Jump to main content
Jump to site search

Issue 67, 2017
Previous Article Next Article

One-pot borylation/Suzuki–Miyaura sp2–sp3 cross-coupling

Author affiliations

Abstract

We describe the first one-pot borylation/Suzuki–Miyaura sp2–sp3 cross-coupling between readily available aryl (pseudo)halides and activated alkyl chlorides. This method streamlines the synthesis of diaryl methanes, α-aryl carbonyls and allyl aryl compounds, substructures that are commonly found in life changing drug molecules.

Graphical abstract: One-pot borylation/Suzuki–Miyaura sp2–sp3 cross-coupling

Back to tab navigation

Supplementary files

Publication details

The article was received on 29 Jun 2017, accepted on 01 Aug 2017 and first published on 02 Aug 2017


Article type: Communication
DOI: 10.1039/C7CC05037B
Citation: Chem. Commun., 2017,53, 9364-9367
  •   Request permissions

    One-pot borylation/Suzuki–Miyaura sp2–sp3 cross-coupling

    L. Whitaker, H. Y. Harb and A. P. Pulis, Chem. Commun., 2017, 53, 9364
    DOI: 10.1039/C7CC05037B

Search articles by author

Spotlight

Advertisements