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Issue 32, 2017
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Synthesis of 3-acylindoles by oxidative rearrangement of 2-aminochalcones using a hypervalent iodine reagent and cyclization sequence

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Abstract

An efficient one-pot method was developed for the construction of 3-acylindoles via oxidative rearrangement of 2-aminochalcones followed by intramolecular cyclization. The reaction was used to convert a variety of 2-aminochalcones into 3-acylindoles in moderate to high yields.

Graphical abstract: Synthesis of 3-acylindoles by oxidative rearrangement of 2-aminochalcones using a hypervalent iodine reagent and cyclization sequence

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Publication details

The article was received on 24 Jun 2017, accepted on 19 Jul 2017 and first published on 19 Jul 2017


Article type: Communication
DOI: 10.1039/C7OB01536D
Citation: Org. Biomol. Chem., 2017,15, 6702-6705
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    Synthesis of 3-acylindoles by oxidative rearrangement of 2-aminochalcones using a hypervalent iodine reagent and cyclization sequence

    A. Nakamura, S. Tanaka, A. Imamiya, R. Takane, C. Ohta, K. Fujimura, T. Maegawa and Y. Miki, Org. Biomol. Chem., 2017, 15, 6702
    DOI: 10.1039/C7OB01536D

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