-Ping Wan and Chengping Wen

Tetrahedron Letters, 2016, 57, 4854
DOI: 10.1016/j.tetlet.2016.09.063

Oxidant‐Controlled Divergent Syntheses of Pyrazoles and Pyrroles by Copper(I)‐Catalyzed Oxidative Coupling of β‐Enamino Esters

Su San Jang, Jun Yeong Chang, Gil Yeong Kang and So Won Youn

Asian J Org Chem, 2019, 8, 1668
DOI: 10.1002/ajoc.201900351

An Efficient, Scalable and Eco‐friendly Synthesis of 4,5‐substituted Pyrrole‐3‐Carbonitriles by Intramolecular Annulation on Pd/C and HZSM‐5

Jianchao Chen, Chengtao Li, Yanan Zhou, Changshan Sun and Tiemin Sun

ChemCatChem, 2019, 11, 1943
DOI: 10.1002/cctc.201900154

Trifluoroethanol as a Unique Additive for the Chemoselective Electrooxidation of Enamines to Access Unsymmetrically Substituted NH‐Pyrroles

Mrinmay Baidya, Debabrata Maiti, Lisa Roy and Suman De Sarkar

Angewandte Chemie, 2022, 134
DOI: 10.1002/ange.202111679

Study of 1,3-dipolar cycloaddition of amino-acid azomethines and Juglone

Vadym Syngaevsky, Andrew Karkhut, Sviatoslav Polovkovych, Andrzej Gzella, Roman Lesyk and Volodymyr Novikov

Synthetic Communications, 2020, 50, 3165
DOI: 10.1080/00397911.2020.1795880

Recent Progress in the Synthesis of Heterocycles through Base Metal‐Catalyzed Acceptorless Dehydrogenative and Borrowing Hydrogen Approach

Avijit Mondal, Rahul Sharma, Debjyoti Pal and Dipankar Srimani

Eur J Org Chem, 2021, 2021, 3690
DOI: 10.1002/ejoc.202100517

The synthesis of pyrrole from C4‐olefinated isoxazole catalyzed by ruthenium: A density functional theory study

Haibo Liu

J of Physical Organic Chem, 2021, 34
DOI: 10.1002/poc.4178

Biocontrol Activity of Aspergillus terreus ANU-301 against Two Distinct Plant Diseases, Tomato Fusarium Wilt and Potato Soft Rot

Hyong Woo Choi and S. M. Ahsan

Plant Pathol J, 2022, 38, 33
DOI: 10.5423/PPJ.OA.12.2021.0187

Click reaction inspired synthesis, antimicrobial evaluation and in silico docking of some pyrrole-chalcone linked 1,2,3-triazole hybrids

Monika Yadav, Kashmiri Lal, Aman Kumar, Prashant Singh, Vijay Kumar Vishvakarma and Ramesh Chandra

Journal of Molecular Structure, 2023, 1273, 134321
DOI: 10.1016/j.molstruc.2022.134321

Heteropolyacid-alumina composites as heterogeneous catalysts for the synthesis of organic compounds: a comprehensive review

María Belén Colombo Migliorero, Valeria Palermo, Agustín Ponzinibbio and Gustavo Pablo Romanelli

Reviews in Chemical Engineering, 2025, 41, 491
DOI: 10.1515/revce-2024-0085

Synthesis, characterization and catalytic activity of PEPPSI-type palladium–NHC complexes

Ichraf Slimani, Lamjed Mansour, Ismail Özdemir, Nevin Gürbüz and Naceur Hamdi

Inorganica Chimica Acta, 2021, 515, 120043
DOI: 10.1016/j.ica.2020.120043

Tandem Synthesis of Polysubstituted Pyrroles via Cu(I)-Catalyzed Cyclization of Ketene N,S-Acetals with β-Ketodinitriles

Anup Kumar Sharma, Mahesh Kumar, Shiv Chand and Krishna Nand Singh

J. Org. Chem., 2025, 90, 3981
DOI: 10.1021/acs.joc.4c03071

A Facile One-Pot Synthesis of New Poly Functionalized Pyrrolotriazoles via a Regioselective Multicomponent Cyclisation and Suzuki–Miyaura Coupling Reactions

Simon Garnier, Kévin Brugemann, Agnieszka Zak, Johnny Vercouillie, Marie Potier-Cartereau, Mathieu Marchivie, Sylvain Routier and Frédéric Buron

Catalysts, 2022, 12, 828
DOI: 10.3390/catal12080828

Visible Light Catalysis Promoted the Synthesis of Tetra‐C‐Substituted Pyrroles under External‐Oxidant‐Free Conditions

Qiong Liu, Xiaoying Niu, Hao‐Yuan Li, Qing‐Yuan Meng and Xiu‐Long Yang

Helvetica Chimica Acta, 2025, 108
DOI: 10.1002/hlca.202500108

Iridium‐Catalyzed Enantioselective Synthesis of Pyrrole‐Annulated Medium‐Sized‐Ring Compounds

Lin Huang, Yue Cai, Chao Zheng, Li‐Xin Dai and Shu‐Li You

Angew Chem Int Ed, 2017, 56, 10545
DOI: 10.1002/anie.201705068

A Palladium-Catalyzed Cascade Process of 1,3-Enynes and Imines to Construct Multisubstituted Pyrrole Derivatives

Tian-Ying Zhang, Bao-Rui Kong, Ze-Liang He, Zhi-Chao Chen, Wei Du and Ying-Chun Chen

Org. Lett., 2025, 27, 13952
DOI: 10.1021/acs.orglett.5c04542

Crystal-guided computational profiling of dichlorophenyl-piperazine ligands as JNK3 binders: Hydrophobic interaction-driven design for neurodegenerative therapy

Keshav Kumar Harish, Ananda Swamynayaka, Omantheswara Nagaraja, Doreswamy B. Haruvegowda, Vindu Vahini M, Divakar Vishwanath, Basappa Basappa, Dukanya Dukanya and Mahendra Madegowda

Journal of Molecular Structure, 2026, 1351, 144361
DOI: 10.1016/j.molstruc.2025.144361

Identification and characterization of antibacterial compound(s) of cockroaches (Periplaneta americana)

Salwa Mansur Ali, Ruqaiyyah Siddiqui, Seng-Kai Ong, Muhammad Raza Shah, Ayaz Anwar, Peter J. Heard and Naveed Ahmed Khan

Appl Microbiol Biotechnol, 2017, 101, 253
DOI: 10.1007/s00253-016-7872-2

One‐Pot Synthesis of Highly Substituted Pyrroles by Three‐Component Reactions of Donor–Acceptor Cyclopropanes, Salicylaldehydes, and Ammonium Acetate

Zhenjie Su, Wenxing Gu, Siran Qian, Shuwen Xue and Cunde Wang

Eur J Org Chem, 2018, 2018, 1019
DOI: 10.1002/ejoc.201701674

Functionalization of 2‐Trifluoromethyl‐1H‐pyrrole: A Convenient Entry into Advanced Fluorinated Building Blocks Including all Isomeric 2‐(Trifluoromethyl)prolines

Vasyl Yu. Hys, Oleksandr I. Shevchuk, Bohdan V. Vashchenko, Oleksandr V. Karpenko, Alina O. Gorlova and Oleksandr O. Grygorenko

Eur J Org Chem, 2020, 2020, 3896
DOI: 10.1002/ejoc.202000519

Synthesis, Molecular Docking, and In Silico ADMET Studies of New Thiadiazoles, Chalcones, and Pyrazolines Incorporating Alkaloid Like Structure as Antibacterial Agent

Yara N. Laboud, Doaa Zahran, Mohamed A. Mohamed. Teleb, Huwaida M. E. Hassaneen, Hamdi M. Hassaneen and Fatma M. Saleh

ChemistrySelect, 2025, 10
DOI: 10.1002/slct.202500672

An Amino Sugar Promoted Green Protocol: A One‐Pot, Meglumine‐Catalyzed, Multicomponent Strategy for Synthesis of Multifaceted Pyrroloacridin‐1(2H)‐one Derivatives

Pratibha Rai, Anu Mishra, Madhulika Srivastava, Snehlata Yadav, Bhartendu Pati Tripathi, Jaya Singh and Jagdamba Singh

ChemistrySelect, 2017, 2, 2245
DOI: 10.1002/slct.201601718

FeCl3-Mediated Domino Reaction of Benzoxazinones with Aroylmethylidene Malonates: Synthesis to Functionalized Pyrrolobenzoxazines

Shweta Bisht and Rama Krishna Peddinti

J. Org. Chem., 2017, 82, 13617
DOI: 10.1021/acs.joc.7b02207

Dual Role of the Arylating Agent in a Highly C(2)-Selective Pd-Catalysed Functionalisation of Pyrrole Derivatives

Milos Petkovic, Milos Jovanovic, Predrag Jovanovic, Milena Simic, Gordana Tasic and Vladimir Savic

Synthesis, 2022, 54, 2839
DOI: 10.1055/a-1758-6312

Pyrrole dicarboxylate substituted porphyrazine, microwave assisted synthesis and properties

Wojciech Szczolko, Michal Kryjewski, Tomasz Koczorowski, Eunice Zuchowska, Lukasz Popenda and Dariusz T. Mlynarczyk

Sci Rep, 2025, 15
DOI: 10.1038/s41598-025-00428-1

Catalytic, Enantioselective Aziridine Desymmetrization with Pyrroles

Dustin Mauldin, Ha Nguyen, Ernest Brubaker, Maxwell Mattejat, Giorgiana Franzese, Calvin Hamerski and Jeremy B. Morgan

