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A Conformationally Stable Acyclic β‐Hairpin Scaffold Tolerating the Incorporation of Poorly β‐Sheet‐Prone Amino Acids

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Rhodium‐Catalyzed Regioselective C7Ar‐Functionalization of Tryptophan with Quinones and its Late Stage Peptide Exemplification

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Unveiling the inhibitory mechanism of peptidomimetic inhibitor against Aβ42 aggregation and protofibril disaggregation by molecular dynamics

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Coupling Interrupted Fischer and Multicomponent Joullié‐Ugi to Chase Chemical Diversity: from Batch to Sustainable Flow Synthesis of Peptidomimetics

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Chemical Biology of Sortase A Inhibition: A Gateway to Anti-infective Therapeutic Agents

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Dehydropeptide Supramolecular Hydrogels and Nanostructures as Potential Peptidomimetic Biomedical Materials

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Harnessing RNA‐Protein Interactions for Therapeutic Interventions

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Recent Advances in Augmenting the Therapeutic Efficacy of Peptide–Drug Conjugates

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Ugi Reaction Synthesis of Oxindole–Lactam Hybrids as Selective Butyrylcholinesterase Inhibitors

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bioTCIs: Middle-to-Macro Biomolecular Targeted Covalent Inhibitors Possessing Both Semi-Permanent Drug Action and Stringent Target Specificity as Potential Antibody Replacements

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A heuristic, computer-driven and top-down approach to identify novel bioactive peptides: A proof-of-principle on angiotensin I converting enzyme inhibitory peptides

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Structure‐Based Design of Bicyclic Helical Peptides That Target the Oncogene β‐Catenin

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Peptidomimetics: An Overview of Recent Medicinal Chemistry Efforts toward the Discovery of Novel Small Molecule Inhibitors

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An Improved Turn Structure for Inducing β‐Hairpin Formation in Peptides

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Peptidomimetic-liganded gold nanoclusters for controlled iron delivery and synergistic suppression of tumor growth

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Antibiotic Potentiation as a Promising Strategy to Combat Macrolide Resistance in Bacterial Pathogens

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Antiviral Activity of Anthranilamide Peptidomimetics against Herpes Simplex Virus 1 and a Coronavirus

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Sustainable Synthesis of Pseudopeptides via Isocyanide-Based Multicomponent Reactions in Water

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Amide bioisosteric replacement in the design and synthesis of quorum sensing modulators

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Identification of a short ACE2-derived stapled peptide targeting the SARS-CoV-2 spike protein

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Topochemical Polymerization of Retro‐Isomeric Peptides for Tuning the Polymer Structure and Properties

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Peptides and peptidomimetics in the development of hydrogels towards the treatment of diabetic wounds

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Photocatalytic Functionalization of Dehydroalanine‐Derived Peptides in Batch and Flow

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Rhodium-Catalyzed Annulation of Vinylated Tyrosines with Internal Alkynes to Access Oxepine-Mounted Unnatural Tyrosines and Its Peptide Late Stage Functionalization

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Unusual Pseudopeptides: Syntheses and Structural Analyses of Ethylenediprolyl Peptides and Their Metal Complexes with Cu(II) Ion

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Novel Retro-Inverso Peptide Antibiotic Efficiently Released by a Responsive Hydrogel-Based System

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From Protein Structures to Functional Biomimetics

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The Use of Antibody-Antibiotic Conjugates to Fight Bacterial Infections

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The Peptide Functionalized Inorganic Nanoparticles for Cancer-Related Bioanalytical and Biomedical Applications

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Total Synthesis of Chaiyaphumines A-D: A Case Study Comparing Macrolactonization and Macrolactamization Approaches

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Revisiting Pyrimidine-Embedded Molecular Frameworks to Probe the Unexplored Chemical Space for Protein–Protein Interactions

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Peptide-Based Inhibitors of ADAM and ADAMTS Metalloproteinases

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Pd‐Catalyzed C(sp2)−H Alkoxycarbonylation of Phenethyl‐ and Benzylamines with Chloroformates as CO Surrogates

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Development of New Peptidomimetic NADPH Oxidase Inhibitors with Antithrombotic Properties

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Modular Synthesis of α-Aryl Acrylamido Carboxylic Acids by Triple C–F Bond Cleavage of (Trifluoromethyl)alkenes with Unprotected Amino Acids

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Design and SAR of Withangulatin A Analogues that Act as Covalent TrxR Inhibitors through the Michael Addition Reaction Showing Potential in Cancer Treatment

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Efficient Entropy‐Driven Inhibition of Dipeptidyl Peptidase III by Hydroxyethylene Transition‐State Peptidomimetics

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