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Recent Advances in Synthesis of Enantioenriched 2‐Substituted Piperidine Derivatives

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A convenient approach to δ-amino-β-ketoesters by vinylogous Mannich reaction of masked acetoacetates

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Tetrahedron, 2007, 63, 12317
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Alternative tandem cyclisation pathways in the reaction between imines and enones

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Tetrahedron, 2016, 72, 1105
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A new approach for the asymmetric synthesis of (2S,3S)-3-hydroxypipecolic acid

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Tetrahedron: Asymmetry, 2008, 19, 1200
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Aminoalkylation of Indoles with α‐Polyfluoroalkylated Cyclic Imines

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Eur J Org Chem, 2013, 2013, 2237
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Stereoselective Synthesis of (−)‐Pinidinone

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Cyclic Imine Nitro-Mannich/Lactamization Cascades: A Direct Stereoselective Synthesis of Multicyclic Piperidinone Derivatives

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Synthesis of Pyridine and Dihydropyridine Derivatives by Regio- and Stereoselective Addition toN-Activated Pyridines

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Asymmetric Disulfonimide‐Catalyzed Synthesis of δ‐Amino‐β‐Ketoester Derivatives by Vinylogous Mukaiyama–Mannich Reactions

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The natural alkaloid isoanabasine: synthesis from 2,3′-bipyridine, efficient resolution with BINOL, and assignment of absolute configuration by Mosher’s method

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Stereoselective synthesis of N-heterocycles: application of the asymmetric Cu-catalyzed addition of Et2Zn to functionalized alkyl and aryl imines

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A new asymmetric synthetic route to substituted piperidines

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Sequential C–H Arylation and Enantioselective Hydrogenation Enables Ideal Asymmetric Entry to the Indenopiperidine Core of an 11β-HSD-1 Inhibitor

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Stereoselective total synthesis of the piperidine alkaloids, (+)-coniine, (+)-pseudoconhydrine, and (+)-sedamine through a common intermediate

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Tetrahedron: Asymmetry, 2011, 22, 1000
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Gallium iodide/iodine as a versatile reagent for the aza-Prins cyclization: an expeditious synthesis of 4-iodopiperidines

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Diastereoselective total synthesis of piperidine alkaloids: (2R,5R)-5-hydroxyhomopipecolic acid and (2R,5R,8R)-5-hydroxysedamine

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Synthesis of 5-Amino- and 4-Hydroxy-2-phenylsulfonylmethylpiperidines

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Enantioselective Synthesis of (+)‐α‐Conhydrine and (–)‐Sedamine by L‐Proline‐Catalysed α‐Aminooxylation

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Expedient Pathway into Optically Active 2‐Oxopiperidines

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Synthetic Transformations of Sulfur‐Substituted 4‐Quinolizidinones

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Enantioselective Synthesis of ent-Sedridine and (+)-Coniine via Proline-Catalyzed Mannich Reaction

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Stereocontrolled reduction of chiral pyrrolidine and piperidine β-enamino esters: formal enantioselective synthesis of (+)-calvine

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Tetrahedron, 2005, 61, 7774
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Addition of dienolates to sulfinimines. Stereoselective synthesis of dihydropyridones

Robert Kawęcki

Tetrahedron, 2001, 57, 8385
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N‐Sulfinyl Amines as a Nitrogen Source in the Asymmetric Intramolecular Aza‐Michael Reaction: Total Synthesis of (−)‐Pinidinol

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Asymmetric syntheses of (−)-epi-pseudoconhydrine and (−)-5-hydroxysedamine based on a cis-diastereoselective 1,4-asymmetric induction

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Tetrahedron: Asymmetry, 2008, 19, 1297
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Synthesis of pyrrolidines and piperidines from ω-azidoalkylboronic esters. Stereocontrolled access to chiral nonracemic 2-and 3-substituted derivatives

Anne Salmon, Jean-Michel Jego and Bertrand Carboni

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Cp*Ir Complex-Catalyzed N-Heterocyclization of Primary Amines with Diols: A New Catalytic System for Environmentally Benign Synthesis of Cyclic Amines

Ken-ichi Fujita, Takeshi Fujii and Ryohei Yamaguchi

Org. Lett., 2004, 6, 3525
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FeCl3·6H2O catalyzed diastereoselective synthesis of (L)-menthyl 4-oxo-2-arylpiperidine-3-carboxylates

Lakshmi V.R. Babu Syamala and Ramakrishna G. Bhat

Tetrahedron Letters, 2017, 58, 4836
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