J. Org. Chem., 2025, 90, 9280
DOI: 10.1021/acs.joc.5c00816

Reaction of 2H-Azirine-Phosphine Oxides and -Phosphonates with Enolates Derived from β-Keto Esters

Ander Vélez del Burgo, Ana M. Ochoa de Retana, Jesús M. de los Santos and Francisco Palacios

J. Org. Chem., 2016, 81, 100
DOI: 10.1021/acs.joc.5b02347

Synthesis and Toxicological Effect of Some New Pyrrole Derivatives as Prospective Insecticidal Agents against the Cotton Leafworm, Spodoptera littoralis (Boisduval)

Antar A. Abdelhamid, Kaoud S. M. Salama, Ahmed M. Elsayed, Mohamed A. Gad and Mahmoud Abd El Aleem Ali Ali El-Remaily

ACS Omega, 2022, 7, 3990
DOI: 10.1021/acsomega.1c05049

Pyrrole-stabilized free carbenes generated from alkynyl imidates or aldimines and electrophilic alkynes give pyrrolone- or pyrrole-containing products

Qian Xu, Jingyang Shi and Thomas R. Hoye

Nat. Synth, 2025, 5, 95
DOI: 10.1038/s44160-025-00899-0

Isosterism in pyrrole via azaboroles substitution, a theoretical investigation for electronic structural, stability and aromaticity

Safinaz H. El-Demerdash, Shaimaa F. Gad, Ibrahim M. El-Mehasseb and Khaled E. El-Kelany

Heliyon, 2023, 9, e20542
DOI: 10.1016/j.heliyon.2023.e20542

Iridium‐Catalyzed Enantioselective Synthesis of Pyrrole‐Annulated Medium‐Sized‐Ring Compounds

Lin Huang, Yue Cai, Chao Zheng, Li‐Xin Dai and Shu‐Li You

Angewandte Chemie, 2017, 129, 10681
DOI: 10.1002/ange.201705068

Brønsted acid-promoted synthesis of polysubstituted pyrroles from enamines/imines and diazopyruvates: A metal-free cascade approach

Farrukh Sajjad and Ming-Hua Xu

Green Synthesis and Catalysis, 2025, 6, 86
DOI: 10.1016/j.gresc.2023.12.002

An Efficient Synthesis of (Aryl)(4-(2-(arylethynyl)-phenyl)-1H-pyrrol-3-yl)methanone from the Reaction of (E)-1-Aryl-3-(2-(arylethynyl)phenyl)prop-2-en-1-one and p-Toluenesulfonylmethyl Isocyanide

Liangce Rong, Zifeng Zhang, Zhongwei Sun, Chengkai Wang and Fang Li

HETEROCYCLES, 2022, 104, 1033
DOI: 10.3987/COM-22-14633

One-Pot Three-Component Synthesis of Novel Pyrazole-2,3-pyrroledicarboxylic Acid 2,3-Diesters

Hiroshi Maruoka, Emi Shirouzu, Eiichi Masumoto, Fumi Okabe-Nakahara and Kenji Yamagata

HETEROCYCLES, 2018, 96, 233
DOI: 10.3987/COM-17-13844

Multi-component synthesis and invitro biological assessment of novel pyrrole derivatives and pyrano[2,3-c]pyrazole derivatives using Co3O4 nanoparticles as recyclable nanocatalyst

Tahani M. Almeleebia, Mokhtar Jasim Naser, Shakir Mahmood Saeed, Majeed M. Abid, Usama S. Altimari, Murtadha Laftah Shaghnab, Fadhil A. Rasen, Ahmed Alawadi, Irfan Ahmad and Ali Alsalamy

Front. Mater., 2024, 11
DOI: 10.3389/fmats.2024.1354560

Recent Progress for the Synthesis of Pyrrole Derivatives – An Update

Dharti Patel, Drashti Shah, Krishi Patel, Ayush Patel, Tushar Bambharoliya, Anjali Mahavar and Ashish Patel

MROC, 2024, 21, 717
DOI: 10.2174/1570193X20666230530161009

Recent Advances in Synthetic Methods for 2H‐Pyrroles

Seoung‐Mi Choi and Ju Hyun Kim

Adv Synth Catal, 2024, 366, 2
DOI: 10.1002/adsc.202301238

Decarboxylative arylation of substituted pyrroles N-protected with 2-(trimethylsilyl)ethoxymethyl (SEM)

Carlotta Figliola, Sarah M. Greening, Connor Lamont, Brandon R. Groves and Alison Thompson

Can. J. Chem., 2018, 96, 534
DOI: 10.1139/cjc-2017-0402

Reaction Pattern and Mechanistic Aspects of Iodine and Iodine-Based Reagents in Selenylation of Aliphatic, Aromatic, and (Hetero)Cyclic Systems

Pankaj Kumar and Aman Bhalla

Top Curr Chem (Z), 2024, 382
DOI: 10.1007/s41061-024-00459-8

New pyrrole derivatives as DNA gyrase and 14α‐demethylase inhibitors: Design, synthesis, antimicrobial evaluation, and molecular docking

Khaled M. H. Hilmy, Fawzya N. M. Kishk, Esmat B. A. Shahen, Eman A. Sobh and Mohamed A. Hawata

Drug Development Research, 2023, 84, 1204
DOI: 10.1002/ddr.22080

Copper in Efficient Synthesis of Aromatic Heterocycles with Single Heteroatom

Tapas Pal, Goutam Kumar Lahiri and Debabrata Maiti

Eur J Org Chem, 2020, 2020, 6859
DOI: 10.1002/ejoc.202000688

An efficient synthesis of polyfunctionalized pyrroles by three-component reaction of arylglyoxals, Meldrum’s acid and ethyl 2-chloro-3-(arylamino)but-2-enoates

Fereshteh Nezhad-shahrokhabadi and Mohammad Anary-Abbasinejad

J IRAN CHEM SOC, 2022, 19, 2655
DOI: 10.1007/s13738-021-02485-5

A Catalyst‐Free Domino Protocol for the Chemoselective Synthesis of Multifunctionalised Pyrroles in Aqueous Media via Nitroketene‐N,S‐Acetal Chemistry

Ankita Chaudhary, Jitender M. Khurana, Garima Khanna and Mohit Saroha

ChemistrySelect, 2018, 3, 6334
DOI: 10.1002/slct.201800831

Synthesis of 2,2,5-Trisubstituted 2H-Pyrroles and 2,3,5-Trisubstituted 1H-Pyrroles by Ligand-Controlled Site-Selective Dearomative C2-Arylation and Direct C3-Arylation

Miyuki Yamaguchi, Sakiko Fujiwara and Kei Manabe

Org. Lett., 2019, 21, 6972
DOI: 10.1021/acs.orglett.9b02559

Synthesis of coumarin-linked naphthoquinone fused pyrrole derivatives by HFIP-mediated multicomponent reaction

Ujjain Chaurasia and Tasneem Parvin

J Chem Sci, 2023, 135
DOI: 10.1007/s12039-023-02185-y

Trifluoromethyl‐β‐dicarbonyls as Versatile Synthons in Synthesis of Heterocycles

Garima Sumran, Naman Jain, Prince Kumar and Ranjana Aggarwal

Chemistry A European J, 2024, 30
DOI: 10.1002/chem.202303599

Regioselective Stepwise Synthesis of Unsymmetrical 1,2,5-Triarylpyrroles via Palladium-Catalyzed Decarboxylative Cross-Coupling and C–H Arylation

Cindy Buonomano, Stephanie Patterson, Judith Sorel Ngou, Cynthia Messina, Sarah Taylor, François Bilodeau and Pat Forgione

Molecules, 2026, 31, 986
DOI: 10.3390/molecules31060986

TCFH–NMI Ketone Synthesis Inspired by Nucleophilicity Scales

Johnson H. Ho, Grant H. Miller, Kasey K. Chung, Sydney D. Neibert, Gregory L. Beutner and David A. Vosburg

Org. Lett., 2024, 26, 8904
DOI: 10.1021/acs.orglett.4c03363

Asymmetric Synthesis of Highly Substituted Spiro[2H‐pyrrole‐2,3‐Succinimide] Derivatives by Copper‐Catalyzed Post‐Ugi Reactions

Javier Gómez‐Ayuso, Israel Carreira‐Barral, Roberto Quesada and María García‐Valverde

Adv Synth Catal, 2025, 367
DOI: 10.1002/adsc.202500166

Oxidative Coupling: An Important Tool for Pyrrole Synthesis

Shrishti Tripathi, Rajnish Kumar, Avijit Mazumder, Salahuddin, Himanshu Singh, Ranjeet Kumar Yadav, Neelima Kukreti, Rashmi Mishra and Saurabh Singh

LOC, 2024, 21, 993
DOI: 10.2174/0115701786304220240320073540

Tunable Synthesis of 4-Acyl- and 4-Formyl Pyrroles by Rhodium-Catalyzed Ring-Expansion of Azirines with Enaminones

Xiuli Li, Jianchao Liu and Jie-Ping Wan

Org. Lett., 2025, 27, 1949
DOI: 10.1021/acs.orglett.5c00230

Green Synthesis and Biological Study of Novel Cyclopenta[b]pyridines: Multicomponent Reactions of Meldrum’s Acid

Faezeh Shafaei, Hadi Jouladehroodbar, Fariba Zamani Hargalani, Zinatossadat Hossaini and Haci Baykara

Journal of Chemistry, 2025, 2025
DOI: 10.1155/joch/6232375

State- and time-resolved observation of ultrafast intermolecular proton transfer in hydrated biomolecules

