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High-Throughput Screening for the Discovery of Enzyme Inhibitors

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Scanning Protein Surfaces with DNA‐Encoded Libraries

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Massively Parallel Optimization of the Linker Domain in Small Molecule Dimers Targeting a Toxic r(CUG) Repeat Expansion

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Synthesis of a DNA‐Encoded Library of Pyrrolo[2,3‐d]pyrimidines

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Identification of isoform/domain-selective fragments from the selection of DNA-encoded dynamic library

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Recording Binding Information Directly into DNA-Encoded Libraries Using Terminal Deoxynucleotidyl Transferase

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G protein-coupled receptors: structure- and function-based drug discovery

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