1-(N,N-Dialkylcarbamoyl)-1,1-difluoromethanesulfonyl ester as a stable and effective precursor for a neopentyl labeling group with astatine-211

Ichiro Sasaki, Masatoshi Tada, Ziyun Liu, Maho Tatsuta, Takeru Okura, Miho Aoki, Kazuhiro Takahashi, Noriko S. Ishioka, Shigeki Watanabe and Hiroshi Tanaka

Org. Biomol. Chem., 2023, 21, 7467
DOI: 10.1039/D3OB00944K

Substrate Study for Dihydroxyboryl Astatine Substitution Reaction with Fibroblast Activation Protein Inhibitor (FAPI)

Ayaka Aso, Kazuko Kaneda-Nakashima, Hinako Nabetani, Yuichiro Kadonaga, Yoshifumi Shirakami, Tadashi Watabe, Taku Yoshiya, Masayoshi Mochizuki, Yuki Koshino, Kazuhiro Ooe, Atsuko Kawakami, Naoya Jinno, Atsushi Toyoshima, Hiromitsu Haba, Yang Wang, Jens Cardinale, Frederik L. Giesel, Atsushi Shimoyama and Koichi Fukase

Chem. Lett., 2022, 51, 1091
DOI: 10.1246/cl.220391

Copper-mediated astatination of 211At-labelled prostate-specific membrane antigen probes in the presence of basic salts

Shigeki Watanabe, Yuto Kondo, Ichiro Sasaki, Yasuhiro Ohshima, Hiroyuki Kimura and Noriko S. Ishioka

Tetrahedron, 2024, 156, 133920
DOI: 10.1016/j.tet.2024.133920

Synthesis Principle and Practice with Radioactive Iodines and Astatine: Advances Made So Far

Taotao Dong, Zhenru Zhang, Weicai Li, Weibin Zhuo, Tongjiang Cui and Zijing Li

J. Org. Chem., 2024, 89, 11837
DOI: 10.1021/acs.joc.4c00593

Iodoarene Activation: Take a Leap Forward toward Green and Sustainable Transformations

Toshifumi Dohi, Elghareeb E. Elboray, Kotaro Kikushima, Koji Morimoto and Yasuyuki Kita

Chem. Rev., 2025, 125, 3440
DOI: 10.1021/acs.chemrev.4c00808

Development of a Neopentyl 211At‐Labeled Activated Ester Providing In Vivo Stable 211At‐Labeled Antibodies for Targeted Alpha Therapy

Masatoshi Tada, Yuta Kaizuka, Kento Kannaka, Hiroyuki Suzuki, Taiki Joho, Kazuhiro Takahashi, Tomoya Uehara and Hiroshi Tanaka

ChemMedChem, 2024
DOI: 10.1002/cmdc.202400369

Rapid Electrophilic 211At‐Astatination of Trimethylgermyl Arenes

Marius Müller, Umberto Maria Battisti, Merlin Zabrocki, Ellinor Hansson, Holger Jensen, Emma Aneheim, Sture Lindegren and Matthias Manfred Herth

ChemPlusChem, 2024
DOI: 10.1002/cplu.202400254

Targeted Molecular Imaging and Therapy Based on Nuclear and Optical Technologies

Mikako Ogawa

Biological & Pharmaceutical Bulletin, 2024, 47, 1066
DOI: 10.1248/bpb.b24-00008

Formation Of Gold‐Astatine Bonds in N‐Heterocyclic Carbene Complexes

Mathilde Ligeour, Sébastien G. Guillet, Clémence Maingueneau, Mikaël Croyal, Aurélien Planchat, Jean‐François Gestin, Nicolas Galland and François Guérard

Chemistry A European J, 2025, 31
DOI: 10.1002/chem.202500826

Astatine-211 radiolabelling chemistry: from basics to advanced biological applications

Maarten Vanermen, Mathilde Ligeour, Maria-Cristina Oliveira, Jean-François Gestin, Filipe Elvas, Laurent Navarro and François Guérard

EJNMMI radiopharm. chem., 2024, 9
DOI: 10.1186/s41181-024-00298-4

Production of 211At and automated radiosynthesis of [211At]MABG via electrophilic astatodesilylation

Yuto Kondo, Taiki Joho, Shigenori Sasaki, Kazumasa Mochizuki, Naoko Hasegawa, Naoyuki Ukon, Ken-ichi Nishijima, Kohshin Washiyama, Hiroshi Tanaka, Tatsuya Higashi, Noriko S. Ishioka and Kazuhiro Takahashi

EJNMMI radiopharm. chem., 2025, 10
DOI: 10.1186/s41181-025-00376-1

Astatine‐211—Towards In Vivo Stable Astatine‐211 Labeled Radiopharmaceuticals and Their (Pre)Clinical Applications

Marius Müller, Nadia Bom Pedersen, Vladimir Shalgunov, Andreas Ingemann Jensen, Umberto Maria Battisti and Matthias Manfred Herth

Medicinal Research Reviews, 2025
DOI: 10.1002/med.70008

211At and 125I‐Labeling of (Hetero)Aryliodonium Ylides: Astatine Wins Again

Clémence Maingueneau, Marion Berdal, Romain Eychenne, Joëlle Gaschet, Michel Chérel, Jean‐François Gestin and François Guérard

Chemistry A European J, 2022, 28
DOI: 10.1002/chem.202104169