Jiaqi Zhou, Lu Wu, Michal Belina, Anna D. Skitnevskaya, Shaokui Jia, Xiaorui Xue, Xintai Hao, Qingrui Zeng, Qibo Ma, Yongtao Zhao, Xiaokai Li, Lanhai He, Sizuo Luo, Dongdong Zhang, Chuncheng Wang, Alexander B. Trofimov, Petr Slavíček, Dajun Ding and Xueguang Ren

Nat Commun, 2025, 16
DOI: 10.1038/s41467-025-61305-z

Synthesis of pyrrole-heterocyclic derivatives as anti-Alzheimer and antidiabetic candidates: An in vitro-in silico study

Ol'ga V. Petrova, Denis N. Tomilin, Halil Şenol, Kseniya V. Belyaeva, Lina P. Nikitina, Ludmila A. Oparina, Lyubov N. Sobenina, Boris A. Trofimov, Nastaran Sadeghian, Parham Taslimi, Vagif Farzaliyev, Afsun Sujayev and İlhami Gulçin

Journal of Molecular Structure, 2024, 1315, 138998
DOI: 10.1016/j.molstruc.2024.138998

Site-selective chlorination of pyrrolic heterocycles by flavin dependent enzyme PrnC

GuangRong Peh, Terence Tay, Lee Ling Tan, Elaine Tiong, Jiawu Bi, Yi Ling Goh, Suming Ye, Fu Lin, Cheryl Jia Xin Tan, Yong Zi Tan, Joel Wong, Huimin Zhao, Fong Tian Wong, Ee Lui Ang and Yee Hwee Lim

Commun Chem, 2024, 7
DOI: 10.1038/s42004-023-01083-1

A series of (E)-5-(arylideneamino)-1-tert-butyl-1H-pyrrole-3-carbonitriles and their reduction products to secondary amines: syntheses and X-ray structural studies

Mario A. Macías, Juan-Carlos Castillo and Jaime Portilla

Acta Crystallogr C Struct Chem, 2018, 74, 82
DOI: 10.1107/S2053229617017260

Synthesis of fused hydroxy dihydropyrroles and unexpected dihydropyrazine and dihydroquinoxaline derivatives based on heterocyclic ketene aminals

Monireh Rezaei, Mohammad Bayat and Behrouz Notash

Journal of Heterocyclic Chem, 2020, 57, 880
DOI: 10.1002/jhet.3834

The pilot study of the basic pharmacokinetic properties of pyrrolylcarnosine — the new pyrrolic derivative of dipeptide carnosine

D. A. Abaimov, Anastasiya V. Khutorova, A. K. Sariev, O. I. Kulikova, M. A. Belousova, S. L. Stvolinsky, V. A. Migulin and T. N. Fedorova

Fk&Fd, 2023, 29
DOI: 10.37489/2587-7836-2023-2-29-36

NPAH formation through ring expansion: Indole formation from acetylene addition to pyrrole

Xinqi Zhang, Huajie Lyu, Peng Liu, Hong Wang, Zhandong Wang and Bingjie Chen

Combustion and Flame, 2026, 283, 114626
DOI: 10.1016/j.combustflame.2025.114626

Silver-Catalyzed Cascade Reaction of β-Enaminones and Isocyanoacetates To Construct Functionalized Pyrroles

Guichun Fang, Jianquan Liu, Junkai Fu, Qun Liu and Xihe Bi

Org. Lett., 2017, 19, 1346
DOI: 10.1021/acs.orglett.7b00201

Solvent Free Synthesis of N‐Substituted Pyrroles Catalyzed by Calcium Nitrate

Rucha R. Wani, Hemchandra K. Chaudhari and Balaram S. Takale

Journal of Heterocyclic Chem, 2019, 56, 1337
DOI: 10.1002/jhet.3507

Design, synthesis, in vitro and in silico evaluation of new pyrrole derivatives as monoamine oxidase inhibitors

Mehlika D. Altintop, Belgin Sever, Derya Osmaniye, Begüm N. Sağlık and Ahmet Özdemir

Archiv der Pharmazie, 2018, 351
DOI: 10.1002/ardp.201800082

Synthesis, structure characterization, and anticancer activity of a novel oxygen-bridged tricyclic Biginelli adduct

Mohamed M. Ibrahim, Hamdy S. El-Sheshtawy, Maged El-Kemary, Salih Al-Juaid, Mohamed Youssef and Islam H. El-Azab

Journal of Molecular Structure, 2017, 1137, 714
DOI: 10.1016/j.molstruc.2017.02.091

A pyrrole-based natural small molecule mitigates HSP90 expression in MDA-MB-231 cells and inhibits tumor angiogenesis in mice by inactivating HSF-1

K.C. Rashmi, H.S. Atreya, M. Harsha Raj, Bharathi P. Salimath and H.S. Aparna

Cell Stress and Chaperones, 2017, 22, 751
DOI: 10.1007/s12192-017-0802-0

Gold-Catalyzed Synthesis of Substituted 3-Trifluoromethylpyrroles from Mesylated Amino Trifluoromethylpropargylic Alcohols

Benjamin Guieu, Myriam Le Roch, Michèle David and Nicolas Gouault

J. Org. Chem., 2017, 82, 13708
DOI: 10.1021/acs.joc.7b02567

Iterative Suzuki‐Miyaura Cross‐coupling/Bromo‐desilylation Reaction Sequences for the Assembly of Chemically Well‐defined, Acyclic Oligopyrrole/Benzenoid Hybrids Embodying Mixed Modes of Connectivity

BoRa Lee, Anthony C. Willis, Jas S. Ward, Warren T. Smith, Ping Lan and Martin G. Banwell

Chemistry An Asian Journal, 2020, 15, 3059
DOI: 10.1002/asia.202000740

Regioselective Synthesis of 3-Trifluoromethylpyrroles by [3 + 2] Cycloaddition of N-Acyl α-Amino Acids and 2-Bromo-3,3,3-trifluoropropene

Weidi Zeng, Hui Li, Duozhi Wang and Lei Zhou

J. Org. Chem., 2023, 88, 14088
DOI: 10.1021/acs.joc.3c01611

Crystallographic, spectroscopic and thermal studies of 1-(4-bromophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-3-methyl-1H-pyrazole

Erika Moreno-Suárez, Rafael Avila-Acosta, Karen Sánchez-Ramírez, Juan-Carlos Castillo and Mario A. Macías

Acta Crystallogr C Struct Chem, 2023, 79, 472
DOI: 10.1107/S2053229623009221

Anti-Trichomonas vaginalis Activity of Marine Ascidians (Tunicates; Ascidiacea) from the Bushehr Province, Iran

Hamideh Malekhayati, Afshar Bargahi, Soleiman Khorami, Mohsen Khataminejad and Moradali Fouladvand

Turkiye Parazitol Derg, 2024, 48, 21
DOI: 10.4274/tpd.galenos.2023.96658

Site- and Regioselective Monoalkenylation of Pyrroles with Alkynes via Cp*CoIII Catalysis

Ryo Tanaka, Hideya Ikemoto, Motomu Kanai, Tatsuhiko Yoshino and Shigeki Matsunaga

Org. Lett., 2016, 18, 5732
DOI: 10.1021/acs.orglett.6b02997

A catalyst-free approach to regioselective synthesis of multi-functional 1 H -pyrrolo[1,2- a ]fused[1,3]diazaheterocycle using ketene dithioacetals in water–ethanol media

Mohammad Bayat and Shima Nasri

Tetrahedron Letters, 2017, 58, 3107
DOI: 10.1016/j.tetlet.2017.06.076

Efficient bulk scale synthesis of popular pesticide synthon: tetrachlorothiophene

G. V. Shiva Reddy, M. Chandrappa, V. N. Padmanabha Gowda, Fazlur Rahaman, S. Girish Kumar, B. N. Narasimha Murthy and Phani Kumar Pullela

Catalysis, Structure & Reactivity, 2017, 3, 138
DOI: 10.1080/2055074X.2017.1327472

Synthesis, Characterization, Molecular Docking, Acetylcholinesterase and α‐Glycosidase Inhibition Profiles of Nitrogen‐Based Novel Heterocyclic Compounds

İlhami Gulcin, Olga V. Petrova, Parham Taslimi, Svetlana F. Malysheva, Elena Yu. Schmidt, Lyubov N. Sobenina, Nina K. Gusarova, Boris A. Trofimov, Burak Tuzun, Vagif M. Farzaliyev, Saleh Alwasel and Afsun R. Sujayev

ChemistrySelect, 2022, 7
DOI: 10.1002/slct.202200370

Synthesis of Polysubstituted Pyrroles by the Reaction of Enaminoketones, Arylglyoxals, and N,N-Dimethylbarbituric Acid

Nadezhda N. Kolos and Nataliia V. Chechina

Chem Heterocycl Comp, 2019, 55, 1278
DOI: 10.1007/s10593-019-02613-3

Design, Synthesis, Characterization and Catalytic Activity in Direct Arylation Reaction of the Benzimidazole-Functionalized PEPPSI-type Pd(II)NHC Complexes bearing 4-Vynylbenzyl Group

Semra DAŞGIN, Yetkin GÖK and Aydın AKTAŞ

EJOSAT, 2022
DOI: 10.31590/ejosat.1168351

An Expedient Lewis‐Acid‐Catalyzed Microwave‐Assisted Domino Approach to Coumarin‐Fused Pyrroles and Related Heterocycles under Neat Conditions

