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The regioselective synthesis of 2-phosphinoylindoles via Rh(III)-catalyzed C–H activation

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Abstract

The redox-neutral annulation of N-nitrosoanilines with 1-alkynylphosphine oxides under rhodium catalysis was achieved. This step-economical protocol affords 2-phosphinoylindoles in excellent regioselectivity with good functional group tolerance.

Graphical abstract: The regioselective synthesis of 2-phosphinoylindoles via Rh(iii)-catalyzed C–H activation

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Publication details

The article was received on 22 Aug 2017, accepted on 21 Sep 2017 and first published on 22 Sep 2017


Article type: Research Article
DOI: 10.1039/C7QO00746A
Citation: Org. Chem. Front., 2017, Advance Article
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    The regioselective synthesis of 2-phosphinoylindoles via Rh(III)-catalyzed C–H activation

    H. Wang, S. Li, B. Wang and B. Li, Org. Chem. Front., 2017, Advance Article , DOI: 10.1039/C7QO00746A

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