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Issue 12, 2018
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Azidoheteroarylation of unactivated olefins through distal heteroaryl migration

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Abstract

The radical-mediated azidoheteroarylation of unactivated olefins has been accomplished for the first time based on the strategy of intramolecular distal heteroaryl migration. A variety of synthetically useful heteroaryl-substituted alkyl azides are readily furnished under mild reaction conditions. The utility of the protocol is manifested by readily converting the products to piperidine, β-pipecolic acid, and triazole derivatives.

Graphical abstract: Azidoheteroarylation of unactivated olefins through distal heteroaryl migration

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Publication details

The article was received on 20 Mar 2018, accepted on 27 Apr 2018 and first published on 28 Apr 2018


Article type: Research Article
DOI: 10.1039/C8QO00301G
Citation: Org. Chem. Front., 2018,5, 1896-1899
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    Azidoheteroarylation of unactivated olefins through distal heteroaryl migration

    M. Wang, Z. Wu, B. Zhang and C. Zhu, Org. Chem. Front., 2018, 5, 1896
    DOI: 10.1039/C8QO00301G

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