Anubha Yadav, Santosh K. Gudimella and Sampak Samanta

ChemistrySelect, 2019, 4, 12768
DOI: 10.1002/slct.201903711

Azomethine ylide cycloaddition of 2-C-formyl glycals with α-amino acids for the synthesis of substituted pyrroles

V. Veerabadhra Reddy and B.V. Subba Reddy

Tetrahedron, 2021, 97, 132389
DOI: 10.1016/j.tet.2021.132389

Pyrrole‐based EGFR inhibitors for the treatment of NCSLC: Binding modes and SARs investigations

Jie He, Leixuan Luo, Shidi Xu, Feiyi Yang and Wufu Zhu

Chem Biol Drug Des, 2023, 101, 195
DOI: 10.1111/cbdd.14169

Biocatalytic decarboxylative Michael addition for synthesis of 1,4-benzoxazinone derivatives

Hossein Bavandi, Mansour Shahedi, Zohreh Habibi, Maryam Yousefi, Jesper Brask and Mehdi Mohammadi

Sci Rep, 2022, 12
DOI: 10.1038/s41598-022-16291-3

Biocompatibility of colloidal polypyrrole

Simona Káčerová, Zdenka Víchová, Kristýna Valášková, Jan Vícha, Lukáš Münster, Věra Kašpárková, Ondřej Vašíček and Petr Humpolíček

Colloids and Surfaces B: Biointerfaces, 2023, 232, 113605
DOI: 10.1016/j.colsurfb.2023.113605

Redox-Neutral 1,3-Dipolar Cycloaddition of 2H-Azirines with 2,4,6-Triarylpyrylium Salts under Visible Light Irradiation

Ayushi Pokhriyal, Bhupal Singh Karki, Ruchir Kant and Namrata Rastogi

J. Org. Chem., 2021, 86, 4661
DOI: 10.1021/acs.joc.1c00082

Synthesis, characterization and semiconducting behavior of N,2,5-trisubstituted pyrroles

Olivia Monroy, Lioudmila Fomina, María Elena Sánchez-Vergara, Rubén Gaviño, Alonso Acosta, José Ramón Álvarez Bada and Roberto Salcedo

Journal of Molecular Structure, 2018, 1171, 45
DOI: 10.1016/j.molstruc.2018.05.086

Selective One-Pot Cascade Synthesis of N-Substituted Highly Functionalized Pyrroles from Unprotected Sugars, Primary Amines, and Oxoacetonitriles

Xia Mengxin, Mallikharjuna Rao Lambu and Zaher M. A. Judeh

J. Org. Chem., 2022, 87, 12115
DOI: 10.1021/acs.joc.2c01270

Synthesis of Deuterium-Labeled Pyrrolylcarnosine

V. P. Shevchenko, I. Yu. Nagaev, T. N. Fedorova and N. F. Myasoedov

Dokl Biochem Biophys, 2022, 507, 374
DOI: 10.1134/S1607672922340130

Exploring the Extracellular Macromolecular Composition of Crude Extracts of Penicillium rubens Strain 212 for Elucidation Its Mode of Action as a Biocontrol Agent

Maria Carreras, Eduardo A. Espeso, Alba Gutierrez-Docio, Silvia Moreno-Fernandez, Marin Prodanov, Maria Dolores Hernando, Paloma Melgarejo and Inmaculada Larena

JoF, 2020, 6, 131
DOI: 10.3390/jof6030131

Copper-catalyzed cycloisomerization of alkynylaziridines to access functionalized 2-substituted-4-formylpyrroles

Anne Westermeyer, Gérard Guillamot, Phannarath Phansavath and Virginie Ratovelomanana-Vidal

Tetrahedron, 2020, 76, 131221
DOI: 10.1016/j.tet.2020.131221

Recent Advances in the Fixation of CO2 to Form N‐Containing Heterocyclic Compounds

Qi Zhang and Xin Jin

Chemistry A European J, 2025, 31
DOI: 10.1002/chem.202500933

Trifluoroethanol as a Unique Additive for the Chemoselective Electrooxidation of Enamines to Access Unsymmetrically Substituted NH‐Pyrroles

Mrinmay Baidya, Debabrata Maiti, Lisa Roy and Suman De Sarkar

Angew Chem Int Ed, 2022, 61
DOI: 10.1002/anie.202111679

Tridentate Nickel(II)-Catalyzed Chemodivergent C–H Functionalization and Cyclopropanation: Regioselective and Diastereoselective Access to Substituted Aromatic Heterocycles

Ekta Nag, Sai Manoj N. V. T. Gorantla, Selvakumar Arumugam, Aditya Kulkarni, Kartik Chandra Mondal and Sudipta Roy

Org. Lett., 2020, 22, 6313
DOI: 10.1021/acs.orglett.0c02138

Recent Applications of Heteropolyacids and Related Compounds in Heterocycle Synthesis. Contributions between 2010 and 2020

Angélica M. Escobar, Guillermo Blustein, Rafael Luque and Gustavo P. Romanelli

Catalysts, 2021, 11, 291
DOI: 10.3390/catal11020291

Cytotoxic pyrrole-based gold(III) chelates target human topoisomerase II as dual-mode inhibitors and interact with human serum albumin

Sheldon Sookai, Matthew Akerman, Mia Færch, Yasien Sayed and Orde Q. Munro

European Journal of Medicinal Chemistry, 2025, 287, 117330
DOI: 10.1016/j.ejmech.2025.117330

Hybrid molecules with potential in vitro antiplasmodial and in vivo antimalarial activity against drug‐resistant Plasmodium falciparum

Lian‐Shun Feng, Zhi Xu, Le Chang, Chuan Li, Xiao‐Fei Yan, Chuan Gao, Chao Ding, Feng Zhao, Feng Shi and Xiang Wu

Medicinal Research Reviews, 2020, 40, 931
DOI: 10.1002/med.21643

Pd(II)-Catalyzed Tandem Heterocyclization of 1-(1-Alkynyl)cyclopropyl Oxime Derivatives for the Synthesis of Functionalized Pyrroles

Dong Pan, Yin Wei and Min Shi

Org. Lett., 2016, 18, 3930
DOI: 10.1021/acs.orglett.6b02068

Design, Synthesis, Biological Evaluation and in Silico Studies of Curcumin Pyrrole Conjugates

Nishi Gandha Gogoi, Aziza Rahman, Pankaj Dutta, Jiban Saikia, Anupaul Baruah and Jyotirekha G. Handique

Chemistry & Biodiversity, 2024, 21
DOI: 10.1002/cbdv.202301605

One-Pot Synthesis of N–H-Free Pyrroles from Aldehydes and Alkynes

Lai Chen, Jing-Qian Huo, He-Long Si, Xin-Yu Xu, Song Kou, Jianyou Mao and Jin-Lin Zhang

Org. Lett., 2021, 23, 4348
DOI: 10.1021/acs.orglett.1c01287

Regioselective competitive synthesis of 3,5-bis(het) aryl pyrrole-2-carboxylates/carbonitriles vs. β-enaminones from β-thioxoketones

Kothanahally S. Sharath Kumar, Hanumappa Ananda, Shobith Rangappa, Sathees C. Raghavan and Kanchugarakoppal S. Rangappa

Tetrahedron Letters, 2021, 82, 153373
DOI: 10.1016/j.tetlet.2021.153373

Sterically Controlled C−H Olefination of Heteroarenes

Hao Chen, Mirxan Farizyan, Francesca Ghiringhelli and Manuel van Gemmeren

Angew Chem Int Ed, 2020, 59, 12213
DOI: 10.1002/anie.202004521

Indium‐Catalyzed Formal N‐Arylation and N‐Alkylation of Pyrroles with Amines

Kyohei Yonekura, Kenji Oki and Teruhisa Tsuchimoto

Adv Synth Catal, 2016, 358, 2895
DOI: 10.1002/adsc.201600656

New protocol for diastereoselective synthesis of spirodihydropyrrole-oxindole derivatives

Robabeh Baharfar, Mohadeseh Verdian and Saadieh Mohajer

Chem. Pap., 2022, 76, 3809
DOI: 10.1007/s11696-022-02121-3

Zr-Catalyzed Synthesis of Tetrasubstituted 1,3-Diacylpyrroles from N-Acyl α-Aminoaldehydes and 1,3-Dicarbonyls

Caria Evans, William J. Berkey, Christopher W. Jones and Stefan France

J. Org. Chem., 2023, 88, 8915
DOI: 10.1021/acs.joc.3c00675

Manganese (III) acetate mediated synthesis of polysubstituted pyrroles under solvent-free ball milling

Ji-Chao Zeng, Hui Xu, Fei Yu and Ze Zhang

Tetrahedron Letters, 2017, 58, 674
DOI: 10.1016/j.tetlet.2017.01.016

Synthesis of N-perfluoroalkyl-3,4-disubstituted pyrroles by rhodium-catalyzed transannulation of N-fluoroalkyl-1,2,3-triazoles with terminal alkynes

Olga Bakhanovich, Viktor Khutorianskyi, Vladimir Motornov and Petr Beier

Beilstein J. Org. Chem., 2021, 17, 504
DOI: 10.3762/bjoc.17.44

A Domino Route toward Polysubstituted Pyrroles from 2-Imidazolines and Electron-Deficient Alkynes

Nikita E. Golantsov, Alexandra S. Golubenkova, Alexey A. Festa, Alexey V. Varlamov and Leonid G. Voskressensky

