Issue 68, 2014

Stereoselective construction of a key hydroindole precursor of epidithiodiketopiperazine (ETP) natural products

Abstract

An asymmetric synthetic strategy for constructing the divergent-synthesis monomer of epidithiodiketopiperazine (ETP) natural products has been successfully developed. The functionalized 2,3,3a,4,7,7a-hexahydroindole scaffold was constructed by a diastereoselective inverse electron-demand Diels–Alder (IEDDA) reaction.

Graphical abstract: Stereoselective construction of a key hydroindole precursor of epidithiodiketopiperazine (ETP) natural products

Supplementary files

Article information

Article type
Communication
Submitted
30 May 2014
Accepted
03 Jul 2014
First published
03 Jul 2014

Chem. Commun., 2014,50, 9690-9692

Author version available

Stereoselective construction of a key hydroindole precursor of epidithiodiketopiperazine (ETP) natural products

M. Feng and X. Jiang, Chem. Commun., 2014, 50, 9690 DOI: 10.1039/C4CC04148H

To request permission to reproduce material from this article, please go to the Copyright Clearance Center request page.

If you are an author contributing to an RSC publication, you do not need to request permission provided correct acknowledgement is given.

If you are the author of this article, you do not need to request permission to reproduce figures and diagrams provided correct acknowledgement is given. If you want to reproduce the whole article in a third-party publication (excluding your thesis/dissertation for which permission is not required) please go to the Copyright Clearance Center request page.

Read more about how to correctly acknowledge RSC content.

Social activity

Spotlight

Advertisements