Jump to main content
Jump to site search


Copper-catalyzed direct borylation of alkyl, alkenyl and aryl halides with B(dan)

Author affiliations

Abstract

Substitutional borylation of C(sp3 or sp2)–halogen bonds with an unsymmetrical diboron [(pin)B–B(dan)] was found to proceed smoothly under copper catalysis. A variety of masked alkyl-, alkenyl- and arylboron compounds [R–B(dan)] were straightforwardly accessible with high functional group compatibility in high yield.

Graphical abstract: Copper-catalyzed direct borylation of alkyl, alkenyl and aryl halides with B(dan)

Back to tab navigation
Please wait while Download options loads

Supplementary files

Publication details

The article was received on 30 Jan 2017, accepted on 10 Apr 2017 and first published on 10 Apr 2017


Article type: Research Article
DOI: 10.1039/C7QO00084G
Citation: Org. Chem. Front., 2017, Advance Article
  •   Request permissions

    Copper-catalyzed direct borylation of alkyl, alkenyl and aryl halides with B(dan)

    H. Yoshida, Y. Takemoto, S. Kamio, I. Osaka and K. Takaki, Org. Chem. Front., 2017, Advance Article , DOI: 10.1039/C7QO00084G

Search articles by author