Org. Lett., 2020, 22, 4726
DOI: 10.1021/acs.orglett.0c01530

3,4-Bisthiolated Pyrroles: Concise Construction and Their Electronic Properties

Jun Tian, Kai Feng, Kang-Ning Yuan, Xing Li, Hong-Hong Chang and Wen-Chao Gao

J. Org. Chem., 2022, 87, 2402
DOI: 10.1021/acs.joc.1c02269

Synthesis and antimicrobial activity of derivatives of 4-R-benzylpyrrol-3-carboxylic acid esters

VKhKhT, 2020, 36
DOI: 10.32434/0321-4095-2020-132-5-36-45

Mechanosynthesis of Pyrrole-2-carboxylic Acids via Copper-Catalyzed Spiroannulation/Ring-Opening Aromatization of 4-Arylidene Isoxazol-5-ones with Enamino Esters

Ming-Jun Li, Hui-Juan Xiao, Peng Xu, Luan-Ting Wu, Si-Qi Chen, Ze Zhang and Hui Xu

Org. Lett., 2024, 26, 4189
DOI: 10.1021/acs.orglett.4c00829

Synthesis and Cytotoxic Studies of Pyrrole and Pyrrolidine Derivatives in Human Tumor Cell Lines

Cleudiomar Inácio Lino, Túlio Resende Freitas, Jesus Alberto Avendaño Villarreal, Eduardo Nicolau dos Santos, Ivana Lula, Adriano de Paula Sabino, Vinícius Gonçalves Maltarollo and Renata Barbosa de Oliveira

ChemistrySelect, 2024, 9
DOI: 10.1002/slct.202400212

Visible Light-Induced Hydroacylation of Benzylidenemalononitriles with Aroyl Chlorides Using Silane as a Hydrogen Donor

Ming-Lin Yang, Chun-Lin Dong, Zhi Guan and Yan-Hong He

J. Org. Chem., 2024, 89, 1285
DOI: 10.1021/acs.joc.3c02616

Antimicrobial activity of transition metal (II) complexes based on a Mannich base ligand

Asha Jebamary Selwyn, Pushpalatha Ramasamy, D S Ivan Jebakumar, Benita Jebasilviya Selwyn, Alex Immanuel Xavier Gunaraj, Rajesh Kumar Manavalan and Joice Sophia Ponraj

Emerging Materials Research, 2021, 10, 85
DOI: 10.1680/jemmr.19.00182

Nickel‐Catalyzed Synthesis of Structurally Diverse N‐(hetero)aryl Pyrroles

Chitrarekha Dewangan, Swapnaneel Sarmah and Kishore Natte

Asian J Org Chem, 2025, 14
DOI: 10.1002/ajoc.202500195

Organo-photocatalytic Synthesis of Functionalized Pyrroles from 2H-Azirines and α-Substituted Nitroalkenes

Lalita Devi, Poornima Mishra, Ayushi Pokhriyal and Namrata Rastogi

SynOpen, 2022, 06, 198
DOI: 10.1055/s-0042-1751360

Direct Synthesis of Pyrroles by Dehydrogenative Coupling of Diols and Amines Catalyzed by Cobalt Pincer Complexes

Prosenjit Daw, Subrata Chakraborty, Jai Anand Garg, Yehoshoa Ben‐David and David Milstein

Angewandte Chemie, 2016, 128, 14585
DOI: 10.1002/ange.201607742

Synthesis, characterization, X-ray crystallographic study and in silico ADME predictions of functionalized nitropyrrole derivatives

Saigal, Mohammad Khizr, Subash C. Sahoo and Md. Musawwer Khan

Journal of Molecular Structure, 2022, 1250, 131655
DOI: 10.1016/j.molstruc.2021.131655

Bifurcated Rhodaelectro-catalyzed C–H Activation for the Synthesis of Pyrroles and Lactones

Simon L. Homölle, Maximilian Stangier, Efraim Reyes and Lutz Ackermann

Precision Chemistry, 2023, 1, 382
DOI: 10.1021/prechem.3c00061

Solvent‐Controlled C2/C5‐Regiodivergent Alkenylation of Pyrroles

Youla Su, Shang Gao, Yue Huang, Aijun Lin and Hequan Yao

Chemistry A European J, 2015, 21, 15820
DOI: 10.1002/chem.201502418

Self-Assembly of Pyrrole-Centered Pentaheterocyclic Ensembles in the System Hetarenecarbonitrile/Ethynylhetarene/t-BuOK/DMSO

E. Yu. Schmidt, N. A. Lobanova, I. V. Tatarinova, I. A. Ushakov and B. A. Trofimov

Russ J Org Chem, 2025, 61, 1279
DOI: 10.1134/S1070428025602663

Cascade Reaction of Morita–Baylis–Hillman Acetates with 1,1-Enediamines or Heterocyclic Ketene Aminals: Synthesis of Highly Functionalized 2-Aminopyrroles

Jin Liu, Qi Li, Zheng-Mao Cao, Yi Jin, Jun Lin and Sheng-Jiao Yan

J. Org. Chem., 2019, 84, 1797
DOI: 10.1021/acs.joc.8b02594

Synthesis and Toxicity Evaluation of New Pyrroles Obtained by the Reaction of Activated Alkynes with 1-Methyl-3-(cyanomethyl)benzimidazolium Bromide

Beatrice-Cristina Ivan, Florea Dumitrascu, Adriana Iuliana Anghel, Robert Viorel Ancuceanu, Sergiu Shova, Denisa Dumitrescu, Constantin Draghici, Octavian Tudorel Olaru, George Mihai Nitulescu, Mihaela Dinu and Stefania-Felicia Barbuceanu

Molecules, 2021, 26, 6435
DOI: 10.3390/molecules26216435

[3+2] Cycloaddition reactions of 1-substituted 3,3,3-trifluoropropenes with isonitriles – synthesis of pyrroles and pyrrolines

Yuriy N. Markitanov, Vadim M. Timoshenko, Eduard B. Rusanov and Yuriy G. Shermolovich

Chem Heterocycl Comp, 2021, 57, 253
DOI: 10.1007/s10593-021-02901-x

Divergent Conversion of Double Isocyanides with Alkenyl Bromide to Polysubstituted Pyrroles and 4-Imino-4,5-dihydropyrrolo[3,4-b]pyrrol-6(1H)-one Derivatives by Pd-Catalyzed Tandem Cyclization Reactions

Zhi-Lin Ren, Ji-Ying Qiu, Ling-Ling Yuan, Yue-Fei Yuan, Shuang Cai, Jun Li, Chi Kong, Ping He and Long Wang

Org. Lett., 2022, 24, 859
DOI: 10.1021/acs.orglett.1c04146

Crystal structure and Hirshfeld surface analysis of (2E)-1-phenyl-3-(1H-pyrrol-2-yl)propen-1-one

Ayten S. Safarova, Ali N. Khalilov, Mehmet Akkurt, Abel M. Maharramov, Ajaya Bhattarai, Farid N. Naghiyev and İbrahim G. Mamedov

Acta Crystallogr E Cryst Commun, 2024, 80, 191
DOI: 10.1107/S2056989024000495

Synthesis, Insecticidal Evaluation, and 3D-QASR of Novel Anthranilic Diamide Derivatives Containing N-Arylpyrrole as Potential Ryanodine Receptor Activators

Changchun Wu, Xiaobo Yu, Baolei Wang, Jingbo Liu, Fanfei Meng, Yangyang Zhao, Lixia Xiong, Na Yang, Yuxin Li and Zhengming Li

J. Agric. Food Chem., 2020, 68, 9319
DOI: 10.1021/acs.jafc.0c04157

Cobalt(II)-Catalyzed Synthesis of γ-Diketones from Aryl Alkenes and Its Utilization in the Synthesis of Various Heterocyclic Compounds

Subham Sau, Krishna Mohan Das, Bijan Mondal and Arunabha Thakur

J. Org. Chem., 2024, 89, 7095
DOI: 10.1021/acs.joc.4c00487

Unusual N H/O H Activation Mechanism for Au-Catalyzed N,O-Functionalization of 1,4-diyn-3-ols with N-hydroxyanilines

Yuxia Liu, Xufang Zhao, Jing Zhang, Jianbo Tong, Guang Chen, Siwei Bi and Tony D. James

Molecular Catalysis, 2024, 559, 114055
DOI: 10.1016/j.mcat.2024.114055

General Transition Metal-Free Synthesis of NH-Pyrroles from Secondary Alcohols and 2-Aminoalcohols

Besir Krasniqi, Kayle Geerts and Wim Dehaen

J. Org. Chem., 2019, 84, 5027
DOI: 10.1021/acs.joc.8b03215

Conversion of Isoxazoles to Functionalized Pyrrole and Isoquinoline Derivatives via ROCC Mechanism

Karri Raghavulu, Varukolu Shanker, Ramakrishna Gudipati, Keloth Basavaiah, Raju Doddipalla, Mahipal Yadav, Satyanarayana Yennam and Manoranjan Behera

Helvetica Chimica Acta, 2024, 107
DOI: 10.1002/hlca.202400057

Bacillus velezensis PEA1 Inhibits Fusarium oxysporum Growth and Induces Systemic Resistance to Cucumber Mosaic Virus

Ahmed Abdelkhalek, Said I. Behiry and Abdulaziz A. Al-Askar

Agronomy, 2020, 10, 1312
DOI: 10.3390/agronomy10091312

Acetic Acid‐Catalyzed Selective Synthesis of N‐Substituted 2‐Amino‐3‐Cyanopyrroles via a Three‐Component Reaction Between Carbohydrates, Primary Amines and Malononitrile

Mengxin Xia, Ziad Moussa and Zaher M. A. Judeh

Asian J Org Chem, 2022, 11
DOI: 10.1002/ajoc.202200367

Synthesis of 4,5-Disubstituted Methyl 1H-Pyrrole-2-carboxylates from 3-Chloroacrylaldehydes and Hippuric Acid

Anna L. Samsonenko, Anastasia S. Kostyuchenko, Tatyana Yu. Zheleznova, Vladislav Yu. Shuvalov, Evgenii B. Uliankin, Anton L. Shatsauskas and Alexander S. Fisyuk

Synthesis, 2024, 56, 2423
DOI: 10.1055/a-2295-8544

Urinary odor molecules in the Otassha Study can distinguish patients with sarcopenia: A pilot study

Takuya Oka, Akiko Fujita, Hisashi Kawai, Shuichi P Obuchi, Hiroyuki Sasai, Hirohiko Hirano, Kazushige Ihara, Yoshinori Fujiwara, Masashi Tanaka and Keiko Kato

Geriatrics Gerontology Int, 2025, 25, 307
DOI: 10.1111/ggi.15072

Barton–Zard Reaction of β-Fluoro-β-nitrostyrenes─a Selective Route to Functionalized 4-Fluoropyrroles

Roman V. Larkovich, Victoria E. Shambalova, Savva A. Ponomarev, Alexander S. Aldoshin, Konstantin A. Lyssenko, Mikhail S. Nechaev and Valentine G. Nenajdenko

J. Org. Chem., 2023, 88, 10122
DOI: 10.1021/acs.joc.3c00935

One-Pot Synthesis of 2-Acetyl-1H-pyrroles from N-Propargylic β-Enaminones via Intermediacy of 1,4-Oxazepines

Nilay Kanova, Buse Aysen Dundar, Yilmaz Kelgokmen and Metin Zora

J. Org. Chem., 2021, 86, 6289
DOI: 10.1021/acs.joc.1c00077

Sustainable Synthesis of N-Alkyl-Pyrrolecarboxylic and Pyrrolepyrazinones Derivatives from Biosourced 3-Hydroxy-2-pyrones and Amines

Gabriella Leonardi, Ada Truscello, Grazia Isa C. Righetti, Giovanni Gennaro Mondrone, Luca Mascheroni, Attilio Citterio and Roberto Sebastiano

ACS Sustainable Chem. Eng., 2022, 10, 12763
DOI: 10.1021/acssuschemeng.2c03661

Research Progress in the Synthesis of DihydropyrrolizineCompounds

祥南孔

JOCR, 2024, 12, 406
DOI: 10.12677/jocr.2024.122039

Structure and electronics in 1H-pyrrol-2-ylmethylene compounds

Briana R. Schrage, Victor N. Nemykin and Christopher J. Ziegler

Tetrahedron, 2020, 76, 131149
DOI: 10.1016/j.tet.2020.131149

The Paal–Knorr Pyrroles Synthesis: A Green Perspective

Shakeel Alvi, Ahmad Hasan and Rashid Ali

Polycyclic Aromatic Compounds, 2024, 44, 3558
DOI: 10.1080/10406638.2023.2225676

Difluoroketenimine: Generation from Difluorocarbene and Isocyanide and Its [3 + 2] Cycloadditions with Alkenes or Alkynes

Rui Zhang, Zhikun Zhang, Kang Wang and Jianbo Wang

J. Org. Chem., 2020, 85, 9791
DOI: 10.1021/acs.joc.0c01120

Synthesis, characterization, and antimicrobial activity investigations of ruthenium (II)–bipyridine complexes of ciprofloxacin derivatives

Dhuha Al‐Wahaib, Ali El‐Dissouky, Nada M. Abrar and Tarek E. Khalil

Applied Organom Chemis, 2021, 35
DOI: 10.1002/aoc.6407

Synthesis of nitrogen, phosphorus, selenium and sulfur-containing heterocyclic compounds – Determination of their carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase and α-glycosidase inhibition properties

İlhami Gülçin, Boris Trofimov, Ruya Kaya, Parham Taslimi, Lyubov Sobenina, Elena Schmidt, Olga Petrova, Svetlana Malysheva, Nina Gusarova, Vagif Farzaliyev, Afsun Sujayev, Saleh Alwasel and Claudiu T. Supuran

Bioorganic Chemistry, 2020, 103, 104171
DOI: 10.1016/j.bioorg.2020.104171

Synthesis of Dihydropyrrolizine and Tetrahydroindolizine Scaffolds from Pyrroles by Titanocene(III) Catalysis

Sven Hildebrandt and Andreas Gansäuer

Angew Chem Int Ed, 2016, 55, 9719
DOI: 10.1002/anie.201603985

Synthesis, dielectric properties, molecular docking and ADME studies of pyrrole-3-ones

İrfan Çapan, Mehmet Gümüş, Halil Gökce, Hidayet Çetin, Yusuf Sert and İrfan Koca

Journal of Biomolecular Structure and Dynamics, 2022, 40, 8655
DOI: 10.1080/07391102.2021.1914174

Synthesis, Molecular Structure, Anticancer Activity, and QSAR Study of N-(aryl/heteroaryl)-4-(1H-pyrrol-1-yl)Benzenesulfonamide Derivatives

Beata Żołnowska, Jarosław Sławiński, Zdzisław Brzozowski, Anna Kawiak, Mariusz Belka, Joanna Zielińska, Tomasz Bączek and Jarosław Chojnacki

IJMS, 2018, 19, 1482
DOI: 10.3390/ijms19051482

Pyrrolo[1,2-a]azepines Coupled with Benzothiazole and Fluorinated Aryl Thiourea Scaffolds as Promising Antioxidant and Anticancer Agents

Rahul V. Patel, Bhupendra M. Mistry, Riyaz Syed, Nikhil M. Parekh and Han-Seung Shin

ACAMC, 2019, 19, 1855
DOI: 10.2174/1871520619666190820151043

Iron-Catalyzed Sustainable Synthesis of Pyrrole

Balakumar Emayavaramban, Malay Sen and Basker Sundararaju

Org. Lett., 2017, 19, 6
DOI: 10.1021/acs.orglett.6b02819

Three-Component Ordered Annulation of Amines, Ketones, and Nitrovinylarenes: Access to Fused Pyrroles and Substituted Indoles under Metal-Free Conditions

Jinjin Chen, Dan Chang, Fuhong Xiao and Guo-Jun Deng

J. Org. Chem., 2019, 84, 568
DOI: 10.1021/acs.joc.8b02410

Delineating the binding site of a series of gold(III) Schiff base chelates on HSA via experimentation and in silico methods

Sheldon Sookai and Orde Q. Munro

International Journal of Biological Macromolecules, 2025, 315, 144317
DOI: 10.1016/j.ijbiomac.2025.144317

Recent advances in sustainable catalytic production of 5-methyl-2-pyrrolidones from bio-derived levulinate

Yiyuan Jiang, Zao Li, Yuncong Li, Long Chen, Heng Zhang, Hu Li and Song Yang

Fuel, 2023, 334, 126629
DOI: 10.1016/j.fuel.2022.126629

Synthesis of N-Substituted Pyrroles Catalyzed by Low-Cost and Commercially Available Aluminas

Omar Portilla-Zúñiga, Óscar Bautista-Aguilera, José Martínez, Hugo Rojas, Mario Macías, Isabel Iriepa, Adrián Pérez-Redondo, Ángel Sathicq, Juan-Carlos Castillo and Gustavo Romanelli

Catalysts, 2023, 13, 603
DOI: 10.3390/catal13030603

N-Aryl Pyrrole Synthesis from Biomass-Derived Furans and Arylamine over Lewis Acidic Hf-Doped Mesoporous SBA-15 Catalyst

Yao-Bing Huang, Yu-Jia Luo, Antonio Del Rio Flores, Li-Cheng Li and Fei Wang

ACS Sustainable Chem. Eng., 2020, 8, 12161
DOI: 10.1021/acssuschemeng.0c03578

Annulation of five-membered cyclic enols with 3-aryl-2H-azirines: Catalytic versus non-catalytic cycloaddition

Pavel A. Sakharov, Nikolai V. Rostovskii, Alexander F. Khlebnikov and Mikhail S. Novikov

Tetrahedron, 2017, 73, 4663
DOI: 10.1016/j.tet.2017.06.037

Molybdenum‐Catalyzed Direct Synthesis of Pyrroles from Nitroarenes with Glycols as Reductants

Sara Gómez‐Gil, Samuel Suárez‐Pantiga, María R. Pedrosa and Roberto Sanz

Adv Synth Catal, 2025, 367
DOI: 10.1002/adsc.202401170

Flexible Construction of Functionalized‐Pyrroles under Palladium or Copper Catalysis in the Presence of BF3 ⋅ Et2O

Yin Liu, Teng Liu, Biwei Yan, Kun Wei and Wusheng Guo

Adv Synth Catal, 2022, 364, 916
DOI: 10.1002/adsc.202101292

Synthesis, characterisation and catalytic activity of 4, 5-imidazoledicarboxylate ligated Co(II) and Cd(II) metal-organic coordination complexes

Kranthi Kumar Gangu, Suresh Maddila, Saratchandra Babu Mukkamala and Sreekantha B. Jonnalagadda

Journal of Molecular Structure, 2017, 1143, 153
DOI: 10.1016/j.molstruc.2017.04.083

Regioselective synthesis of pyrrole and indole-fused isocoumarins catalysed by N $$^\wedge $$ ∧ O chelate ruthenium(II) complex

Keisham S Singh, Sneha G Sawant and Werner Kaminsky

J Chem Sci, 2018, 130
DOI: 10.1007/s12039-018-1519-z

Mass Spectra of New Heterocycles: XVIII. Electron Impact and Chemical Ionization Mass Spectra of Alkyl 5-Amino-3-methyl-4-(1H-pyrrol-1-yl)thiophene-2-carboxylates

L. V. Klyba, N. A. Nedolya, E. R. Sanzheeva and O. A. Tarasova

Russ J Org Chem, 2019, 55, 518
DOI: 10.1134/S1070428019040171

Unpredictable Dynamic Behaviour of Ruthenium Chelate Pyrrole Derivatives

Giacomo Drius, Riccardo Tarroni, Matteo Birchmeier, Carola Parolin, Carla Boga, Magda Monari and Silvia Bordoni

Molecules, 2024, 29, 3068
DOI: 10.3390/molecules29133068

Small molecule based targeting of the CssA RNA thermometer: insights from computational and biophysical approaches

Akanksha Sharma, Priyanka Gopi, Rimjhim Trivedi, Dinesh Kumar, Janeka Gartia, Adukamparai Rajukrishnan Suresh Babu, Prateek Pandya, Gurpal Singh and Ravi Pratap Barnwal

Biochimie, 2025, 237, 110
DOI: 10.1016/j.biochi.2025.07.017

Development of a palladium-catalyzed decarboxylative arene cross-coupling of pyrrole derivatives in a flow reactor

Cindy Buonomano, Michael Holtz-Mulholland, Sydney Sullivan and Pat Forgione

J Flow Chem, 2022, 12, 275
DOI: 10.1007/s41981-022-00222-4

One-Pot Synthesis of Unprotected 2-Acylpyrroles from 1,2,3-Triazoles and 2-Hydroxymethylallyl Carbonates

Jong-Un Park, Liang-Zhu Huang, Ho-Jun Cho, Boyoung Y. Park and Ju Hyun Kim

J. Org. Chem., 2023, 88, 585
DOI: 10.1021/acs.joc.2c02602

Non-Covalent Functionalisation of C30 Fullerene by Pyrrole-n-Carboxylic Acid (n=2, 3): Density Functional Theory Studies

Kun Harismah, Mahmoud Mirzaei, Nahid Ghasemi and Mohammad Nejati

Zeitschrift für Naturforschung A, 2017, 73, 51
DOI: 10.1515/zna-2017-0233

Evaluation of ecotoxicological impact of new pyrrole-derived aminophosphonates using selected bioassay battery

Jarosław Lewkowski, Marta Morawska, Rafał Karpowicz, Piotr Rychter, Diana Rogacz, Kamila Lewicka and Piotr Dobrzyński

Ecotoxicology, 2017, 26, 914
DOI: 10.1007/s10646-017-1821-4

Iodine-catalyzed tandem oxidative coupling reaction: A one-pot strategy for the synthesis of new coumarin-fused pyrroles

Hoda Yahyavi, Majid M. Heravi, Mohammad Mahdavi and Alireza Foroumadi

Tetrahedron Letters, 2018, 59, 94
DOI: 10.1016/j.tetlet.2017.11.055

Discovery of Conformationally Constrained Dihydro Benzo-Indole Derivatives as Metallo-β-Lactamase Inhibitors to Tackle Multidrug-Resistant Bacterial Infections

Pulkit Dhiman, Satyajeet Das, Vikas Pathania, Suraj Rawat, Hemraj S. Nandanwar, Krishan G. Thakur and Vinod D. Chaudhari

J. Med. Chem., 2025, 68, 7062
DOI: 10.1021/acs.jmedchem.4c02207

Chemical fixation of CO2 to 2-aminobenzonitriles: A straightforward route to quinazoline-2,4(1H,3H)-diones with green and sustainable chemistry perspectives

Esmail Vessally, Somayeh Soleimani-Amiri, Akram Hosseinian, Ladan Edjlali and Mirzaagha Babazadeh

Journal of CO2 Utilization, 2017, 21, 342
DOI: 10.1016/j.jcou.2017.08.006

Evidence of cluster formation of pyrrole with mixed silver metal clusters, Agx-My (x = 4,5, y = 2/1 and M = Au/Ni/Cu) using DFT/SERS analysis

Jamelah S. Al-Otaibi, Y. Sheena Mary, Y. Shyma Mary and Renjith Thomas

Computational and Theoretical Chemistry, 2022, 1208, 113569
DOI: 10.1016/j.comptc.2021.113569

Application of the ring-closing metathesis to the formation of 2-aryl-1H-pyrrole-3-carboxylates as building blocks for biologically active compounds

Katarzyna Grychowska, Bartłomiej Kubica, Marcin Drop, Evelina Colacino, Xavier Bantreil, Maciej Pawłowski, Jean Martinez, Gilles Subra, Paweł Zajdel and Frédéric Lamaty

Tetrahedron, 2016, 72, 7462
DOI: 10.1016/j.tet.2016.09.059

Computational-Based Discovery of the Anti-Cancer Activities of Pyrrole-Based Compounds Targeting the Colchicine-Binding Site of Tubulin

Sergei Boichuk, Kirill Syuzov, Firuza Bikinieva, Aigul Galembikova, Svetlana Zykova, Ksenia Gankova, Sergei Igidov and Nazim Igidov

Molecules, 2022, 27, 2873
DOI: 10.3390/molecules27092873

The Dawn of Functional Organoarsenic Chemistry

Hiroaki Imoto and Kensuke Naka

Chemistry A European J, 2019, 25, 1883
DOI: 10.1002/chem.201804114

A Copper‐Catalyzed Three‐Component Reaction for the Preparation of Polysubstituted Pyrroles from Alkynyl Ketones, Amines and Isocyanoacetates

Yingying Shan, Jianming Li, Yutong Zhao, Dianpeng Chen, Qinyu Li and Jinmao You

ChemistrySelect, 2019, 4, 9497
DOI: 10.1002/slct.201902968

Transition‐Metal Free Arylation of Therapeutically Important Heterocycles

Ambarish Priyadarshan, Garima Tripathi, Naresh Murty Venneti, Kaushal Kishor, Anil Kumar Singh and Abhijeet Kumar

ChemistrySelect, 2024, 9
DOI: 10.1002/slct.202400363

Metallo Protic N-Allyl Enammonium Ylide 3-Aza-Cope Rearrangement Enabled by Resonance-Assisted H-Bonding: Direct Access to Functionalized Pyrroles

Laxman Anandrao Thorbole, Sudhir Muduli and Sreenivas Katukojvala

Org. Lett., 2026
DOI: 10.1021/acs.orglett.6c01121

[3+2] Anionic Cycloaddition of Isocyanides to Acyclic Enamines and Enaminones: A New, Simple, and Convenient Method for the Synthesis of 2,4‐Disubstituted Pyrroles

Ilya V. Efimov, Maria D. Matveeva, Rafael Luque, Vasiliy A. Bakulev and Leonid G. Voskressensky

Eur J Org Chem, 2020, 2020, 1108
DOI: 10.1002/ejoc.201901776

Synthesis of Azulene-Substituted Tetraarylpyrroles by Reaction of 1-Azulenyl Ketones with Benzoin and Ammonium Acetate

Taku Shoji, Sho Takagaki, Miwa Tanaka, Takanori Araki, Shuhei Sugiyama, Ryuta Sekiguchi, Akira Ohta, Shunji Ito and Tetsuo Okujima

HETEROCYCLES, 2017, 94, 1870
DOI: 10.3987/COM-17-13781

A review on multi-component green synthesis of N-containing heterocycles using mixed oxides as heterogeneous catalysts

Sandeep V.H.S. Bhaskaruni, Suresh Maddila, Kranthi Kumar Gangu and Sreekantha B. Jonnalagadda

Arabian Journal of Chemistry, 2020, 13, 1142
DOI: 10.1016/j.arabjc.2017.09.016

Base‐Promoted Synthesis of N−H Free Pyrroles via net [3+2]‐Cycloaddition

Huimin Jin, Fan Zhou, Zhenhua Xiang, Lingfeng Chen, Guang Liang, Patrick J. Walsh and Jie Li

Adv Synth Catal, 2024, 366, 942
DOI: 10.1002/adsc.202301053

Effect of Methyl Substitution on the N–H···O Interaction in Complexes of Pyrrole with Water, Methanol, and Dimethyl Ether: Matrix Isolation Infrared Spectroscopy and ab Initio Computational Studies

Shubhra Sarkar, N. Ramanathan and K. Sundararajan

J. Phys. Chem. A, 2018, 122, 2445
DOI: 10.1021/acs.jpca.8b00023

Self-Assembly of 4,4′-Linked Dipyrromethanes from Unconventional Reactants─Propargylamines, 2-(Vinyloxy)ethyl Isothiocyanate, and Alkylating Agents under Basic Conditions

Nina A. Nedolya, Ol’ga A. Tarasova, Alexander I. Albanov, Lyudmila V. Klyba and Boris A. Trofimov

J. Org. Chem., 2024, 89, 864
DOI: 10.1021/acs.joc.3c01732

An Efficient One-Pot Synthesis of 5-Sulfanyl-1-[2-(vinyloxy)ethyl]-1H-pyrrol-2-amines as Precursors of 1-Vinylpyrroles

Olga A. Tarasova, Nina A. Nedolya, Alexander I. Albanov and Boris A. Trofimov

Synthesis, 2022, 54, 4033
DOI: 10.1055/a-1820-6160

Synthesis of Highly Substituted 3-Pyrrolin-2-ones from N,N-Disubstituted α-Amino Acids

Víctor Samper Barceló and Stefan Bienz

J. Org. Chem., 2018, 83, 2734
DOI: 10.1021/acs.joc.7b03187

Synthesis and odor characteristics of N‐substituted pyrrolyl ketones derived from N‐substituted acetylpyrroles and alcohols

Mingqin Zhao, Jingyi Hu, Xiaoming Ji, Lu Han, Mengxiao Li and Miao Lai

Journal of Heterocyclic Chem, 2023, 60, 596
DOI: 10.1002/jhet.4612

Phosphorus-Containing Alkynes in the Synthesis of Heterocyclic Compounds (A Review)

A. A. Sokolov, D. M. Egorov, A. V. Dogadina and N. I. Svintsitskaya

Russ J Gen Chem, 2024, 94, 558
DOI: 10.1134/S1070363224030095

Synthesis of New 2-Pyridinone and 2-Iminochromene Derivatives Bearing Biologically Active Pyrrole Moiety as Expected Antibacterial and Antifungal Agents

Reem A. K. Al-Harbi, Marwa A. M. Sh. El-Sharief and Samir Y. Abbas

Polycyclic Aromatic Compounds, 2024, 44, 4430
DOI: 10.1080/10406638.2023.2254892

Development of a new method for activation of isotope exchange

V. P. Shevchenko, I. Yu. Nagaev, K. V. Shevchenko and N. F. Myasoedov

Radiohimiâ, 2023, 65, 349
DOI: 10.31857/S0033831123040068

Lewis acid-catalyzed solvent-free multicomponent reactions: Synthesis and structural features of fused pyrrole-chromenes

Silmara L.G. Alves, Matheus V. Machado, Andreza M. Moraes, Leonã S. Flores, Charlane C. Corrêa, Jefferson L. Princival and José A.F.P. Villar

Tetrahedron, 2026, 196, 135270
DOI: 10.1016/j.tet.2026.135270

Direct Synthesis of Pyrroles via Heterogeneous Catalytic Condensation of Anilines with Bioderived Furans

Lei Tao, Zi-Jian Wang, Tian-Hao Yan, Yong-Mei Liu, He-Yong He and Yong Cao

ACS Catal., 2017, 7, 959
DOI: 10.1021/acscatal.6b02953

β,β,β‐Trichloroethyl‐NH‐Enamine as Viable System for 5‐Endo‐trig Radical Cyclization via Multifaceted CuI−CuII Redox Catalysis: Single Step Synthesis of Multi‐Functionalized NH‐Pyrroles

Ram N. Ram, Sandhya Sadanandan and Dharmendra Kumar Gupta

Adv Synth Catal, 2019, 361, 5661
DOI: 10.1002/adsc.201900938

Synthesis of cyclodextrin–pyrrole conjugates possessing tuneable carbon linkers

Jan Lukášek, Markéta Řezanková, Ivan Stibor and Michal Řezanka

J Incl Phenom Macrocycl Chem, 2018, 92, 339
DOI: 10.1007/s10847-018-0854-5

Palladium-Catalyzed Enantioselective Decarboxylative Allylic Alkylation of Acyclic α-N-Pyrrolyl/Indolyl Ketones

Remi Lavernhe, Eric J. Alexy, Haiming Zhang and Brian M. Stoltz

Org. Lett., 2020, 22, 4272
DOI: 10.1021/acs.orglett.0c01303

Oxime ethers as useful synthons in the synthesis of a number of key medicinal heteroaromatic compounds

Esmail Vessally and Morteza Abdoli

J IRAN CHEM SOC, 2016, 13, 1235
DOI: 10.1007/s13738-016-0838-6

Unlocking the Potential of Pyrrole: Recent Advances in New Pyrrole-Containing Compounds with Antibacterial Potential

Aura Rusu, Octavia-Laura Oancea, Corneliu Tanase and Livia Uncu

IJMS, 2024, 25, 12873
DOI: 10.3390/ijms252312873

Drought Exposed Burkholderia seminalis JRBHU6 Exhibits Antimicrobial Potential Through Pyrazine-1,4-Dione Derivatives Targeting Multiple Bacterial and Fungal Proteins

Jay Kishor Prasad, Priyanka Pandey, Richa Anand and Richa Raghuwanshi

Front. Microbiol., 2021, 12
DOI: 10.3389/fmicb.2021.633036

Solvent-free Approaches towards the Synthesis of Therapeutically Important Heterocycles

Ambarish Priyadarshan, Garima Tripathi, Anil Kumar Singh, Sanchayita Rajkhowa, Abhijeet Kumar and Vinod Kumar Tiwari

CGC, 2024, 11, 127
DOI: 10.2174/2213346110666230915163034

Proteinase Resistance of Carnosine, Pyrrolylcarnosine and Salicylcarnosine

K. V. Shevchenko, I. Yu. Nagaev, O. I. Kulikova, S. L. Stvolinsky, V. P. Shevchenko and N. F. Myasoedov

Russ J Bioorg Chem, 2024, 50, 401
DOI: 10.1134/S1068162024020201

Tandem Enantioselective Cycloaromatization/Intramolecular Friedel–Crafts Desymmetrization of Cyclohexadienones

Daniel Gaviña, Marta Durán, Lidia Prieto, Marcos Escolano, Santiago Díaz‐Oltra, María Sánchez‐Roselló and Carlos del Pozo

Adv Synth Catal, 2024, 366, 3881
DOI: 10.1002/adsc.202400576

Isoxazole Strategy for the Synthesis of α-Aminopyrrole Derivatives

Ekaterina E. Galenko, Stanislav A. Linnik, Olesya V. Khoroshilova, Mikhail S. Novikov and Alexander F. Khlebnikov

J. Org. Chem., 2019, 84, 11275
DOI: 10.1021/acs.joc.9b01634

Inhibitory Effects of Nitrogenous Metabolites from a Marine-Derived Streptomyces bacillaris on Isocitrate Lyase of Candida albicans

Beomkoo Chung, Ji-Yeon Hwang, Sung Chul Park, Oh-Seok Kwon, Eunji Cho, Jayho Lee, Hyi-Seung Lee, Dong-Chan Oh, Jongheon Shin and Ki-Bong Oh

Marine Drugs, 2022, 20, 138
DOI: 10.3390/md20020138

Diastereoselective Synthesis of Rauhut–Currier-Type Adducts via an Unexpected α-Addition of α,β-Unsaturated γ-Butyrolactams to Coumarin Derivatives

Shu-Mei Yang, Ganapuram Madhusudhan Reddy, Meng-Hsien Liu, Tzu-Ping Wang, Jhen-Kuei Yu and Wenwei Lin

J. Org. Chem., 2017, 82, 781
DOI: 10.1021/acs.joc.6b02526

A comprehensive survey upon diverse and prolific applications of chitosan-based catalytic systems in one-pot multi-component synthesis of heterocyclic rings

Hossein Mousavi

International Journal of Biological Macromolecules, 2021, 186, 1003
DOI: 10.1016/j.ijbiomac.2021.06.123

Calcium‐Catalyzed Intramolecular Hydroamination‐Deacylation Reaction of in situ formed β‐Amino Allenes

Srinivasarao Yaragorla, Dandugula Sneha Latha and Pallava Rajesh

Adv Synth Catal, 2021, 363, 5486
DOI: 10.1002/adsc.202101022

Photochemical Hydroacylation of Activated Alkenes via H‐Bonded Donor–Acceptor Complex

Rahul Singh, Pratibha Choudhary, Harshit Jain and Debashis Adhikari

Adv Synth Catal, 2026, 368
DOI: 10.1002/adsc.70344

Bis(imido)vanadium(V)-Catalyzed [2+2+1] Coupling of Alkynes and Azobenzenes Giving Multisubstituted Pyrroles

Kento Kawakita, Evan P. Beaumier, Yuya Kakiuchi, Hayato Tsurugi, Ian A. Tonks and Kazushi Mashima

J. Am. Chem. Soc., 2019, 141, 4194
DOI: 10.1021/jacs.8b13390

MPC@But-SO3H a mesoporous heterogeneous organocatalyst in one-pot tandem synthesis of dihydroindeno[1,2-b]pyrrole derivatives

Atif Mustafa, Nazia Zameer, Nida Khan and Zeba N. Siddiqui

Tetrahedron, 2024, 167, 134233
DOI: 10.1016/j.tet.2024.134233

In vitro screening and in silico prediction of antifungal metabolites from rhizobacterium Achromobacter kerstersii JKP9

Karuppiah Vijay, Thangarasu Suganya Devi, Karthikeyan Kirupa Sree, Abdallah M. Elgorban, Ponnuchamy Kumar, Muthusamy Govarthanan and Thangavel Kavitha

Arch Microbiol, 2020, 202, 2855
DOI: 10.1007/s00203-020-01982-0

Photoredox Catalyzed Cyclization of Enaminones/Ketene N,S-Acetals with β-Ketodinitriles to Access Polysubstituted Pyrroles

Anup Kumar Sharma, Pratima Singh and Krishna Nand Singh

J. Org. Chem., 2025, 90, 13679
DOI: 10.1021/acs.joc.5c01759

Stable Bio-oil Production from Proteinaceous Cyanobacteria: Tail Gas Reactive Pyrolysis of Spirulina

Bruna M. E. Chagas, Charles A. Mullen, Christina Dorado, Yaseen Elkasabi, Akwasi A. Boateng, Marcus A.F. Melo and Carlos H. Ataíde

Ind. Eng. Chem. Res., 2016, 55, 6734
DOI: 10.1021/acs.iecr.6b00490